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Pyrido [4,3 D] Pyrimidine Derivatives As Mek Inhibitors

Abstract: The present disclosure is related to heteroaryl compounds as MEK inhibitors. These compounds include heteroaryl compounds of Formula (I) their pharmaceutically acceptable salts combinations with suitable medicament and pharmaceutical compositions thereof. The present disclosure also includes processes of preparation of the compounds and their use in methods of treatment. The compounds as disclosed herein are of Formula (I) below:

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Notices, Deadlines & Correspondence

Patent Information

Application #
Filing Date
01 September 2014
Publication Number
27/2015
Publication Type
INA
Invention Field
CHEMICAL
Status
Email
Parent Application
Patent Number
Legal Status
Grant Date
2021-02-04
Renewal Date

Applicants

LUPIN LIMITED
159 CST Road Kalina Santacruz (East)State of Maharashtra Mumbai 400 098 India

Inventors

1. DAVE Bhavesh
Lupin Limited (Research Park) 46A / 47A Nande Village Mulshi Taluka Pune 412 115
2. BANERJEE Rakesh Kumar
Lupin Limited (Research Park) 46A / 47A Nande Village Mulshi Taluka Pune 412 115
3. PHUKAN Samiron
Lupin Limited (Research Park) 46A / 47A Nande Village Mulshi Taluka Pune 412 115
4. KHOJE Abhijit Datta
Lupin Limited (Research Park) 46A / 47A Nande Village Mulshi Taluka Pune 412 115
5. HANGARGE Rajkumar
Lupin Limited (Research Park) 46A / 47A Nande Village Mulshi Taluka Pune 412 115
6. JADHAV Jitendra Sambhaji
Lupin Limited (Research Park) 46A / 47A Nande Village Mulshi Taluka Pune 412 115
7. PALLE Venkata P.
Lupin Limited (Research Park) 46A / 47A Nande Village Mulshi Taluka Pune 412 115
8. KAMBOJ Rajender Kumar
Lupin Limited (Research Park) 46A / 47A Nande Village Mulshi Taluka Pune 412 115

Specification

Documents

Application Documents

# Name Date
1 1755-MUMNP-2014-FORM 1(26-09-2014).pdf 2014-09-26
1 1755-MUMNP-2014-RELEVANT DOCUMENTS [01-09-2023(online)].pdf 2023-09-01
2 1755-MUMNP-2014-CORRESPONDENCE(26-09-2014).pdf 2014-09-26
2 1755-MUMNP-2014-RELEVANT DOCUMENTS [21-09-2022(online)]-1.pdf 2022-09-21
3 1755-MUMNP-2014-RELEVANT DOCUMENTS [21-09-2022(online)].pdf 2022-09-21
3 1755-MUMNP-2014-CORRESPONDENCE(21-10-2014).pdf 2014-10-21
4 1755-MUMNP-2014-US(14)-ExtendedHearingNotice-(HearingDate-08-10-2020).pdf 2021-10-03
4 1755-MUMNP-2014-ANNEXURE TO FORM 3E(21-10-2014).pdf 2014-10-21
5 1755-MUMNP-2014-RELEVANT DOCUMENTS [25-09-2021(online)]-1.pdf 2021-09-25
5 1755-MUMNP-2014-CORRESPONDENCE-05-03-2015.pdf 2015-03-05
6 1755-MUMNP-2014-RELEVANT DOCUMENTS [25-09-2021(online)].pdf 2021-09-25
6 1755-MUMNP-2014-ANNEXURE TO FORM-05-03-2015.pdf 2015-03-05
7 1755-MUMNP-2014-IntimationOfGrant04-02-2021.pdf 2021-02-04
7 1755-MUMNP-2014-ANNEXURE TO FORM 3-05-03-2015.pdf 2015-03-05
8 Other Document [24-08-2016(online)].pdf 2016-08-24
8 1755-MUMNP-2014-PatentCertificate04-02-2021.pdf 2021-02-04
9 1755-MUMNP-2014-FORM 3 [26-11-2020(online)].pdf 2020-11-26
9 Form 13 [24-08-2016(online)].pdf 2016-08-24
10 1755-MUMNP-2014-PETITION UNDER RULE 137 [22-10-2020(online)].pdf 2020-10-22
10 Other Patent Document [27-02-2017(online)].pdf 2017-02-27
11 1755-MUMNP-2014-Written submissions and relevant documents [22-10-2020(online)].pdf 2020-10-22
11 Other Patent Document [09-05-2017(online)].pdf 2017-05-09
12 1755-MUMNP-2014-FORM 3 [04-12-2017(online)].pdf 2017-12-04
12 1755-MUMNP-2014-FORM 3 [09-10-2020(online)].pdf 2020-10-09
13 1755-MUMNP-2014-FORM 3 [23-03-2018(online)].pdf 2018-03-23
13 1755-MUMNP-2014-Information under section 8(2) [09-10-2020(online)].pdf 2020-10-09
14 1755-MUMNP-2014-FORM 3 [11-04-2018(online)].pdf 2018-04-11
14 1755-MUMNP-2014-US(14)-HearingNotice-(HearingDate-08-10-2020).pdf 2020-08-18
15 1755-MUMNP-2014-FORM 3 [25-06-2020(online)].pdf 2020-06-25
15 PCT IB 304.pdf 2018-08-11
16 1755-MUMNP-2014-FORM 3 [22-06-2020(online)].pdf 2020-06-22
16 GPA of Lupin Limited.pdf 2018-08-11
17 Form-18(Online).pdf 2018-08-11
17 1755-MUMNP-2014-FORM 3 [22-01-2020(online)].pdf 2020-01-22
18 1755-MUMNP-2014-FORM 3 [19-11-2019(online)].pdf 2019-11-19
18 FORM 5.pdf 2018-08-11
19 1755-MUMNP-2014-FORM 3 [19-09-2019(online)].pdf 2019-09-19
19 FORM 3.pdf 2018-08-11
20 1755-MUMNP-2014-ABSTRACT [21-11-2018(online)].pdf 2018-11-21
20 FORM 2 & Complete Specification.pdf 2018-08-11
21 1755-MUMNP-2014-CLAIMS [21-11-2018(online)].pdf 2018-11-21
21 ABSTRACT1.jpg 2018-08-11
22 1755-MUMNP-2014-COMPLETE SPECIFICATION [21-11-2018(online)].pdf 2018-11-21
22 1755-MUMNP-2014.pdf 2018-08-11
23 1755-MUMNP-2014-FER_SER_REPLY [21-11-2018(online)].pdf 2018-11-21
23 1755-MUMNP-2014-FORM 3-230215.pdf 2018-08-11
24 1755-MUMNP-2014-OTHERS [21-11-2018(online)].pdf 2018-11-21
24 1755-MUMNP-2014-FER.pdf 2018-08-11
25 1755-MUMNP-2014-CORRESPONDENCE-230215.pdf 2018-08-11
25 1755-MUMNP-2014-FORM 3 [10-11-2018(online)].pdf 2018-11-10
26 1755-MUMNP-2014-ANNEXURE TO FORM 3(15-4-2015).pdf 2018-08-11
26 1755-MUMNP-2014-CORRESPONDENCE(15-4-2015).pdf 2018-08-11
27 1755-MUMNP-2014-ANNEXURE TO FORM 3(15-4-2015).pdf 2018-08-11
27 1755-MUMNP-2014-CORRESPONDENCE(15-4-2015).pdf 2018-08-11
28 1755-MUMNP-2014-CORRESPONDENCE-230215.pdf 2018-08-11
28 1755-MUMNP-2014-FORM 3 [10-11-2018(online)].pdf 2018-11-10
29 1755-MUMNP-2014-FER.pdf 2018-08-11
29 1755-MUMNP-2014-OTHERS [21-11-2018(online)].pdf 2018-11-21
30 1755-MUMNP-2014-FER_SER_REPLY [21-11-2018(online)].pdf 2018-11-21
30 1755-MUMNP-2014-FORM 3-230215.pdf 2018-08-11
31 1755-MUMNP-2014-COMPLETE SPECIFICATION [21-11-2018(online)].pdf 2018-11-21
31 1755-MUMNP-2014.pdf 2018-08-11
32 1755-MUMNP-2014-CLAIMS [21-11-2018(online)].pdf 2018-11-21
32 ABSTRACT1.jpg 2018-08-11
33 1755-MUMNP-2014-ABSTRACT [21-11-2018(online)].pdf 2018-11-21
33 FORM 2 & Complete Specification.pdf 2018-08-11
34 1755-MUMNP-2014-FORM 3 [19-09-2019(online)].pdf 2019-09-19
34 FORM 3.pdf 2018-08-11
35 1755-MUMNP-2014-FORM 3 [19-11-2019(online)].pdf 2019-11-19
35 FORM 5.pdf 2018-08-11
36 Form-18(Online).pdf 2018-08-11
36 1755-MUMNP-2014-FORM 3 [22-01-2020(online)].pdf 2020-01-22
37 1755-MUMNP-2014-FORM 3 [22-06-2020(online)].pdf 2020-06-22
37 GPA of Lupin Limited.pdf 2018-08-11
38 1755-MUMNP-2014-FORM 3 [25-06-2020(online)].pdf 2020-06-25
38 PCT IB 304.pdf 2018-08-11
39 1755-MUMNP-2014-FORM 3 [11-04-2018(online)].pdf 2018-04-11
39 1755-MUMNP-2014-US(14)-HearingNotice-(HearingDate-08-10-2020).pdf 2020-08-18
40 1755-MUMNP-2014-FORM 3 [23-03-2018(online)].pdf 2018-03-23
40 1755-MUMNP-2014-Information under section 8(2) [09-10-2020(online)].pdf 2020-10-09
41 1755-MUMNP-2014-FORM 3 [04-12-2017(online)].pdf 2017-12-04
41 1755-MUMNP-2014-FORM 3 [09-10-2020(online)].pdf 2020-10-09
42 1755-MUMNP-2014-Written submissions and relevant documents [22-10-2020(online)].pdf 2020-10-22
42 Other Patent Document [09-05-2017(online)].pdf 2017-05-09
43 1755-MUMNP-2014-PETITION UNDER RULE 137 [22-10-2020(online)].pdf 2020-10-22
43 Other Patent Document [27-02-2017(online)].pdf 2017-02-27
44 1755-MUMNP-2014-FORM 3 [26-11-2020(online)].pdf 2020-11-26
44 Form 13 [24-08-2016(online)].pdf 2016-08-24
45 1755-MUMNP-2014-PatentCertificate04-02-2021.pdf 2021-02-04
45 Other Document [24-08-2016(online)].pdf 2016-08-24
46 1755-MUMNP-2014-IntimationOfGrant04-02-2021.pdf 2021-02-04
46 1755-MUMNP-2014-ANNEXURE TO FORM 3-05-03-2015.pdf 2015-03-05
47 1755-MUMNP-2014-RELEVANT DOCUMENTS [25-09-2021(online)].pdf 2021-09-25
47 1755-MUMNP-2014-ANNEXURE TO FORM-05-03-2015.pdf 2015-03-05
48 1755-MUMNP-2014-RELEVANT DOCUMENTS [25-09-2021(online)]-1.pdf 2021-09-25
48 1755-MUMNP-2014-CORRESPONDENCE-05-03-2015.pdf 2015-03-05
49 1755-MUMNP-2014-US(14)-ExtendedHearingNotice-(HearingDate-08-10-2020).pdf 2021-10-03
49 1755-MUMNP-2014-ANNEXURE TO FORM 3E(21-10-2014).pdf 2014-10-21
50 1755-MUMNP-2014-RELEVANT DOCUMENTS [21-09-2022(online)].pdf 2022-09-21
50 1755-MUMNP-2014-CORRESPONDENCE(21-10-2014).pdf 2014-10-21
51 1755-MUMNP-2014-CORRESPONDENCE(26-09-2014).pdf 2014-09-26
51 1755-MUMNP-2014-RELEVANT DOCUMENTS [21-09-2022(online)]-1.pdf 2022-09-21
52 1755-MUMNP-2014-FORM 1(26-09-2014).pdf 2014-09-26
52 1755-MUMNP-2014-RELEVANT DOCUMENTS [01-09-2023(online)].pdf 2023-09-01

Search Strategy

1 SEARCHSTRATEGY_24-05-2018.pdf

ERegister / Renewals

3rd: 08 Feb 2021

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4th: 08 Feb 2021

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5th: 08 Feb 2021

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6th: 08 Feb 2021

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7th: 08 Feb 2021

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8th: 08 Feb 2021

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9th: 08 Feb 2021

From 11/03/2021 - To 11/03/2022

10th: 11 Feb 2022

From 11/03/2022 - To 11/03/2023

11th: 09 Feb 2023

From 11/03/2023 - To 11/03/2024

12th: 13 Jan 2024

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13th: 10 Jan 2025

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