Heterocyclic Compounds As Cbp/Ep300 Bromodomain Inhibitors

Abstract: The present invention provides heterocyclic compounds of formula (I), which are therapeutically useful as CBP/EP300 inhibitors. These compounds are useful in the treatment and/or prevention of diseases or disorders mediated by CBP and/or EP300 in an individual. The present invention also provides preparation of the compounds and pharmaceutical compositions comprising at least one of the compounds of formula (I) or a pharmaceutically acceptable salt, or a stereoisomer or a tautomer, an N-oxide or an ester thereof.

Patent Information

Application #

Filing Date

07 April 2023

Publication Number

18/2023

Publication Type

INA

Invention Field

CHEMICAL

Status

Email

Parent Application

Applicants

AURIGENE ONCOLOGY LIMITED

39-40, KIADB Industrial Area Electronic City Phase II Hosur Road Bangalore 560100

Inventors

1. ABBINENI, Chandrasekhar

H. No: 15-21-48/14/G-3, Sri Sai Datta Enclave Balaji Nagar, Kukatpally, Telangana. Hyderabad 500 072

2. SAMAJDAR, Susanta

Flat # R801, H. M Tambourine, Jaraganahalli, J.P. Nagar 6th Phase Bangalore 560 078

3. S. SENAIAR, Ramesh

Nambi SUBBIAH 8, Kiran building, Nareen Nagar Society Station Road Thakurli East Dist: Thane (Mumbai) Mumbai 421201

4. AGGUNDA RENUKAPPA, Girish

#63, S/O Renukappa, Henchin Depo main road Behind Mini vidhana Saudha, Arasikere, Karnataka Bangalore 573103

5. MUKHERJEE, Subhendu

132/A/3, Thakurbari Street (Kokil Bagan), P.O. Serampore, HOOGHLY 712201

6. TATYASAHEB GORE, Suraj

Nandur Bk, Taluka: Rahata, Dist: Ahmednagar Maharashtra 413720

7. WOHLFAHRT, Gerd

Vattuniemenkatu 14 C 35,Helsinki Finland, FI-00210 00210 Helsinki

8. MYLLYMAKI, Mikko

C/O Orion corporation, ESPOO, Finland, FI-02200 02200 Espoo

Specification

Documents

Application Documents

#	Name	Date
1	202347026201.pdf	2023-04-07
2	202347026201-STATEMENT OF UNDERTAKING (FORM 3) [07-04-2023(online)].pdf	2023-04-07
3	202347026201-FORM 1 [07-04-2023(online)].pdf	2023-04-07
4	202347026201-DECLARATION OF INVENTORSHIP (FORM 5) [07-04-2023(online)].pdf	2023-04-07
5	202347026201-COMPLETE SPECIFICATION [07-04-2023(online)].pdf	2023-04-07
6	202347026201-CLAIMS UNDER RULE 1 (PROVISIO) OF RULE 20 [07-04-2023(online)].pdf	2023-04-07
7	202347026201-Proof of Right [07-10-2023(online)].pdf	2023-10-07
8	202347026201-PETITION UNDER RULE 137 [08-12-2023(online)].pdf	2023-12-08
9	202347026201-FORM 3 [08-12-2023(online)].pdf	2023-12-08
10	202347026201-FORM 18 [05-09-2024(online)].pdf	2024-09-05