A Compound Of Formula 1 For Inhibiting The Activity Of Gpcr

A compound of formula I for inhibiting the activity of GPCR, said compound having the formula:wherein the ring may be of any configuration;Z is selected from the group consisting of: sulphur, oxygen, or NRA wherein RA is selected from the set defined for R1 to R5 or C1 to C15 acyl, C4 to C15 arylacyl or C4 to C15 heteroarylacyl, with the proviso that both R1 and RA are not hydrogen,X is selected from the group consisting of: oxygen or NRA providing that at least one X of General Formula I is NRA,R1 to R5 are independently selected from the group consisting of: H, C1 to C12 alkyl, C1 to C12 alkenyl, C1 to C12 alkynyl, C1 to C12 heteroalkyl, C4 to C15 aryl, C4 to C15 heteroaryl, C4 to C15 arylalkyl or C4 to C15 heteroarylalkyl substituent,wherein, when X is NRA, both RA and the corresponding R1 to R5 are not hydrogen.

Patent Information

Application #

Filing Date

11 May 2005

Publication Number

23/2006

Publication Type

Invention Field

BIOTECHNOLOGY

Status

Email

Parent Application

Patent Number

Legal Status

Grant Date

2008-06-11

Renewal Date

Applicants

ALCHEMIA LIMITED

3 HI-TECH COURT, BRISBANE TECHNOLOGY PARK, EIGHT MILES PLAINS, QUEENSLAND 4113

Inventors

1. MEUTERMANS, WIM

293 BIRDWOOD TERRACE, TOOWONG, QUEENSLAND 4066

2. LE THANH, GIANG

38 TARRANT STREET, MT GRAVATT, QUEENSLAND 4122

3. ABBENANTE, GIOVANNI

53 PRINGLES ROAD, SAMPSONVALE, QUEENSLAND 4520

4. TOMETZKI, GERALD

106 LHARDGREAVES ROAD, MANLY WEST, QUEENSLAND 4179

5. HALLIDAY, JUDY

9 MINNO STREET, CHAPEL HILL, QUEENSLAND 4069

6. ZEUGG, JOHANNES

43 WASSELL STREET, WYNNUM, QUEENSLAND 4178

Specification

Documents

Application Documents

#	Name	Date
1	858-KOLNP-2005-FER-[31-01-2004].pdf	2004-01-31
2	858-KOLNP-2005-LETTER OF PATENT CERTIFICATE-[11-06-2008].pdf	2008-06-11
3	858-kolnp-2005-granted-specification.pdf	2011-10-07
4	858-kolnp-2005-granted-reply to examination report.pdf	2011-10-07
5	858-kolnp-2005-granted-letter patent.pdf	2011-10-07
6	858-kolnp-2005-granted-form 5.pdf	2011-10-07
7	858-kolnp-2005-granted-form 3.pdf	2011-10-07
8	858-kolnp-2005-granted-form 26.pdf	2011-10-07
9	858-kolnp-2005-granted-form 2.pdf	2011-10-07
10	858-kolnp-2005-granted-form 18.pdf	2011-10-07
11	858-kolnp-2005-granted-form 13.pdf	2011-10-07
12	858-kolnp-2005-granted-form 1.pdf	2011-10-07
13	858-kolnp-2005-granted-examination report.pdf	2011-10-07
14	858-kolnp-2005-granted-description (complete).pdf	2011-10-07
15	858-kolnp-2005-granted-correspondence.pdf	2011-10-07
16	858-kolnp-2005-granted-claims.pdf	2011-10-07
17	858-kolnp-2005-granted-abstract.pdf	2011-10-07
18	858-kolnp-2005-21-01-2023-relevent documents.pdf	2023-01-21
19	858-KOLNP-2005-02-02-2023-Relevant Document.PDF	2023-02-02