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Fused Compounds That Inhibit Vanilloid Receptor Subtype 1 (Vr1) Receptor

Abstract: The present invention discloses novel compounds of general formula (I), or a pharmaceutically acceptable salt or prodrug thereof (in which X1 - X5, R5 - R8b, Z1 - Z2 and Ar1 are defined herein), a method for inhibiting the VR1 receptor in mammals using these compounds, a method for controlling pain in mammals, and pharmaceutical compositions including those compounds and a process for making those compounds.

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Notices, Deadlines & Correspondence

Patent Information

Application #
Filing Date
09 January 2006
Publication Number
26/2007
Publication Type
INA
Invention Field
PHARMACEUTICALS
Status
Email
Parent Application
Patent Number
Legal Status
Grant Date
2009-03-16
Renewal Date

Applicants

ABBOTT LABORATORIES
Dept. 377 AP6A-1, 100 Abbott Park Road, Abbott Park, Illinois 60064-6008.

Inventors

1. GOMTSYAN, ARTHUR
104 Adair Court, Vernon Hills, Illinois 60061.
2. BAYBURT, EROL
17462 Chestnut, Gurnee, Illinois 60031.
3. KOENIG, JOHN
1618 W. Edgewater Avenue, Unit 3 East, Chicago, Illinois 60060.
4. SCHMIDT, ROBERT
2001 W Eagle Ridge Drive, Waukegan, Illinois 60087.
5. LUKIN, KIRILL
158 E. Colonial Drive, Vernon Hills, Illinois 60061.
6. CHAMBOURNIER GILLES
29549 N. Waukegan Road, LAKE BLUFF, Illinois 60044.
7. HSU, MARGARET
321 Southfield Drive, VERNON HILLS, Illinois 60061.
8. LEANNA, ROBERT
1025 Pope's Creek Circle, Grayslake, Illinois 60030.
9. CINK, RUSSEL
1447 Fairport Drive, Grayslake, Illinois 60030.
10. LEE, CHIH-HUNG
569 S. CENTRAL PARK PLACE, VERNON HILLS, ILLINOIS 60061,

Specification

N/A

Documents

Application Documents

# Name Date
1 34-MUMNP-2006-ABSTRACT(AMENDED)-(5-12-2007).pdf 2018-08-09
1 34-MUMNP-2006-CORRESPONDENCE(RENEWAL PAYMENT LETTER)-(08-06-2011).pdf 2011-06-08
2 34-MUMNP-2006-ANNEXURE(5-12-2007).pdf 2018-08-09
2 34-MUMNP-2006-CORRESPONDENCE(RENEWAL PAYMENT LETTER)-(05-06-2013).pdf 2013-06-05
3 34-MUMNP-2006-WO INTERNATIONAL PUBLICATION REPORT(9-1-2006).pdf 2018-08-09
3 34-MUMNP-2006-ASSIGNMENT(1-12-2007).pdf 2018-08-09
4 34-MUMNP-2006-SPECIFICATION(AMENDED)-(5-12-2007).pdf 2018-08-09
4 34-MUMNP-2006-ASSIGNMENT(14-8-2013).pdf 2018-08-09
5 34-MUMNP-2006-PETITION UNDER RULE 137(3-12-2007).pdf 2018-08-09
5 34-MUMNP-2006-CANCELLED PAGES(5-12-2007).pdf 2018-08-09
6 34-MUMNP-2006-GENERAL POWER OF ATTORNEY(14-8-2013).pdf 2018-08-09
6 34-MUMNP-2006-CLAIMS(23-1-2009).pdf 2018-08-09
7 34-MUMNP-2006-GENERAL POWER OF ATTORNEY(1-12-2007).pdf 2018-08-09
7 34-MUMNP-2006-CLAIMS(9-1-2006).pdf 2018-08-09
8 34-MUMNP-2006-FORM 5(6-12-2007).pdf 2018-08-09
8 34-MUMNP-2006-CLAIMS(AMENDED)-(23-2-2009).pdf 2018-08-09
9 34-mumnp-2006-claims(granted)-(16-3-2009).pdf 2018-08-09
9 34-MUMNP-2006-FORM 5(5-12-2007).pdf 2018-08-09
10 34-MUMNP-2006-COPY OF EP(23-1-2009).pdf 2018-08-09
10 34-MUMNP-2006-FORM 3(6-12-2007).pdf 2018-08-09
11 34-MUMNP-2006-CORRESPONDENCE 1(17-6-2009).pdf 2018-08-09
11 34-MUMNP-2006-FORM 3(5-12-2007).pdf 2018-08-09
12 34-MUMNP-2006-CORRESPONDENCE(14-8-2013).pdf 2018-08-09
12 34-MUMNP-2006-FORM 26(1-12-2007).pdf 2018-08-09
13 34-MUMNP-2006-CORRESPONDENCE(23-2-2009).pdf 2018-08-09
13 34-mumnp-2006-form 2(title page)-(granted)-(16-3-2009).pdf 2018-08-09
14 34-MUMNP-2006-CORRESPONDENCE(27-1-2009).pdf 2018-08-09
14 34-MUMNP-2006-FORM 2(TITLE PAGE)-(9-1-2006).pdf 2018-08-09
15 34-MUMNP-2006-CORRESPONDENCE(4-1-2006).pdf 2018-08-09
15 34-mumnp-2006-form 2(granted)-(16-3-2009).pdf 2018-08-09
16 34-MUMNP-2006-CORRESPONDENCE(IPO)-(27-8-2009).pdf 2018-08-09
16 34-MUMNP-2006-FORM 2(COMPLETE)-(9-1-2006).pdf 2018-08-09
17 34-MUMNP-2006-FORM 18(9-1-2006).pdf 2018-08-09
17 34-MUMNP-2006-DESCRIPTION(COMPLETE)-(9-1-2006).pdf 2018-08-09
18 34-mumnp-2006-description(granted)-(16-3-2009).pdf 2018-08-09
18 34-MUMNP-2006-FORM 16(14-8-2013).pdf 2018-08-09
19 34-MUMNP-2006-DRAWING(23-1-2009).pdf 2018-08-09
19 34-MUMNP-2006-FORM 13(3-12-2007).pdf 2018-08-09
20 34-MUMNP-2006-DRAWING(23-2-2009).pdf 2018-08-09
20 34-MUMNP-2006-FORM 13(29-5-2007).pdf 2018-08-09
21 34-MUMNP-2006-DRAWING(9-1-2006).pdf 2018-08-09
21 34-MUMNP-2006-FORM 1(9-1-2006).pdf 2018-08-09
22 34-MUMNP-2006-DRAWING(AMENDED)-(23-1-2009).pdf 2018-08-09
22 34-MUMNP-2006-FORM 1(5-12-2007).pdf 2018-08-09
23 34-MUMNP-2006-DRAWING(AMENDED)-(5-12-2007).pdf 2018-08-09
23 34-MUMNP-2006-E P PATENT(23-2-2009).pdf 2018-08-09
24 34-mumnp-2006-drawing(granted)-(16-3-2009).pdf 2018-08-09
25 34-MUMNP-2006-E P PATENT(23-2-2009).pdf 2018-08-09
25 34-MUMNP-2006-DRAWING(AMENDED)-(5-12-2007).pdf 2018-08-09
26 34-MUMNP-2006-DRAWING(AMENDED)-(23-1-2009).pdf 2018-08-09
26 34-MUMNP-2006-FORM 1(5-12-2007).pdf 2018-08-09
27 34-MUMNP-2006-DRAWING(9-1-2006).pdf 2018-08-09
27 34-MUMNP-2006-FORM 1(9-1-2006).pdf 2018-08-09
28 34-MUMNP-2006-DRAWING(23-2-2009).pdf 2018-08-09
28 34-MUMNP-2006-FORM 13(29-5-2007).pdf 2018-08-09
29 34-MUMNP-2006-DRAWING(23-1-2009).pdf 2018-08-09
29 34-MUMNP-2006-FORM 13(3-12-2007).pdf 2018-08-09
30 34-mumnp-2006-description(granted)-(16-3-2009).pdf 2018-08-09
30 34-MUMNP-2006-FORM 16(14-8-2013).pdf 2018-08-09
31 34-MUMNP-2006-DESCRIPTION(COMPLETE)-(9-1-2006).pdf 2018-08-09
31 34-MUMNP-2006-FORM 18(9-1-2006).pdf 2018-08-09
32 34-MUMNP-2006-CORRESPONDENCE(IPO)-(27-8-2009).pdf 2018-08-09
32 34-MUMNP-2006-FORM 2(COMPLETE)-(9-1-2006).pdf 2018-08-09
33 34-MUMNP-2006-CORRESPONDENCE(4-1-2006).pdf 2018-08-09
33 34-mumnp-2006-form 2(granted)-(16-3-2009).pdf 2018-08-09
34 34-MUMNP-2006-CORRESPONDENCE(27-1-2009).pdf 2018-08-09
34 34-MUMNP-2006-FORM 2(TITLE PAGE)-(9-1-2006).pdf 2018-08-09
35 34-MUMNP-2006-CORRESPONDENCE(23-2-2009).pdf 2018-08-09
35 34-mumnp-2006-form 2(title page)-(granted)-(16-3-2009).pdf 2018-08-09
36 34-MUMNP-2006-FORM 26(1-12-2007).pdf 2018-08-09
36 34-MUMNP-2006-CORRESPONDENCE(14-8-2013).pdf 2018-08-09
37 34-MUMNP-2006-CORRESPONDENCE 1(17-6-2009).pdf 2018-08-09
37 34-MUMNP-2006-FORM 3(5-12-2007).pdf 2018-08-09
38 34-MUMNP-2006-COPY OF EP(23-1-2009).pdf 2018-08-09
38 34-MUMNP-2006-FORM 3(6-12-2007).pdf 2018-08-09
39 34-mumnp-2006-claims(granted)-(16-3-2009).pdf 2018-08-09
39 34-MUMNP-2006-FORM 5(5-12-2007).pdf 2018-08-09
40 34-MUMNP-2006-CLAIMS(AMENDED)-(23-2-2009).pdf 2018-08-09
40 34-MUMNP-2006-FORM 5(6-12-2007).pdf 2018-08-09
41 34-MUMNP-2006-CLAIMS(9-1-2006).pdf 2018-08-09
41 34-MUMNP-2006-GENERAL POWER OF ATTORNEY(1-12-2007).pdf 2018-08-09
42 34-MUMNP-2006-GENERAL POWER OF ATTORNEY(14-8-2013).pdf 2018-08-09
42 34-MUMNP-2006-CLAIMS(23-1-2009).pdf 2018-08-09
43 34-MUMNP-2006-PETITION UNDER RULE 137(3-12-2007).pdf 2018-08-09
43 34-MUMNP-2006-CANCELLED PAGES(5-12-2007).pdf 2018-08-09
44 34-MUMNP-2006-SPECIFICATION(AMENDED)-(5-12-2007).pdf 2018-08-09
44 34-MUMNP-2006-ASSIGNMENT(14-8-2013).pdf 2018-08-09
45 34-MUMNP-2006-WO INTERNATIONAL PUBLICATION REPORT(9-1-2006).pdf 2018-08-09
45 34-MUMNP-2006-ASSIGNMENT(1-12-2007).pdf 2018-08-09
46 34-MUMNP-2006-CORRESPONDENCE(RENEWAL PAYMENT LETTER)-(05-06-2013).pdf 2013-06-05
46 34-MUMNP-2006-ANNEXURE(5-12-2007).pdf 2018-08-09
47 34-MUMNP-2006-ABSTRACT(AMENDED)-(5-12-2007).pdf 2018-08-09
47 34-MUMNP-2006-CORRESPONDENCE(RENEWAL PAYMENT LETTER)-(08-06-2011).pdf 2011-06-08

ERegister / Renewals

3rd: 10 Jun 2009

From 10/06/2007 - To 10/06/2008

4th: 10 Jun 2009

From 10/06/2008 - To 10/06/2009

5th: 10 Jun 2009

From 10/06/2009 - To 10/06/2010

6th: 10 Jun 2009

From 10/06/2010 - To 10/06/2011

7th: 01 Jun 2010

From 10/06/2011 - To 10/06/2012

8th: 08 Jun 2011

From 10/06/2012 - To 10/06/2013

9th: 05 Jun 2013

From 10/06/2013 - To 10/06/2014

10th: 05 Jun 2013

From 10/06/2014 - To 10/06/2015