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Kras Inhibitors

Abstract: The present invention provides compounds of the formula: wherein A, B, D1, X, Y, Z, G, R1, R2, and R3a are as described herein, pharmaceutically acceptable salts thereof, and methods of using these compounds and pharmaceutically acceptable salts thereof for treating patients for cancer.

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Notices, Deadlines & Correspondence

Patent Information

Application #
Filing Date
16 September 2024
Publication Number
2/2025
Publication Type
INA
Invention Field
CHEMICAL
Status
Email
Parent Application

Applicants

ELI LILLY AND COMPANY
Lilly Corporate Center Indianapolis, Indiana 46285

Inventors

1. BARDA, David Anthony
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
2. BASTIAN, Jolie Anne
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
3. FURNESS, Kelly Wayne
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
4. GUO, Deqi
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
5. HENRY, James Robert
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
6. JOHNSTON, Richard Duane
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
7. LAMAR, Jason Eric
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
8. LIU, Tao
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
9. RODRIGUEZ, Michael John
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
10. RUBIO, Almudena
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
11. SI, Chong
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
12. ZHAO, Gaiying
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
13. ZIA-EBRAHIMI, Mohammad Sadegh
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
14. BAUMGARTNER, Matthew Patrick
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
15. ROJO, Isabel
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
16. BARBERIS, Mario
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288 Indianapolis, IN 46206-6288
17. CARBALLARES MARTIN, Santiago
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, IN 46206-6288
18. GARCIA LOSADA, Pablo
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, IN 46206-6288
19. GUTIERREZ SANFELICIANO, Sonia Maria
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, IN 46206-6288
20. LUMERAS AMADOR, Wenceslao
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, IN 46206-6288
21. MOLERO FLOREZ, Victoriano
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, IN 46206-6288
22. PRIETO VALLEJO, Maria Lourdes
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, IN 46206-6288

Specification

Documents

Application Documents

# Name Date
1 202417069852-STATEMENT OF UNDERTAKING (FORM 3) [16-09-2024(online)].pdf 2024-09-16
2 202417069852-REQUEST FOR EXAMINATION (FORM-18) [16-09-2024(online)].pdf 2024-09-16
3 202417069852-PRIORITY DOCUMENTS [16-09-2024(online)].pdf 2024-09-16
4 202417069852-POWER OF AUTHORITY [16-09-2024(online)].pdf 2024-09-16
5 202417069852-NOTIFICATION OF INT. APPLN. NO. & FILING DATE (PCT-RO-105-PCT Pamphlet) [16-09-2024(online)].pdf 2024-09-16
6 202417069852-FORM 18 [16-09-2024(online)].pdf 2024-09-16
7 202417069852-FORM 1 [16-09-2024(online)].pdf 2024-09-16
8 202417069852-DECLARATION OF INVENTORSHIP (FORM 5) [16-09-2024(online)].pdf 2024-09-16
9 202417069852-COMPLETE SPECIFICATION [16-09-2024(online)].pdf 2024-09-16
10 202417069852-CLAIMS UNDER RULE 1 (PROVISIO) OF RULE 20 [16-09-2024(online)].pdf 2024-09-16
11 202417069852-FORM 3 [16-01-2025(online)].pdf 2025-01-16
12 202417069852-Proof of Right [10-03-2025(online)].pdf 2025-03-10