Abstract: The object of the present invention is benzothiazine derivatives having the capability of inhibiting 11ß-HSD1 not only at an enzymatic level but also at a cell level. The compounds of the present invention are of general formula (I). Wherein notably R1 represents a hydrogen or OR1 represents an ester or an ether. R2 represents a naphthyl or a 1, 2, 3, 4-tetrahydro-naphthalene or a biphenyl or phenyl pyridine or a substituted phenyl. R3 represents a methyl or ethyl; R4 and R'4 represent a hydrogen.
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| # | Name | Date |
|---|---|---|
| 1 | 7244-delnp-2011-GPA-(10-10-2011).pdf | 2011-10-10 |
| 1 | 7244-DELNP-2011-RELEVANT DOCUMENTS [09-03-2020(online)].pdf | 2020-03-09 |
| 2 | 7244-delnp-2011-Correspondence Others-(10-10-2011).pdf | 2011-10-10 |
| 2 | 7244-DELNP-2011-RELEVANT DOCUMENTS [20-02-2019(online)].pdf | 2019-02-20 |
| 3 | 7244-DELNP-2011-IntimationOfGrant24-04-2018.pdf | 2018-04-24 |
| 3 | 7244-delnp-2011-Correspondence Others-(20-04-2012).pdf | 2012-04-20 |
| 4 | Abstract.jpg | 2012-04-30 |
| 4 | 7244-DELNP-2011-PatentCertificate24-04-2018.pdf | 2018-04-24 |
| 5 | 7244-DELNP-2011-PETITION UNDER RULE 137 [19-04-2018(online)].pdf | 2018-04-19 |
| 5 | 7244-delnp-2011-Form-5.pdf | 2012-04-30 |
| 6 | 7244-delnp-2011-Response to office action (Mandatory) [19-04-2018(online)].pdf | 2018-04-19 |
| 6 | 7244-delnp-2011-Form-3.pdf | 2012-04-30 |
| 7 | 7244-delnp-2011-Form-2.pdf | 2012-04-30 |
| 7 | 7244-delnp-2011-2. Marked Copy under Rule 14(2) (MANDATORY) [26-12-2017(online)].pdf | 2017-12-26 |
| 8 | 7244-delnp-2011-Form-1.pdf | 2012-04-30 |
| 8 | 7244-delnp-2011-CLAIMS [26-12-2017(online)].pdf | 2017-12-26 |
| 9 | 7244-delnp-2011-Description (Complete).pdf | 2012-04-30 |
| 9 | 7244-delnp-2011-FER_SER_REPLY [26-12-2017(online)].pdf | 2017-12-26 |
| 10 | 7244-delnp-2011-Correspondence-others.pdf | 2012-04-30 |
| 10 | 7244-delnp-2011-OTHERS [26-12-2017(online)].pdf | 2017-12-26 |
| 11 | 7244-delnp-2011-Claims.pdf | 2012-04-30 |
| 11 | 7244-DELNP-2011-PETITION UNDER RULE 137 [26-12-2017(online)].pdf | 2017-12-26 |
| 12 | 7244-delnp-2011-Abstract.pdf | 2012-04-30 |
| 12 | 7244-delnp-2011-Retyped Pages under Rule 14(1) (MANDATORY) [26-12-2017(online)].pdf | 2017-12-26 |
| 13 | 7244-DELNP-2011-Correspondence-201117.pdf | 2017-12-07 |
| 13 | 7244-delnp-2011-Form-18-(06-02-2013).pdf | 2013-02-06 |
| 14 | 7244-delnp-2011-Correspondence Others-(06-02-2013).pdf | 2013-02-06 |
| 14 | 7244-DELNP-2011-Others-201117.pdf | 2017-12-07 |
| 15 | 7244-delnp-2011-Correspondence Others-(24-09-2013).pdf | 2013-09-24 |
| 15 | 7244-DELNP-2011-Proof of Right (MANDATORY) [16-11-2017(online)].pdf | 2017-11-16 |
| 16 | 7244-DELNP-2011-FER.pdf | 2017-06-27 |
| 16 | 7244-DELNP-2011-FORM 3 [23-10-2017(online)].pdf | 2017-10-23 |
| 17 | 7244-DELNP-2011-Information under section 8(2) (MANDATORY) [23-10-2017(online)].pdf | 2017-10-23 |
| 17 | 7244-DELNP-2011-DUPLICATE-FER-06-30-2017.pdf | 2017-06-30 |
| 18 | 7244-DELNP-2011-DUPLICATE-FER-06-30-2017.pdf | 2017-06-30 |
| 18 | 7244-DELNP-2011-Information under section 8(2) (MANDATORY) [23-10-2017(online)].pdf | 2017-10-23 |
| 19 | 7244-DELNP-2011-FER.pdf | 2017-06-27 |
| 19 | 7244-DELNP-2011-FORM 3 [23-10-2017(online)].pdf | 2017-10-23 |
| 20 | 7244-delnp-2011-Correspondence Others-(24-09-2013).pdf | 2013-09-24 |
| 20 | 7244-DELNP-2011-Proof of Right (MANDATORY) [16-11-2017(online)].pdf | 2017-11-16 |
| 21 | 7244-delnp-2011-Correspondence Others-(06-02-2013).pdf | 2013-02-06 |
| 21 | 7244-DELNP-2011-Others-201117.pdf | 2017-12-07 |
| 22 | 7244-DELNP-2011-Correspondence-201117.pdf | 2017-12-07 |
| 22 | 7244-delnp-2011-Form-18-(06-02-2013).pdf | 2013-02-06 |
| 23 | 7244-delnp-2011-Abstract.pdf | 2012-04-30 |
| 23 | 7244-delnp-2011-Retyped Pages under Rule 14(1) (MANDATORY) [26-12-2017(online)].pdf | 2017-12-26 |
| 24 | 7244-DELNP-2011-PETITION UNDER RULE 137 [26-12-2017(online)].pdf | 2017-12-26 |
| 24 | 7244-delnp-2011-Claims.pdf | 2012-04-30 |
| 25 | 7244-delnp-2011-Correspondence-others.pdf | 2012-04-30 |
| 25 | 7244-delnp-2011-OTHERS [26-12-2017(online)].pdf | 2017-12-26 |
| 26 | 7244-delnp-2011-Description (Complete).pdf | 2012-04-30 |
| 26 | 7244-delnp-2011-FER_SER_REPLY [26-12-2017(online)].pdf | 2017-12-26 |
| 27 | 7244-delnp-2011-CLAIMS [26-12-2017(online)].pdf | 2017-12-26 |
| 27 | 7244-delnp-2011-Form-1.pdf | 2012-04-30 |
| 28 | 7244-delnp-2011-2. Marked Copy under Rule 14(2) (MANDATORY) [26-12-2017(online)].pdf | 2017-12-26 |
| 28 | 7244-delnp-2011-Form-2.pdf | 2012-04-30 |
| 29 | 7244-delnp-2011-Form-3.pdf | 2012-04-30 |
| 29 | 7244-delnp-2011-Response to office action (Mandatory) [19-04-2018(online)].pdf | 2018-04-19 |
| 30 | 7244-delnp-2011-Form-5.pdf | 2012-04-30 |
| 30 | 7244-DELNP-2011-PETITION UNDER RULE 137 [19-04-2018(online)].pdf | 2018-04-19 |
| 31 | Abstract.jpg | 2012-04-30 |
| 31 | 7244-DELNP-2011-PatentCertificate24-04-2018.pdf | 2018-04-24 |
| 32 | 7244-DELNP-2011-IntimationOfGrant24-04-2018.pdf | 2018-04-24 |
| 32 | 7244-delnp-2011-Correspondence Others-(20-04-2012).pdf | 2012-04-20 |
| 33 | 7244-DELNP-2011-RELEVANT DOCUMENTS [20-02-2019(online)].pdf | 2019-02-20 |
| 33 | 7244-delnp-2011-Correspondence Others-(10-10-2011).pdf | 2011-10-10 |
| 34 | 7244-DELNP-2011-RELEVANT DOCUMENTS [09-03-2020(online)].pdf | 2020-03-09 |
| 34 | 7244-delnp-2011-GPA-(10-10-2011).pdf | 2011-10-10 |
| 1 | 7244delnp2011searchstrategy1_23-06-2017.pdf |