3', 3' N Bis Substituted Macrolide Lhrh Antagonists

Abstract: Disclosed are 3",3"-N-bisdesmethyl-3",3"-N-bis-substituted-6-O-methyl-11-deoxy-11,12-cyclic carbamate erythromycin A derivatives of formula (I) which are antagonists of lutenizing hormone-releasing hormone (LHRH). Also disclosed are pharmaceutical compositions comprising the compounds, methods of using the compounds and the process of making the same. Disclosed are 3",3"-N-bisdesmethyl-3",3"-N-bis-substituted-6-O-methyl-11-deoxy-11,12 -cyclic carbamate erythromycin A derivatives of formula (I) which are antagonists of lutenizing hormone-releasing hormone (LHRH). Also disclosed are pharmaceutical compositions comprising the compounds, methods of using the compounds and the process of making the same.

Patent Information

Application #

Filing Date

15 September 2000

Publication Number

02/2007

Publication Type

INA

Invention Field

PHARMACEUTICALS

Status

Email

Parent Application

Applicants

ABBOTT LABORATORIES

100 ABBOTT PARK ROAD, ABBOTT PARK, ILLINOIS 600 064-6008,

Inventors

1. SAUER DARYL R

23619 112TH STREET, TREVOR, WI 53179

Specification

Documents

Application Documents

#	Name	Date
1	in-pct-2000-00402-mum-claims(15-9-2000).pdf	2018-08-08
1	in-pct-2000-00402-mum-correspondence(ipo)-(26-10-2006).pdf	2006-10-26
2	in-pct-2000-00402-mum-correspondence(10-5-2004).pdf	2018-08-08
2	in-pct-2000-00402-mum-wo international publication report(15-9-2000).pdf	2018-08-08
3	in-pct-2000-00402-mum-correspondence(ipo)-(29-6-2010).pdf	2018-08-08
3	in-pct-2000-00402-mum-form 19(17-5-2004).pdf	2018-08-08
4	in-pct-2000-00402-mum-description(complete)-(15-9-2000).pdf	2018-08-08
5	in-pct-2000-00402-mum-correspondence(ipo)-(29-6-2010).pdf	2018-08-08
5	in-pct-2000-00402-mum-form 19(17-5-2004).pdf	2018-08-08
6	in-pct-2000-00402-mum-correspondence(10-5-2004).pdf	2018-08-08
6	in-pct-2000-00402-mum-wo international publication report(15-9-2000).pdf	2018-08-08
7	in-pct-2000-00402-mum-claims(15-9-2000).pdf	2018-08-08
7	in-pct-2000-00402-mum-correspondence(ipo)-(26-10-2006).pdf	2006-10-26