Abstract: The present invention discloses novel compounds of general formula (I), or a pharmaceutically acceptable salt or prodrug thereof (in which X1 - X5, R5 - R8b, Z1 - Z2 and Ar1 are defined herein), a method for inhibiting the VR1 receptor in mammals using these compounds, a method for controlling pain in mammals, and pharmaceutical compositions including those compounds and a process for making those compounds.
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| # | Name | Date |
|---|---|---|
| 1 | 34-MUMNP-2006-ABSTRACT(AMENDED)-(5-12-2007).pdf | 2018-08-09 |
| 1 | 34-MUMNP-2006-CORRESPONDENCE(RENEWAL PAYMENT LETTER)-(08-06-2011).pdf | 2011-06-08 |
| 2 | 34-MUMNP-2006-ANNEXURE(5-12-2007).pdf | 2018-08-09 |
| 2 | 34-MUMNP-2006-CORRESPONDENCE(RENEWAL PAYMENT LETTER)-(05-06-2013).pdf | 2013-06-05 |
| 3 | 34-MUMNP-2006-WO INTERNATIONAL PUBLICATION REPORT(9-1-2006).pdf | 2018-08-09 |
| 3 | 34-MUMNP-2006-ASSIGNMENT(1-12-2007).pdf | 2018-08-09 |
| 4 | 34-MUMNP-2006-SPECIFICATION(AMENDED)-(5-12-2007).pdf | 2018-08-09 |
| 4 | 34-MUMNP-2006-ASSIGNMENT(14-8-2013).pdf | 2018-08-09 |
| 5 | 34-MUMNP-2006-PETITION UNDER RULE 137(3-12-2007).pdf | 2018-08-09 |
| 5 | 34-MUMNP-2006-CANCELLED PAGES(5-12-2007).pdf | 2018-08-09 |
| 6 | 34-MUMNP-2006-GENERAL POWER OF ATTORNEY(14-8-2013).pdf | 2018-08-09 |
| 6 | 34-MUMNP-2006-CLAIMS(23-1-2009).pdf | 2018-08-09 |
| 7 | 34-MUMNP-2006-GENERAL POWER OF ATTORNEY(1-12-2007).pdf | 2018-08-09 |
| 7 | 34-MUMNP-2006-CLAIMS(9-1-2006).pdf | 2018-08-09 |
| 8 | 34-MUMNP-2006-FORM 5(6-12-2007).pdf | 2018-08-09 |
| 8 | 34-MUMNP-2006-CLAIMS(AMENDED)-(23-2-2009).pdf | 2018-08-09 |
| 9 | 34-mumnp-2006-claims(granted)-(16-3-2009).pdf | 2018-08-09 |
| 9 | 34-MUMNP-2006-FORM 5(5-12-2007).pdf | 2018-08-09 |
| 10 | 34-MUMNP-2006-COPY OF EP(23-1-2009).pdf | 2018-08-09 |
| 10 | 34-MUMNP-2006-FORM 3(6-12-2007).pdf | 2018-08-09 |
| 11 | 34-MUMNP-2006-CORRESPONDENCE 1(17-6-2009).pdf | 2018-08-09 |
| 11 | 34-MUMNP-2006-FORM 3(5-12-2007).pdf | 2018-08-09 |
| 12 | 34-MUMNP-2006-CORRESPONDENCE(14-8-2013).pdf | 2018-08-09 |
| 12 | 34-MUMNP-2006-FORM 26(1-12-2007).pdf | 2018-08-09 |
| 13 | 34-MUMNP-2006-CORRESPONDENCE(23-2-2009).pdf | 2018-08-09 |
| 13 | 34-mumnp-2006-form 2(title page)-(granted)-(16-3-2009).pdf | 2018-08-09 |
| 14 | 34-MUMNP-2006-CORRESPONDENCE(27-1-2009).pdf | 2018-08-09 |
| 14 | 34-MUMNP-2006-FORM 2(TITLE PAGE)-(9-1-2006).pdf | 2018-08-09 |
| 15 | 34-MUMNP-2006-CORRESPONDENCE(4-1-2006).pdf | 2018-08-09 |
| 15 | 34-mumnp-2006-form 2(granted)-(16-3-2009).pdf | 2018-08-09 |
| 16 | 34-MUMNP-2006-CORRESPONDENCE(IPO)-(27-8-2009).pdf | 2018-08-09 |
| 16 | 34-MUMNP-2006-FORM 2(COMPLETE)-(9-1-2006).pdf | 2018-08-09 |
| 17 | 34-MUMNP-2006-FORM 18(9-1-2006).pdf | 2018-08-09 |
| 17 | 34-MUMNP-2006-DESCRIPTION(COMPLETE)-(9-1-2006).pdf | 2018-08-09 |
| 18 | 34-mumnp-2006-description(granted)-(16-3-2009).pdf | 2018-08-09 |
| 18 | 34-MUMNP-2006-FORM 16(14-8-2013).pdf | 2018-08-09 |
| 19 | 34-MUMNP-2006-DRAWING(23-1-2009).pdf | 2018-08-09 |
| 19 | 34-MUMNP-2006-FORM 13(3-12-2007).pdf | 2018-08-09 |
| 20 | 34-MUMNP-2006-DRAWING(23-2-2009).pdf | 2018-08-09 |
| 20 | 34-MUMNP-2006-FORM 13(29-5-2007).pdf | 2018-08-09 |
| 21 | 34-MUMNP-2006-DRAWING(9-1-2006).pdf | 2018-08-09 |
| 21 | 34-MUMNP-2006-FORM 1(9-1-2006).pdf | 2018-08-09 |
| 22 | 34-MUMNP-2006-DRAWING(AMENDED)-(23-1-2009).pdf | 2018-08-09 |
| 22 | 34-MUMNP-2006-FORM 1(5-12-2007).pdf | 2018-08-09 |
| 23 | 34-MUMNP-2006-DRAWING(AMENDED)-(5-12-2007).pdf | 2018-08-09 |
| 23 | 34-MUMNP-2006-E P PATENT(23-2-2009).pdf | 2018-08-09 |
| 24 | 34-mumnp-2006-drawing(granted)-(16-3-2009).pdf | 2018-08-09 |
| 25 | 34-MUMNP-2006-E P PATENT(23-2-2009).pdf | 2018-08-09 |
| 25 | 34-MUMNP-2006-DRAWING(AMENDED)-(5-12-2007).pdf | 2018-08-09 |
| 26 | 34-MUMNP-2006-DRAWING(AMENDED)-(23-1-2009).pdf | 2018-08-09 |
| 26 | 34-MUMNP-2006-FORM 1(5-12-2007).pdf | 2018-08-09 |
| 27 | 34-MUMNP-2006-DRAWING(9-1-2006).pdf | 2018-08-09 |
| 27 | 34-MUMNP-2006-FORM 1(9-1-2006).pdf | 2018-08-09 |
| 28 | 34-MUMNP-2006-DRAWING(23-2-2009).pdf | 2018-08-09 |
| 28 | 34-MUMNP-2006-FORM 13(29-5-2007).pdf | 2018-08-09 |
| 29 | 34-MUMNP-2006-DRAWING(23-1-2009).pdf | 2018-08-09 |
| 29 | 34-MUMNP-2006-FORM 13(3-12-2007).pdf | 2018-08-09 |
| 30 | 34-mumnp-2006-description(granted)-(16-3-2009).pdf | 2018-08-09 |
| 30 | 34-MUMNP-2006-FORM 16(14-8-2013).pdf | 2018-08-09 |
| 31 | 34-MUMNP-2006-DESCRIPTION(COMPLETE)-(9-1-2006).pdf | 2018-08-09 |
| 31 | 34-MUMNP-2006-FORM 18(9-1-2006).pdf | 2018-08-09 |
| 32 | 34-MUMNP-2006-CORRESPONDENCE(IPO)-(27-8-2009).pdf | 2018-08-09 |
| 32 | 34-MUMNP-2006-FORM 2(COMPLETE)-(9-1-2006).pdf | 2018-08-09 |
| 33 | 34-MUMNP-2006-CORRESPONDENCE(4-1-2006).pdf | 2018-08-09 |
| 33 | 34-mumnp-2006-form 2(granted)-(16-3-2009).pdf | 2018-08-09 |
| 34 | 34-MUMNP-2006-CORRESPONDENCE(27-1-2009).pdf | 2018-08-09 |
| 34 | 34-MUMNP-2006-FORM 2(TITLE PAGE)-(9-1-2006).pdf | 2018-08-09 |
| 35 | 34-MUMNP-2006-CORRESPONDENCE(23-2-2009).pdf | 2018-08-09 |
| 35 | 34-mumnp-2006-form 2(title page)-(granted)-(16-3-2009).pdf | 2018-08-09 |
| 36 | 34-MUMNP-2006-FORM 26(1-12-2007).pdf | 2018-08-09 |
| 36 | 34-MUMNP-2006-CORRESPONDENCE(14-8-2013).pdf | 2018-08-09 |
| 37 | 34-MUMNP-2006-CORRESPONDENCE 1(17-6-2009).pdf | 2018-08-09 |
| 37 | 34-MUMNP-2006-FORM 3(5-12-2007).pdf | 2018-08-09 |
| 38 | 34-MUMNP-2006-COPY OF EP(23-1-2009).pdf | 2018-08-09 |
| 38 | 34-MUMNP-2006-FORM 3(6-12-2007).pdf | 2018-08-09 |
| 39 | 34-mumnp-2006-claims(granted)-(16-3-2009).pdf | 2018-08-09 |
| 39 | 34-MUMNP-2006-FORM 5(5-12-2007).pdf | 2018-08-09 |
| 40 | 34-MUMNP-2006-CLAIMS(AMENDED)-(23-2-2009).pdf | 2018-08-09 |
| 40 | 34-MUMNP-2006-FORM 5(6-12-2007).pdf | 2018-08-09 |
| 41 | 34-MUMNP-2006-CLAIMS(9-1-2006).pdf | 2018-08-09 |
| 41 | 34-MUMNP-2006-GENERAL POWER OF ATTORNEY(1-12-2007).pdf | 2018-08-09 |
| 42 | 34-MUMNP-2006-GENERAL POWER OF ATTORNEY(14-8-2013).pdf | 2018-08-09 |
| 42 | 34-MUMNP-2006-CLAIMS(23-1-2009).pdf | 2018-08-09 |
| 43 | 34-MUMNP-2006-PETITION UNDER RULE 137(3-12-2007).pdf | 2018-08-09 |
| 43 | 34-MUMNP-2006-CANCELLED PAGES(5-12-2007).pdf | 2018-08-09 |
| 44 | 34-MUMNP-2006-SPECIFICATION(AMENDED)-(5-12-2007).pdf | 2018-08-09 |
| 44 | 34-MUMNP-2006-ASSIGNMENT(14-8-2013).pdf | 2018-08-09 |
| 45 | 34-MUMNP-2006-WO INTERNATIONAL PUBLICATION REPORT(9-1-2006).pdf | 2018-08-09 |
| 45 | 34-MUMNP-2006-ASSIGNMENT(1-12-2007).pdf | 2018-08-09 |
| 46 | 34-MUMNP-2006-CORRESPONDENCE(RENEWAL PAYMENT LETTER)-(05-06-2013).pdf | 2013-06-05 |
| 46 | 34-MUMNP-2006-ANNEXURE(5-12-2007).pdf | 2018-08-09 |
| 47 | 34-MUMNP-2006-ABSTRACT(AMENDED)-(5-12-2007).pdf | 2018-08-09 |
| 47 | 34-MUMNP-2006-CORRESPONDENCE(RENEWAL PAYMENT LETTER)-(08-06-2011).pdf | 2011-06-08 |