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Fgfr2 Inhibitor Compounds

Abstract: The present invention provides compounds of the formula (I):, or a pharmaceutically acceptable salt thereof, wherein A, X1, X2, X3, Y, Z, Z1, Z2, R2 and R6 are as defined herein, for use in the treatment of cancer and a method of treating cancer.

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Notices, Deadlines & Correspondence

Patent Information

Application #
Filing Date
23 October 2024
Publication Number
51/2024
Publication Type
INA
Invention Field
CHEMICAL
Status
Email
Parent Application

Applicants

ELI LILLY AND COMPANY
Lilly Corporate Center Indianapolis, Indiana 46285

Inventors

1. ADEVA BARTOLOMÉ, Marta
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
2. FERNANDEZ FIGUEROA, Maria Carmen
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
3. DEL PRADO CATALINA, Miriam Filadelfa
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
4. GARCIA-CERRADA, Susana Maria
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
5. GARCIA LOSADA, Pablo
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
6. GARZÓN SANZ, Miguel
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
7. GUTIERREZ SANFELICIANO, Sonia Maria
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
8. MARTINEZ PEREZ, Jose Antonio
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
9. METCALF, Andrew Terrance
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
10. PEIRÓ CADAHIA, Jorge
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
11. VALERO DE LA CRUZ, Alberto
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288
12. PRIETO VALLEJO, Maria Lourdes
c/o ELI LILLY AND COMPANY P.O. Box 6288 Indianapolis, Indiana 46206-6288

Specification

Documents

Application Documents

# Name Date
1 202417080526-STATEMENT OF UNDERTAKING (FORM 3) [23-10-2024(online)].pdf 2024-10-23
2 202417080526-PRIORITY DOCUMENTS [23-10-2024(online)].pdf 2024-10-23
3 202417080526-POWER OF AUTHORITY [23-10-2024(online)].pdf 2024-10-23
4 202417080526-NOTIFICATION OF INT. APPLN. NO. & FILING DATE (PCT-RO-105-PCT Pamphlet) [23-10-2024(online)].pdf 2024-10-23
5 202417080526-MARKED COPIES OF AMENDEMENTS [23-10-2024(online)].pdf 2024-10-23
6 202417080526-FORM 18 [23-10-2024(online)].pdf 2024-10-23
7 202417080526-FORM 13 [23-10-2024(online)].pdf 2024-10-23
8 202417080526-FORM 1 [23-10-2024(online)].pdf 2024-10-23
9 202417080526-FIGURE OF ABSTRACT [23-10-2024(online)].pdf 2024-10-23
10 202417080526-DECLARATION OF INVENTORSHIP (FORM 5) [23-10-2024(online)].pdf 2024-10-23
11 202417080526-COMPLETE SPECIFICATION [23-10-2024(online)].pdf 2024-10-23
12 202417080526-CLAIMS UNDER RULE 1 (PROVISIO) OF RULE 20 [23-10-2024(online)].pdf 2024-10-23
13 202417080526-AMMENDED DOCUMENTS [23-10-2024(online)].pdf 2024-10-23
14 202417080526-Proof of Right [14-04-2025(online)].pdf 2025-04-14
15 202417080526-FORM 3 [15-04-2025(online)].pdf 2025-04-15