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Aryl Alkynamide Derivatives
Abstract: A compound which is useful as a STING inhibitor is provided. The present inventors have found aryl alkynamide derivatives having an inhibitory action on STING. The aryl alkynamide derivatives of the present invention have an inhibitory action on STING and can be used as an agent for treating an autoimmune disease, a neurodegenerative disease, a type I interferonopathy and/or other STING-mediated disease.
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Notices, Deadlines & Correspondence
Notices, Deadlines & Correspondence
Patent Information
Application #
Filing Date
19 September 2024
Publication Number
2/2025
Publication Type
INA
Invention Field
CHEMICAL
Status
Email
Parent Application
Applicants
ASTELLAS PHARMA, INC.
5-1, Nihonbashi-honcho 2-chome
Chuo-ku
Tokyo 103-8411
ASTELLAS ENGINEERED SMALL MOLECULES US, INCORPORATED
441 Morgan Ave., Suite 700
Cambridge, MA 02141
Inventors
1. MAEDA, Junko
c/o Astellas Pharma Inc.
5-1, Nihonbashi-honcho 2-chome
Chuo-ku
Tokyo 103-8411
2. KURIWAKI, Ikumi
c/o Astellas Pharma Inc.
5-1, Nihonbashi-honcho 2-chome
Chuo-ku
Tokyo 103-8411
3. KITAMURA, Kai
c/o Astellas Pharma Inc.
5-1, Nihonbashi-honcho 2-chome
Chuo-ku
Tokyo 103-8411
4. YAMASHITA, Yumi
c/o Astellas Pharma Inc.
5-1, Nihonbashi-honcho 2-chome
Chuo-ku
Tokyo 103-8411
5. KAKEFUDA, Kenichi
c/o Astellas Pharma Inc.
5-1, Nihonbashi-honcho 2-chome
Chuo-ku
Tokyo 103-8411
6. KAMIKAWA, Akio
c/o Astellas Pharma Inc.
5-1, Nihonbashi-honcho 2-chome
Chuo-ku
Tokyo 103-8411
7. NEGORO, Kenji
c/o Astellas Pharma Inc.
5-1, Nihonbashi-honcho 2-chome
Chuo-ku
Tokyo 103-8411
8. SEO, Ryushi
c/o Astellas Pharma Inc.
5-1, Nihonbashi-honcho 2-chome
Chuo-ku
Tokyo 103-8411
9. CIAVARRI, Jeffrey
c/o Astellas Engineered Small Molecules US, Incorporated
441 Morgan Ave.
Suite 700
Cambridge, MA 02141
10. HAMAGUCHI, Wataru
c/o Astellas Pharma Inc.
5-1, Nihonbashi-honcho 2-chome
Chuo-ku
Tokyo 103-8411
Specification
Documents
Application Documents
| # | Name | Date |
|---|---|---|
| 1 | 202447070819-STATEMENT OF UNDERTAKING (FORM 3) [19-09-2024(online)].pdf | 2024-09-19 |
| 2 | 202447070819-REQUEST FOR EXAMINATION (FORM-18) [19-09-2024(online)].pdf | 2024-09-19 |
| 3 | 202447070819-PROOF OF RIGHT [19-09-2024(online)].pdf | 2024-09-19 |
| 4 | 202447070819-PRIORITY DOCUMENTS [19-09-2024(online)].pdf | 2024-09-19 |
| 5 | 202447070819-FORM 18 [19-09-2024(online)].pdf | 2024-09-19 |
| 6 | 202447070819-FORM 1 [19-09-2024(online)].pdf | 2024-09-19 |
| 7 | 202447070819-DRAWINGS [19-09-2024(online)].pdf | 2024-09-19 |
| 8 | 202447070819-DECLARATION OF INVENTORSHIP (FORM 5) [19-09-2024(online)].pdf | 2024-09-19 |
| 9 | 202447070819-COMPLETE SPECIFICATION [19-09-2024(online)].pdf | 2024-09-19 |
| 10 | 202447070819-FORM-26 [20-09-2024(online)].pdf | 2024-09-20 |
| 11 | 202447070819-FORM-26 [25-10-2024(online)].pdf | 2024-10-25 |
| 12 | 202447070819-FORM 3 [18-03-2025(online)].pdf | 2025-03-18 |