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“6 Substituted 2,3,4,5 Tetrahydro 1 H Benzo[D]Azepines As 5 Ht2 C Receptor Agonists”
Abstract: The present invention provides 6-substituted 2,3,4,5-tetrahydro-1H-benzo[d]azepines of Formula (I) as selective 5-HT2C receptor agonists for the treatment of 5-HT2C associated disorders including obesity, obsessive/compulsive disorder, depression, and anxiety: where R6 is -C=C-R10, -CH=CR11R11" , or -(C0-C8)alkyl-Ar2 optionally substituted on the alkyl moiety with 1 to 6 fluoro substituents and other substituents are as defined in the specification.
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Notices, Deadlines & Correspondence
Notices, Deadlines & Correspondence
Patent Information
Application #
Filing Date
11 March 2008
Publication Number
35/2016
Publication Type
INA
Invention Field
PHARMACEUTICALS
Status
Email
Parent Application
Applicants
ELI LILLY AND COMPANY
Lilly Corporate Center City of Indianapolis State of Indiana 46285 United States of America
Inventors
1. John Gordon ALLEN
5255 Via capote Newbury Park California 91320 United States of America
2. Karin BRINER
7649 Pinesprings East Drive Indianapolis Indiana 46256 United States of America
3. Anne Marie CAMP
Eli Lilly and Company Limited Lilly house Priestly Road Basingstoke Hampshire RG24 9NL United Kingdom
4. Manuel Javier CASES-THOMAS
Eli Lilly and Company Limited Lilly house Priestly Road Basingstoke Hampshire RG24 9NL United Kingdom
5. Richard Charles HOYING
8136 Timberwood Plainfield Indiana 46168 United States of America
6. Maria Angeles MARTINEZ-GRAU
Lilly S.A. avenida de la Industria 30 28108 Alcobendas (Madrid) Spain
7. Michael Phillip MAZANETZ
Eli Lilly and Company Limited Lilly house Priestly Road Basingstoke Hampshire RG24 9NL United Kingdom
8. Natalia POKROVSKAIA
202-335 Carnarvon Street New Westminister British Columbia V3L 1B9 Canada
9. Richard Edmund RATHMELL
Eli Lilly and Company Limited Lilly house Priestly Road Basingstoke Hampshire RG24 9NL United Kingdom
10. Roger Ryan ROTHHAAR
5282 West 775 South Reelsville Indiana 46171 United States of America
11. Selma SAPMAZ
Eli Lilly and Company Limited Lilly house Priestly Road Basingstoke Hampshire RG24 9NL United Kingdom
12. Andrew Caerwyn WILLIAMS
Eli Lilly and Company Limited Lilly house Priestly Road Basingstoke Hampshire RG24 9NL United Kingdom
Specification
The neurotransmitter serotonin (5-hydroxytryptamine, 5-HT) has a rich pharmacology arising from a heterogenous population of at least seven receptor classes. The serotonin .....
Documents
Application Documents
| # | Name | Date |
|---|---|---|
| 1 | 1039-KOLNP-2008-AbandonedLetter.pdf | 2024-06-18 |
| 1 | Form-5.pdf | 2011-10-07 |
| 2 | 1039-KOLNP-2008-FER.pdf | 2017-04-13 |
| 2 | Form-3.pdf | 2011-10-07 |
| 3 | Form-1.pdf | 2011-10-07 |
| 3 | 1039-KOLNP-2008-FORM 13.pdf | 2017-02-10 |
| 4 | 1039-KOLNP-2008-PCT REQUEST FORM.pdf | 2011-10-07 |
| 4 | 1039-KOLNP-2008-(19-02-2014)-CORRESPONDENCE.pdf | 2014-02-19 |
| 5 | 1039-KOLNP-2008-PCT PRIORITY DOCUMENT NOTIFICATION.pdf | 2011-10-07 |
| 5 | 1039-KOLNP-2008-(19-02-2014)-OTHERS.pdf | 2014-02-19 |
| 6 | 1039-KOLNP-2008-PA.pdf | 2011-10-07 |
| 6 | 1039-KOLNP-2008-(04-02-2013)-CORRESPONDENCE.pdf | 2013-02-04 |
| 7 | 1039-KOLNP-2008-INTERNATIONAL SEARCH REPORT.pdf | 2011-10-07 |
| 7 | 1039-KOLNP-2008-(04-02-2013)-OTHERS.pdf | 2013-02-04 |
| 8 | 1039-KOLNP-2008-INTERNATIONAL PUBLICATION.pdf | 2011-10-07 |
| 8 | 1039-KOLNP-2008-(26-10-2012)-CORRESPONDENCE.pdf | 2012-10-26 |
| 9 | 1039-KOLNP-2008-(26-10-2012)-FORM-1.pdf | 2012-10-26 |
| 9 | 1039-KOLNP-2008-INTERNATIONAL EXM REPORT.pdf | 2011-10-07 |
| 10 | 1039-KOLNP-2008-(21-08-2012)-CORRESPONDENCE.pdf | 2012-08-21 |
| 10 | 1039-KOLNP-2008-FORM 5-1.1.pdf | 2011-10-07 |
| 11 | 1039-KOLNP-2008-(21-08-2012)-OTHERS.pdf | 2012-08-21 |
| 11 | 1039-KOLNP-2008-FORM 3-1.1.pdf | 2011-10-07 |
| 12 | 1039-KOLNP-2008-ABSTRACT.pdf | 2011-10-07 |
| 12 | 1039-KOLNP-2008-FORM 2.pdf | 2011-10-07 |
| 13 | 1039-KOLNP-2008-ASSIGNMENT.pdf | 2011-10-07 |
| 13 | 1039-kolnp-2008-form 18.pdf | 2011-10-07 |
| 14 | 1039-KOLNP-2008-CLAIMS.pdf | 2011-10-07 |
| 14 | 1039-KOLNP-2008-FORM 1-1.1.pdf | 2011-10-07 |
| 15 | 1039-KOLNP-2008-CORRESPONDENCE OTHERS 1.2.pdf | 2011-10-07 |
| 15 | 1039-KOLNP-2008-DESCRIPTION COMPLETE.pdf | 2011-10-07 |
| 16 | 1039-KOLNP-2008-CORRESPONDENCE OTHERS-1.1.pdf | 2011-10-07 |
| 16 | 1039-KOLNP-2008-CORRESPONDENCE.pdf | 2011-10-07 |
| 17 | 1039-KOLNP-2008-CORRESPONDENCE.pdf | 2011-10-07 |
| 17 | 1039-KOLNP-2008-CORRESPONDENCE OTHERS-1.1.pdf | 2011-10-07 |
| 18 | 1039-KOLNP-2008-CORRESPONDENCE OTHERS 1.2.pdf | 2011-10-07 |
| 18 | 1039-KOLNP-2008-DESCRIPTION COMPLETE.pdf | 2011-10-07 |
| 19 | 1039-KOLNP-2008-CLAIMS.pdf | 2011-10-07 |
| 19 | 1039-KOLNP-2008-FORM 1-1.1.pdf | 2011-10-07 |
| 20 | 1039-KOLNP-2008-ASSIGNMENT.pdf | 2011-10-07 |
| 20 | 1039-kolnp-2008-form 18.pdf | 2011-10-07 |
| 21 | 1039-KOLNP-2008-ABSTRACT.pdf | 2011-10-07 |
| 21 | 1039-KOLNP-2008-FORM 2.pdf | 2011-10-07 |
| 22 | 1039-KOLNP-2008-(21-08-2012)-OTHERS.pdf | 2012-08-21 |
| 22 | 1039-KOLNP-2008-FORM 3-1.1.pdf | 2011-10-07 |
| 23 | 1039-KOLNP-2008-(21-08-2012)-CORRESPONDENCE.pdf | 2012-08-21 |
| 23 | 1039-KOLNP-2008-FORM 5-1.1.pdf | 2011-10-07 |
| 24 | 1039-KOLNP-2008-INTERNATIONAL EXM REPORT.pdf | 2011-10-07 |
| 24 | 1039-KOLNP-2008-(26-10-2012)-FORM-1.pdf | 2012-10-26 |
| 25 | 1039-KOLNP-2008-INTERNATIONAL PUBLICATION.pdf | 2011-10-07 |
| 25 | 1039-KOLNP-2008-(26-10-2012)-CORRESPONDENCE.pdf | 2012-10-26 |
| 26 | 1039-KOLNP-2008-INTERNATIONAL SEARCH REPORT.pdf | 2011-10-07 |
| 26 | 1039-KOLNP-2008-(04-02-2013)-OTHERS.pdf | 2013-02-04 |
| 27 | 1039-KOLNP-2008-PA.pdf | 2011-10-07 |
| 27 | 1039-KOLNP-2008-(04-02-2013)-CORRESPONDENCE.pdf | 2013-02-04 |
| 28 | 1039-KOLNP-2008-PCT PRIORITY DOCUMENT NOTIFICATION.pdf | 2011-10-07 |
| 28 | 1039-KOLNP-2008-(19-02-2014)-OTHERS.pdf | 2014-02-19 |
| 29 | 1039-KOLNP-2008-PCT REQUEST FORM.pdf | 2011-10-07 |
| 29 | 1039-KOLNP-2008-(19-02-2014)-CORRESPONDENCE.pdf | 2014-02-19 |
| 30 | Form-1.pdf | 2011-10-07 |
| 30 | 1039-KOLNP-2008-FORM 13.pdf | 2017-02-10 |
| 31 | 1039-KOLNP-2008-FER.pdf | 2017-04-13 |
| 31 | Form-3.pdf | 2011-10-07 |
| 32 | 1039-KOLNP-2008-AbandonedLetter.pdf | 2024-06-18 |
| 32 | Form-5.pdf | 2011-10-07 |
Search Strategy
| 1 | SEARCHREPORT_31-03-2017.pdf |