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Glycine Compound
Abstract: The present invention provides a compound which is useful as an active ingredient of a pharmaceutical composition, in particular, a pharmaceutical composition for preventing and/or treating VAP-1-related diseases. [Means for Solution] The present inventors have conducted intensive studies on a compound having a VAP-1 inhibitory activity, and as a result, they have found that a compound of the present invention or a salt thereof exhibits an excellent VAP-1 inhibitory activity and is useful for preventing and/or treating VAP-1-related diseases, in particular, diabetic nephropathy or diabetic macular edema, thereby completing the present invention. The present invention further relates to a pharmaceutical composition, in particular, a pharmaceutical composition for preventing and/or treating VAP-1-related diseases, which comprises the compound of the present invention or a salt thereof, and an excipient. [Selected Figure] Nil
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Notices, Deadlines & Correspondence
Notices, Deadlines & Correspondence
Patent Information
Application #
Filing Date
16 March 2012
Publication Number
22/2013
Publication Type
INA
Invention Field
CHEMICAL
Status
Email
patent@depenning.com
Parent Application
Applicants
ASTELLAS PHARMA INC.
3-11, NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO-103-8411
Inventors
1. YOSHIHARA, KOUSEI
C/O ASTELLAS PHARMA INC., 3-11, NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411
2. SUZUKI, DAISUKE
C/O ASTELLAS PHARMA INC., 3-11, NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411
3. YAMAKI, SUSUMU
C/O ASTELLAS PHARMA INC., 3-11, NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411
4. KOGA, YUJI
C/O ASTELLAS PHARMA INC., 3-11, NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411
5. SEKI, NORIO
C/O ASTELLAS PHARMA INC., 3-11, NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411
6. FUJIYASU, JIRO
C/O ASTELLAS PHARMA INC., 3-11, NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411
Specification
Documents
Application Documents
| # | Name | Date |
|---|---|---|
| 1 | 2472-CHENP-2012 POWER OF ATTORNEY 16-03-2012.pdf | 2012-03-16 |
| 1 | 2472-CHENP-2012-AbandonedLetter.pdf | 2018-06-22 |
| 2 | 2472-CHENP-2012 FORM-2 16-03-2012.pdf | 2012-03-16 |
| 2 | 2472-CHENP-2012-FER.pdf | 2017-12-12 |
| 3 | 2472-CHENP-2012 DESCRIPTION(COMPLETE)-3 16-03-2012.pdf | 2012-03-16 |
| 3 | 2472-CHENP-2012 CORRESPONDENCE OTHERS 08-09-2014.pdf | 2014-09-08 |
| 4 | 2472-CHENP-2012 FORM-3 08-09-2014.pdf | 2014-09-08 |
| 4 | 2472-CHENP-2012 DESCRIPTION(COMPLETE)-2 16-03-2012.pdf | 2012-03-16 |
| 5 | 2472-CHENP-2012 DESCRIPTION(COMPLETE)-1 16-03-2012.pdf | 2012-03-16 |
| 5 | 2472-CHENP-2012 FORM-13 06-09-2013.pdf | 2013-09-06 |
| 6 | 2472-CHENP-2012 DESCRIPTION(COMPLETE) 16-03-2012.pdf | 2012-03-16 |
| 6 | 2472-CHENP-2012 AMENDED CLAIMS 06-09-2013.pdf | 2013-09-06 |
| 7 | 2472-CHENP-2012 CLAIMS 16-03-2012.pdf | 2012-03-16 |
| 7 | 2472-CHENP-2012 AMENDED PAGES OF SPECIFICATION 06-09-2013.pdf | 2013-09-06 |
| 8 | 2472-CHENP-2012 CORRESPONDENCE OTHERS 06-09-2013.pdf | 2013-09-06 |
| 8 | 2472-CHENP-2012 ABSTRACT 16-03-2012.pdf | 2012-03-16 |
| 9 | 2472-CHENP-2012 PCT 16-03-2012..pdf | 2012-03-16 |
| 9 | 2472-CHENP-2012 FORM-18 06-09-2013.pdf | 2013-09-06 |
| 10 | 2472-CHENP-2012 FORM-5 16-03-2012..pdf | 2012-03-16 |
| 10 | 2472-CHENP-2012 CORRESPONDENCE OTHERS 19-06-2013.pdf | 2013-06-19 |
| 11 | 2472-CHENP-2012 CORRESPONDENCE OTHERS 12-09-2012.pdf | 2012-09-12 |
| 11 | 2472-CHENP-2012 FORM-3 16-03-2012..pdf | 2012-03-16 |
| 12 | 2472-CHENP-2012 FORM-1 16-03-2012..pdf | 2012-03-16 |
| 12 | 2472-CHENP-2012 FORM-3 12-09-2012.pdf | 2012-09-12 |
| 13 | 2472-CHENP-2012 CORRESPONDENCE OTHERS 16-03-2012..pdf | 2012-03-16 |
| 13 | 2472-CHENP-2012 AMENDED CLAIMS 29-06-2012.pdf | 2012-06-29 |
| 14 | 2472-CHENP-2012 FORM-13 29-06-2012.pdf | 2012-06-29 |
| 14 | 2472-CHENP-2012 FORM-5 08-05-2012..pdf | 2012-05-08 |
| 15 | 2472-CHENP-2012 CORRESPONDENCE OTHERS 29-06-2012.pdf | 2012-06-29 |
| 15 | 2472-CHENP-2012 FORM-13 08-05-2012.pdf | 2012-05-08 |
| 16 | 2472-CHENP-2012 ENGLISH TRANSLATION 27-06-2012.pdf | 2012-06-27 |
| 16 | 2472-CHENP-2012 FORM-1 08-05-2012..pdf | 2012-05-08 |
| 17 | 2472-CHENP-2012 CORRESPONDENCE OTHERS 08-05-2012..pdf | 2012-05-08 |
| 17 | 2472-CHENP-2012 CORRESPONDENCE OTHERS 27-06-2012.pdf | 2012-06-27 |
| 18 | 2472-CHENP-2012 FORM-13 27-06-2012.pdf | 2012-06-27 |
| 19 | 2472-CHENP-2012 CORRESPONDENCE OTHERS 27-06-2012.pdf | 2012-06-27 |
| 19 | 2472-CHENP-2012 CORRESPONDENCE OTHERS 08-05-2012..pdf | 2012-05-08 |
| 20 | 2472-CHENP-2012 ENGLISH TRANSLATION 27-06-2012.pdf | 2012-06-27 |
| 20 | 2472-CHENP-2012 FORM-1 08-05-2012..pdf | 2012-05-08 |
| 21 | 2472-CHENP-2012 CORRESPONDENCE OTHERS 29-06-2012.pdf | 2012-06-29 |
| 21 | 2472-CHENP-2012 FORM-13 08-05-2012.pdf | 2012-05-08 |
| 22 | 2472-CHENP-2012 FORM-13 29-06-2012.pdf | 2012-06-29 |
| 22 | 2472-CHENP-2012 FORM-5 08-05-2012..pdf | 2012-05-08 |
| 23 | 2472-CHENP-2012 CORRESPONDENCE OTHERS 16-03-2012..pdf | 2012-03-16 |
| 23 | 2472-CHENP-2012 AMENDED CLAIMS 29-06-2012.pdf | 2012-06-29 |
| 24 | 2472-CHENP-2012 FORM-3 12-09-2012.pdf | 2012-09-12 |
| 24 | 2472-CHENP-2012 FORM-1 16-03-2012..pdf | 2012-03-16 |
| 25 | 2472-CHENP-2012 CORRESPONDENCE OTHERS 12-09-2012.pdf | 2012-09-12 |
| 25 | 2472-CHENP-2012 FORM-3 16-03-2012..pdf | 2012-03-16 |
| 26 | 2472-CHENP-2012 FORM-5 16-03-2012..pdf | 2012-03-16 |
| 26 | 2472-CHENP-2012 CORRESPONDENCE OTHERS 19-06-2013.pdf | 2013-06-19 |
| 27 | 2472-CHENP-2012 PCT 16-03-2012..pdf | 2012-03-16 |
| 27 | 2472-CHENP-2012 FORM-18 06-09-2013.pdf | 2013-09-06 |
| 28 | 2472-CHENP-2012 ABSTRACT 16-03-2012.pdf | 2012-03-16 |
| 28 | 2472-CHENP-2012 CORRESPONDENCE OTHERS 06-09-2013.pdf | 2013-09-06 |
| 29 | 2472-CHENP-2012 AMENDED PAGES OF SPECIFICATION 06-09-2013.pdf | 2013-09-06 |
| 29 | 2472-CHENP-2012 CLAIMS 16-03-2012.pdf | 2012-03-16 |
| 30 | 2472-CHENP-2012 AMENDED CLAIMS 06-09-2013.pdf | 2013-09-06 |
| 30 | 2472-CHENP-2012 DESCRIPTION(COMPLETE) 16-03-2012.pdf | 2012-03-16 |
| 31 | 2472-CHENP-2012 DESCRIPTION(COMPLETE)-1 16-03-2012.pdf | 2012-03-16 |
| 31 | 2472-CHENP-2012 FORM-13 06-09-2013.pdf | 2013-09-06 |
| 32 | 2472-CHENP-2012 FORM-3 08-09-2014.pdf | 2014-09-08 |
| 32 | 2472-CHENP-2012 DESCRIPTION(COMPLETE)-2 16-03-2012.pdf | 2012-03-16 |
| 33 | 2472-CHENP-2012 DESCRIPTION(COMPLETE)-3 16-03-2012.pdf | 2012-03-16 |
| 33 | 2472-CHENP-2012 CORRESPONDENCE OTHERS 08-09-2014.pdf | 2014-09-08 |
| 34 | 2472-CHENP-2012-FER.pdf | 2017-12-12 |
| 34 | 2472-CHENP-2012 FORM-2 16-03-2012.pdf | 2012-03-16 |
| 35 | 2472-CHENP-2012-AbandonedLetter.pdf | 2018-06-22 |
| 35 | 2472-CHENP-2012 POWER OF ATTORNEY 16-03-2012.pdf | 2012-03-16 |
Search Strategy
| 1 | 2472_CHENP_2012_14-11-2017.pdf |