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A Substituted Diaryl Ether As Opioid Receptor Antagonist

A compound of the formula (I) wherein the variables X1 to X10, R1 to R7 including R3', E, v, y, z, A and B are as described, or a pharmaceutically acceptable salt, solvate, enantiomer, racemate, diastereomer or mixtures thereof, useful for the treatment, prevention or amelioration of obesity and Related Diseases is disclosed.

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Notices, Deadlines & Correspondence

Patent Information

Application #
Filing Date
18 March 2005
Publication Number
09/2006
Publication Type
Invention Field
PHARMACEUTICALS
Status
Email
Parent Application
Patent Number
Legal Status
Grant Date
2008-11-19
Renewal Date

Applicants

ELI LILLY AND COMPANY
LILLY CORPORATE CENTER, INDIANAPOLIS, INDIANA

Inventors

1. BLANCO-PILLADO
7278 NORTH HAWTHORNE LANE, INDIANAPOLIS, IN 46250
2. CHAPPELL, MARK, DONALD
541 PITNEY DRIVE, NOBLESVILLE, IN 46060
3. DE LA TORRE, MARTA, GARCIA
LILLY, S.A. AVDA. INDUSTRIA, 30, 28108 ALCOBENDAS-MADRID
4. DIAZ BUEZO, NURIA
LILLY, S.A. AVDA. INDUSTRIA, 30, 28108 ALCOBENDAS-MADRID
5. FRITZ, JAMES, ERWIN
9757 NORTH MOONSTONE PLACE, MCCORDSVILLE, IN 46055
6. HOLLOWAY, WILLIAM, GLEN
9590 EAST 600 SOUTH, ZIONSVILLE, IN 46077
7. MATT, JAMES, EDWARD, JUNIOR
11436 HARLEQUIN LANE, APARTMENT 413, FISHER, IN 46038
8. MITCH, CHARLES, HOWARD
3210 GROVE PARKWAY, COLUMBUS, IN 47203
9. PEDREGAL-TERCERO, CONCEPCION
LILLY, S.A. AVDA. INDUSTRIA, 30, 28108 ALCOBENDAS-MADRID
10. QUIMBY, STEVEN, JAMES
10657 KESTREL COURT, NOBELSVILLE, IN 46060
11. SIEGEL, MILES, GOODMAN
1708 WEST 74TH PLACE, INDIANAPOLIS, IN 46260
12. SMITH, DANA, RAE
13287 BECKWITH DRIVE, WESTFIELD, IN 46074
13. STUCKY, RUSSELL, DEAN
6045 BARTH AVENUE, INDIANAPOLIS, IN 46227
14. TAKEUCHI, KUMIKO
6342 ROBINSROCK DRIVE, INDIANAPOLIS, IN 46268
15. THOMAS, ELIZABETH, MARIE
4133 SANDPIPER LANE, COLUMBUS, IN 47203
16. WOLFE, CHAD, NOLAN
16096 TENOR WAY, NOBLESVILLE, IN 46060

Specification

Documents

Application Documents

# Name Date
1 457-KOLNP-2005-FORM-27 [29-10-2024(online)].pdf 2024-10-29
1 457-KOLNP-2005-PA.pdf 2011-10-06
2 457-KOLNP-2005-Form-4 u-r 131 [16-10-2024(online)].pdf 2024-10-16
2 457-kolnp-2005-granted-specification.pdf 2011-10-06
3 457-kolnp-2005-granted-reply to examination report.pdf 2011-10-06
3 457-KOLNP-2005-08-02-2023-LETTER OF PATENT, PETITION.pdf 2023-02-08
4 457-kolnp-2005-granted-form 5.pdf 2011-10-06
4 457-KOLNP-2005-02-02-2023-RELEVANT DOCUMENTS.pdf 2023-02-02
5 457-KOLNP-2005-RELEVANT DOCUMENTS [17-11-2021(online)].pdf 2021-11-17
5 457-kolnp-2005-granted-form 3.pdf 2011-10-06
6 457-KOLNP-2005-RELEVANT DOCUMENTS [24-03-2020(online)].pdf 2020-03-24
6 457-kolnp-2005-granted-form 26.pdf 2011-10-06
7 457-kolnp-2005-granted-form 2.pdf 2011-10-06
7 457-KOLNP-2005-Annexure [17-02-2020(online)].pdf 2020-02-17
8 457-KOLNP-2005-Response to office action [17-02-2020(online)].pdf 2020-02-17
8 457-kolnp-2005-granted-form 18.pdf 2011-10-06
9 457-kolnp-2005-granted-form 13.pdf 2011-10-06
9 457-KOLNP-2005-RELEVANT DOCUMENTS [27-01-2020(online)].pdf 2020-01-27
10 457-kolnp-2005-granted-form 1.pdf 2011-10-06
10 457-KOLNP-2005-RELEVANT DOCUMENTS [24-01-2019(online)].pdf 2019-01-24
11 457-KOLNP-2005-ASSIGNMENT WITH VERIFIED COPY [10-01-2019(online)].pdf 2019-01-10
11 457-kolnp-2005-granted-examination report.pdf 2011-10-06
12 457-KOLNP-2005-FORM-16 [10-01-2019(online)].pdf 2019-01-10
12 457-kolnp-2005-granted-description (complete).pdf 2011-10-06
13 457-kolnp-2005-granted-correspondence.pdf 2011-10-06
13 457-KOLNP-2005-POWER OF AUTHORITY [10-01-2019(online)].pdf 2019-01-10
14 457-kolnp-2005-granted-claims.pdf 2011-10-06
14 457-KOLNP-2005-RELEVANT DOCUMENTS [08-03-2018(online)].pdf 2018-03-08
15 457-kolnp-2005-granted-abstract.pdf 2011-10-06
15 Form 27 [02-02-2017(online)].pdf 2017-02-02
16 457-KOLNP-2005-FORM 27.pdf 2011-10-06
16 Form 27 [16-02-2016(online)].pdf 2016-02-16
17 ipindiaonline.gov.in_epatentfiling_online_frmPreview.asp.pdf 2015-03-20
17 457-KOLNP-2005-CORRESPONDENCE.pdf 2011-10-06
18 457-KOLNP-2005-(18-03-2015)-FORM-27.pdf 2015-03-18
18 457-KOLNP-2005-CORRESPONDENCE 1.1.pdf 2011-10-06
19 457-KOLNP-2005-(29-03-2012)-FORM-27.pdf 2012-03-29
19 Form 27.pdf 2014-04-02
20 457-KOLNP-2005-(17-03-2014)-FORM-27.pdf 2014-03-17
20 457-KOLNP-2005-(29-03-2012)-CORRESPONDENCE.pdf 2012-03-29
21 457-KOLNP-2005-(18-11-2013)-CORRESPONDENCE.pdf 2013-11-18
21 457-KOLNP-2005-(25-03-2013)-FORM-27.pdf 2013-03-25
22 457-KOLNP-2005-(18-11-2013)-OTHERS.pdf 2013-11-18
22 457-KOLNP-2005-(30-04-2013)-PA.pdf 2013-04-30
23 457-KOLNP-2005-(23-08-2013)-CORRESPONDENCE.pdf 2013-08-23
23 457-KOLNP-2005-(30-04-2013)-OTHERS.pdf 2013-04-30
24 457-KOLNP-2005-(30-04-2013)-FORM 16.pdf 2013-04-30
24 457-KOLNP-2005-(23-08-2013)-OTHERS.pdf 2013-08-23
25 457-KOLNP-2005-(30-04-2013)-CORRESPONDENCE.pdf 2013-04-30
26 457-KOLNP-2005-(23-08-2013)-OTHERS.pdf 2013-08-23
26 457-KOLNP-2005-(30-04-2013)-FORM 16.pdf 2013-04-30
27 457-KOLNP-2005-(23-08-2013)-CORRESPONDENCE.pdf 2013-08-23
27 457-KOLNP-2005-(30-04-2013)-OTHERS.pdf 2013-04-30
28 457-KOLNP-2005-(18-11-2013)-OTHERS.pdf 2013-11-18
28 457-KOLNP-2005-(30-04-2013)-PA.pdf 2013-04-30
29 457-KOLNP-2005-(18-11-2013)-CORRESPONDENCE.pdf 2013-11-18
29 457-KOLNP-2005-(25-03-2013)-FORM-27.pdf 2013-03-25
30 457-KOLNP-2005-(17-03-2014)-FORM-27.pdf 2014-03-17
30 457-KOLNP-2005-(29-03-2012)-CORRESPONDENCE.pdf 2012-03-29
31 457-KOLNP-2005-(29-03-2012)-FORM-27.pdf 2012-03-29
31 Form 27.pdf 2014-04-02
32 457-KOLNP-2005-(18-03-2015)-FORM-27.pdf 2015-03-18
32 457-KOLNP-2005-CORRESPONDENCE 1.1.pdf 2011-10-06
33 457-KOLNP-2005-CORRESPONDENCE.pdf 2011-10-06
33 ipindiaonline.gov.in_epatentfiling_online_frmPreview.asp.pdf 2015-03-20
34 457-KOLNP-2005-FORM 27.pdf 2011-10-06
34 Form 27 [16-02-2016(online)].pdf 2016-02-16
35 Form 27 [02-02-2017(online)].pdf 2017-02-02
35 457-kolnp-2005-granted-abstract.pdf 2011-10-06
36 457-KOLNP-2005-RELEVANT DOCUMENTS [08-03-2018(online)].pdf 2018-03-08
36 457-kolnp-2005-granted-claims.pdf 2011-10-06
37 457-kolnp-2005-granted-correspondence.pdf 2011-10-06
37 457-KOLNP-2005-POWER OF AUTHORITY [10-01-2019(online)].pdf 2019-01-10
38 457-KOLNP-2005-FORM-16 [10-01-2019(online)].pdf 2019-01-10
38 457-kolnp-2005-granted-description (complete).pdf 2011-10-06
39 457-KOLNP-2005-ASSIGNMENT WITH VERIFIED COPY [10-01-2019(online)].pdf 2019-01-10
39 457-kolnp-2005-granted-examination report.pdf 2011-10-06
40 457-kolnp-2005-granted-form 1.pdf 2011-10-06
40 457-KOLNP-2005-RELEVANT DOCUMENTS [24-01-2019(online)].pdf 2019-01-24
41 457-kolnp-2005-granted-form 13.pdf 2011-10-06
41 457-KOLNP-2005-RELEVANT DOCUMENTS [27-01-2020(online)].pdf 2020-01-27
42 457-kolnp-2005-granted-form 18.pdf 2011-10-06
42 457-KOLNP-2005-Response to office action [17-02-2020(online)].pdf 2020-02-17
43 457-KOLNP-2005-Annexure [17-02-2020(online)].pdf 2020-02-17
43 457-kolnp-2005-granted-form 2.pdf 2011-10-06
44 457-kolnp-2005-granted-form 26.pdf 2011-10-06
44 457-KOLNP-2005-RELEVANT DOCUMENTS [24-03-2020(online)].pdf 2020-03-24
45 457-kolnp-2005-granted-form 3.pdf 2011-10-06
45 457-KOLNP-2005-RELEVANT DOCUMENTS [17-11-2021(online)].pdf 2021-11-17
46 457-kolnp-2005-granted-form 5.pdf 2011-10-06
46 457-KOLNP-2005-02-02-2023-RELEVANT DOCUMENTS.pdf 2023-02-02
47 457-kolnp-2005-granted-reply to examination report.pdf 2011-10-06
47 457-KOLNP-2005-08-02-2023-LETTER OF PATENT, PETITION.pdf 2023-02-08
48 457-kolnp-2005-granted-specification.pdf 2011-10-06
48 457-KOLNP-2005-Form-4 u-r 131 [16-10-2024(online)].pdf 2024-10-16
49 457-KOLNP-2005-PA.pdf 2011-10-06
49 457-KOLNP-2005-FORM-27 [29-10-2024(online)].pdf 2024-10-29

ERegister / Renewals

3rd: 30 Jan 2009

From 17/09/2005 - To 17/09/2006

4th: 30 Jan 2009

From 17/09/2006 - To 17/09/2007

5th: 30 Jan 2009

From 17/09/2007 - To 17/09/2008

6th: 30 Jan 2009

From 17/09/2008 - To 17/09/2009

7th: 13 Jul 2009

From 17/09/2009 - To 17/09/2010

8th: 23 Aug 2010

From 17/09/2010 - To 17/09/2011

9th: 09 Sep 2011

From 17/09/2011 - To 17/09/2012

10th: 05 Sep 2012

From 17/09/2012 - To 17/09/2013

11th: 10 Sep 2013

From 17/09/2013 - To 17/09/2014

12th: 12 Sep 2014

From 17/09/2014 - To 17/09/2015

13th: 13 Jul 2015

From 17/09/2015 - To 17/09/2016

14th: 08 Jul 2016

From 17/09/2016 - To 17/09/2017

15th: 18 Aug 2017

From 17/09/2017 - To 17/09/2018

16th: 17 Jul 2018

From 17/09/2018 - To 17/09/2019

17th: 30 Jul 2019

From 17/09/2019 - To 17/09/2020

18th: 26 Aug 2020

From 17/09/2020 - To 17/09/2021

19th: 10 Sep 2021

From 17/09/2021 - To 17/09/2022

20th: 15 Sep 2022

From 17/09/2022 - To 17/09/2023