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Benzothiophene Compound

Abstract: The inventors perfected the present invention as a result of a study into IK1 channel activators and a confirmation that a benzothiophene compound exhibits efficacy against visceral pain inflammatory pain osteoarthritic pain neuropathic pain or fibromyalgia. This compound represented by formula (I) has IK1 channel activating action and may be used as a drug to prevent or treat visceral pain inflammatory pain osteoarthritic pain neuropathic pain fibromyalgia or the like. The IK1 channel activator may be used as a drug to prevent or treat inflammatory pain osteoarthritic pain neuropathic pain or fibromyalgia.

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Notices, Deadlines & Correspondence

Patent Information

Application #
Filing Date
30 December 2015
Publication Number
36/2016
Publication Type
INA
Invention Field
CHEMICAL
Status
Email
patent@depenning.com
Parent Application
Patent Number
Legal Status
Grant Date
2020-02-26
Renewal Date

Applicants

ASTELLAS PHARMA INC.
5-1, Nihonbashi-Honcho 2-chome, Chuo-ku, Tokyo 103-8411

Inventors

1. ISHIHARA, Tsukasa
c/o Astellas Pharma Inc., 5-1, Nihonbashi-Honcho 2- chome, Chuo-ku, Tokyo 103-8411,
2. IKEGAI, Kazuhiro
c/o Astellas Pharma Inc., 5-1, Nihonbashi-Honcho 2- chome, Chuo-ku, Tokyo 103-8411,
3. KURIWAKI, Ikumi
c/o Astellas Pharma Inc., 5-1, Nihonbashi-Honcho 2- chome, Chuo-ku, Tokyo 103-8411,
4. HISAMICHI, Hiroyuki
c/o Astellas Pharma Inc., 5-1, Nihonbashi-Honcho 2- chome, Chuo-ku, Tokyo 103-8411,
5. TAKESHITA, Nobuaki
c/o Astellas Pharma Inc., 5-1, Nihonbashi-Honcho 2- chome, Chuo-ku, Tokyo 103-8411,
6. TAKEZAWA, Ryuichi
c/o Astellas Pharma Inc., 5-1, Nihonbashi-Honcho 2- chome, Chuo-ku, Tokyo 103-8411,

Specification

SOFT COPY ATTACHED IN PDF

Documents

Application Documents

# Name Date
1 Power of Attorney [30-12-2015(online)].pdf 2015-12-30
2 Form 5 [30-12-2015(online)].pdf 2015-12-30
3 Form 3 [30-12-2015(online)].pdf 2015-12-30
4 Form 1 [30-12-2015(online)].pdf 2015-12-30
5 Description(Complete) [30-12-2015(online)].pdf 2015-12-30
6 8055-CHENP-2015.pdf 2016-01-01
7 Form 3 [27-05-2016(online)].pdf 2016-05-27
8 8055-CHENP-2015-Form 1-290116.pdf 2016-06-28
9 8055-CHENP-2015-Correspondence-Form 1-290116.pdf 2016-06-28
10 Other Document [23-03-2017(online)].pdf 2017-03-23
11 Marked Copy [23-03-2017(online)].pdf 2017-03-23
12 Form 18 [23-03-2017(online)].pdf 2017-03-23
13 Form 13 [23-03-2017(online)].pdf 2017-03-23
14 Description(Complete) [23-03-2017(online)].pdf_138.pdf 2017-03-23
15 Description(Complete) [23-03-2017(online)].pdf 2017-03-23
16 Form 3 [20-06-2017(online)].pdf 2017-06-20
17 8055-CHENP-2015-FER.pdf 2019-04-01
18 8055-CHENP-2015-certified copy of translation (MANDATORY) [15-04-2019(online)].pdf 2019-04-15
19 8055-CHENP-2015-PETITION UNDER RULE 137 [03-09-2019(online)].pdf 2019-09-03
20 8055-CHENP-2015-OTHERS [03-09-2019(online)].pdf 2019-09-03
21 8055-CHENP-2015-FORM 3 [03-09-2019(online)].pdf 2019-09-03
22 8055-CHENP-2015-FER_SER_REPLY [03-09-2019(online)].pdf 2019-09-03
23 8055-CHENP-2015-CLAIMS [03-09-2019(online)].pdf 2019-09-03
24 8055-CHENP-2015-certified copy of translation (MANDATORY) [03-09-2019(online)].pdf 2019-09-03
25 8055-CHENP-2015-ABSTRACT [03-09-2019(online)].pdf 2019-09-03
26 8055-CHENP-2015_Marked Up Claims_Granted_332991_26-02-2020.pdf 2020-02-26
27 8055-CHENP-2015_Description_Granted_332991_26-02-2020.pdf 2020-02-26
28 8055-CHENP-2015_Claims_Granted_332991_26-02-2020.pdf 2020-02-26
29 8055-CHENP-2015_Abstract_Granted_332991_26-02-2020.pdf 2020-02-26
30 8055-CHENP-2015-PatentCertificate26-02-2020.pdf 2020-02-26
31 8055-CHENP-2015-IntimationOfGrant26-02-2020.pdf 2020-02-26
32 8055-CHENP-2015-RELEVANT DOCUMENTS [24-04-2020(online)].pdf 2020-04-24
33 8055-CHENP-2015-MARKED COPIES OF AMENDEMENTS [24-04-2020(online)].pdf 2020-04-24
34 8055-CHENP-2015-FORM 13 [24-04-2020(online)].pdf 2020-04-24
35 8055-CHENP-2015-AMENDED DOCUMENTS [24-04-2020(online)].pdf 2020-04-24
36 8055-CHENP-2015-RELEVANT DOCUMENTS [10-08-2021(online)].pdf 2021-08-10
37 8055-CHENP-2015-RELEVANT DOCUMENTS [28-09-2022(online)].pdf 2022-09-28
38 8055-CHENP-2015-RELEVANT DOCUMENTS [21-09-2023(online)].pdf 2023-09-21

Search Strategy

1 8055search_19-03-2019.pdf

ERegister / Renewals

3rd: 15 May 2020

From 06/06/2016 - To 06/06/2017

4th: 15 May 2020

From 06/06/2017 - To 06/06/2018

5th: 15 May 2020

From 06/06/2018 - To 06/06/2019

6th: 15 May 2020

From 06/06/2019 - To 06/06/2020

7th: 15 May 2020

From 06/06/2020 - To 06/06/2021

8th: 01 May 2021

From 06/06/2021 - To 06/06/2022

9th: 11 May 2022

From 06/06/2022 - To 06/06/2023

10th: 30 May 2023

From 06/06/2023 - To 06/06/2024