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Histamine H3 Receptor Agents, Preparation And Therapeutic Uses.
Abstract: The present invention discloses novel compounds of Formula I or pharmaceutically acceptable salts thereof which have histamine-H3 receptor antagonist or inverse agonist activity, as well as methods for preparing such compounds. In another embodiment, the invention discloses pharmaceutical compositions comprising compounds of Formula I as well as methods of using them to treat obesity, cognitive deficiencies, narcolepsy, and other histamine H3 receptor-related diseases.
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Notices, Deadlines & Correspondence
Notices, Deadlines & Correspondence
Patent Information
Application #
Filing Date
05 October 2006
Publication Number
23/2007
Publication Type
INA
Invention Field
PHARMACEUTICALS
Status
Email
Parent Application
Applicants
ELI LILLY AND COMPANY
A CORPORATION OF THE STATE OF INDIANA,U.S.A.
HAVING A PRINCIPAL PLACE OF BUISNESS AT,
LILLY CORPORATE CENTER,
CITY OF INDIANAPOLIS,
STATE OF INDIANA 46285,
U.S.A.
Inventors
1. BEAVERS,LISA,SELSAM
74 NORTH EDWARDS STREET,
FRANKLIN,INDIANA 46131,
U.S.A.
2. FINLEY,DON,RICHARD
4644 MACY DRIVE,GREENWOOD,
INDIANA 46142,
U.S.A.
3. FINN,TERRY,PATRICK
ELI LILLY AND COMPANY LTD.,
KINGSCLERE ROAD,
BASINGSTOKE HAMPSHIRE RG21 6XA,
U.K.
4. GADSKI,ROBERT,ALAN
4431 NORTH ILLINOIS,
INDIANAPOLIS,
INDIANA 46208,
U.S.A.
5. HIPSKIND,PHILIP,ARTHUR
4255 CABIN COURT,
NEW PALESTINE,
INDIANA 46163,
U.S.A.
6. HORNBACK,WILLIAM,JOSHEPH
10063 BENT TREE LANE,
FISHERS,INDIANA 46038,
U.S.A.
7. JESUDASON,CYNTHIA,DARSHINI
1090 FLEETWOOD DRIVE,
INDIANAPOLIS,INDIANA 46228,
U.S.A.
8. PICKARD,RICHARD,TODD
20980 PRAIRIE BAPTIST ROAD,NOBLESVILLE,
INDIANA 46060,
U.S.A.
9. TAKAKUWA,TAKAKO
7653 GERMANDER LANE,
INDIANAPOLIS,
INDIANA 46237,
U.S.A.
10. VAUGHAT,GRANT,MATHEWS
7352 TARRAGON LANE,
INDIANAPOLIS,INDIANA 46237,
U.S.A.
Specification
The present invention discloses novel compounds of Formula I or pharmaceutically acceptable salts thereof which have histamine-H3 receptor antagonist or inverse agonist activity, as well as methods for preparing such compounds. In another embodiment, the invention discloses pharmaceutical compositions comprising compounds of Formula I as well as methods of using them to treat obesity, cognitive deficiencies, narcolepsy, and other histamine H3 receptor-related diseases.
Documents
Orders
| Section | Controller | Decision Date |
|---|---|---|
Application Documents
| # | Name | Date |
|---|---|---|
| 1 | 2868-KOLNP-2006-(20-12-2007)-FORM 13.pdf | 2007-12-20 |
| 1 | 2868-KOLNP-2006_EXAMREPORT.pdf | 2016-06-30 |
| 2 | 2868-KOLNP-2006-(28-01-2016)-CORRESPONDENCE.pdf | 2016-01-28 |
| 2 | 2868-kolnp-2006-FORM 18.pdf | 2011-10-07 |
| 3 | 2868-KOLNP-2006-(10-09-2013)-CLAIMS.pdf | 2013-09-10 |
| 3 | 02868-kolnp-2006-priority document.pdf | 2011-10-07 |
| 4 | 2868-KOLNP-2006-(10-09-2013)-CORRESPONDENCE.pdf | 2013-09-10 |
| 4 | 02868-kolnp-2006-form-3-1.1.pdf | 2011-10-07 |
| 5 | 2868-KOLNP-2006-(10-09-2013)-FORM-1.pdf | 2013-09-10 |
| 5 | 02868-kolnp-2006-correspondence others-1.1.pdf | 2011-10-07 |
| 6 | 2868-KOLNP-2006-(10-09-2013)-FORM-13.pdf | 2013-09-10 |
| 6 | 02868-kolnp-2006 pct request.pdf | 2011-10-07 |
| 7 | 2868-KOLNP-2006-(10-09-2013)-FORM-5.pdf | 2013-09-10 |
| 7 | 02868-kolnp-2006 pct others.pdf | 2011-10-07 |
| 8 | 2868-KOLNP-2006-(10-09-2013)-OTHERS.pdf | 2013-09-10 |
| 8 | 02868-kolnp-2006 international search authority report.pdf | 2011-10-07 |
| 9 | 02868-kolnp-2006 international publication.pdf | 2011-10-07 |
| 9 | 2868-KOLNP-2006-(10-09-2013)-PETITION UNDER RULE 137.pdf | 2013-09-10 |
| 10 | 02868-kolnp-2006 general form of authorisation.pdf | 2011-10-07 |
| 10 | 2868-KOLNP-2006-(31-07-2013)-ANNEXURE TO FORM 3.pdf | 2013-07-31 |
| 11 | 02868-kolnp-2006 form-5.pdf | 2011-10-07 |
| 11 | 2868-KOLNP-2006-(31-07-2013)-CORRESPONDENCE.pdf | 2013-07-31 |
| 12 | 02868-kolnp-2006 form-3.pdf | 2011-10-07 |
| 12 | 2868-KOLNP-2006-(31-07-2013)-FORM-3.pdf | 2013-07-31 |
| 13 | 02868-kolnp-2006 form-2.pdf | 2011-10-07 |
| 13 | 2868-KOLNP-2006-(31-07-2013)-OTHERS.pdf | 2013-07-31 |
| 14 | 02868-kolnp-2006 form-1.pdf | 2011-10-07 |
| 14 | 2868-KOLNP-2006-(04-02-2013)-CORRESPONDENCE.pdf | 2013-02-04 |
| 15 | 02868-kolnp-2006 description(complete).pdf | 2011-10-07 |
| 15 | 2868-KOLNP-2006-(04-02-2013)-OTHERS.pdf | 2013-02-04 |
| 16 | 02868-kolnp-2006 correspondence others.pdf | 2011-10-07 |
| 16 | 2868-KOLNP-2006 last claim amendment.pdf | 2013-01-15 |
| 17 | 02868-kolnp-2006 claims.pdf | 2011-10-07 |
| 18 | 2868-KOLNP-2006-(26-10-2012)-CORRESPONDENCE.pdf | 2012-10-26 |
| 18 | 02868-kolnp-2006 abstract.pdf | 2011-10-07 |
| 19 | 2868-KOLNP-2006-(26-10-2012)-OTHERS.pdf | 2012-10-26 |
| 19 | 2868-KOLNP-2006-(26-10-2012)-PA.pdf | 2012-10-26 |
| 20 | 2868-KOLNP-2006-(26-10-2012)-OTHERS.pdf | 2012-10-26 |
| 20 | 2868-KOLNP-2006-(26-10-2012)-PA.pdf | 2012-10-26 |
| 21 | 02868-kolnp-2006 abstract.pdf | 2011-10-07 |
| 21 | 2868-KOLNP-2006-(26-10-2012)-CORRESPONDENCE.pdf | 2012-10-26 |
| 22 | 02868-kolnp-2006 claims.pdf | 2011-10-07 |
| 23 | 02868-kolnp-2006 correspondence others.pdf | 2011-10-07 |
| 23 | 2868-KOLNP-2006 last claim amendment.pdf | 2013-01-15 |
| 24 | 2868-KOLNP-2006-(04-02-2013)-OTHERS.pdf | 2013-02-04 |
| 24 | 02868-kolnp-2006 description(complete).pdf | 2011-10-07 |
| 25 | 2868-KOLNP-2006-(04-02-2013)-CORRESPONDENCE.pdf | 2013-02-04 |
| 25 | 02868-kolnp-2006 form-1.pdf | 2011-10-07 |
| 26 | 02868-kolnp-2006 form-2.pdf | 2011-10-07 |
| 26 | 2868-KOLNP-2006-(31-07-2013)-OTHERS.pdf | 2013-07-31 |
| 27 | 02868-kolnp-2006 form-3.pdf | 2011-10-07 |
| 27 | 2868-KOLNP-2006-(31-07-2013)-FORM-3.pdf | 2013-07-31 |
| 28 | 02868-kolnp-2006 form-5.pdf | 2011-10-07 |
| 28 | 2868-KOLNP-2006-(31-07-2013)-CORRESPONDENCE.pdf | 2013-07-31 |
| 29 | 02868-kolnp-2006 general form of authorisation.pdf | 2011-10-07 |
| 29 | 2868-KOLNP-2006-(31-07-2013)-ANNEXURE TO FORM 3.pdf | 2013-07-31 |
| 30 | 02868-kolnp-2006 international publication.pdf | 2011-10-07 |
| 30 | 2868-KOLNP-2006-(10-09-2013)-PETITION UNDER RULE 137.pdf | 2013-09-10 |
| 31 | 2868-KOLNP-2006-(10-09-2013)-OTHERS.pdf | 2013-09-10 |
| 31 | 02868-kolnp-2006 international search authority report.pdf | 2011-10-07 |
| 32 | 2868-KOLNP-2006-(10-09-2013)-FORM-5.pdf | 2013-09-10 |
| 32 | 02868-kolnp-2006 pct others.pdf | 2011-10-07 |
| 33 | 2868-KOLNP-2006-(10-09-2013)-FORM-13.pdf | 2013-09-10 |
| 33 | 02868-kolnp-2006 pct request.pdf | 2011-10-07 |
| 34 | 2868-KOLNP-2006-(10-09-2013)-FORM-1.pdf | 2013-09-10 |
| 34 | 02868-kolnp-2006-correspondence others-1.1.pdf | 2011-10-07 |
| 35 | 2868-KOLNP-2006-(10-09-2013)-CORRESPONDENCE.pdf | 2013-09-10 |
| 35 | 02868-kolnp-2006-form-3-1.1.pdf | 2011-10-07 |
| 36 | 2868-KOLNP-2006-(10-09-2013)-CLAIMS.pdf | 2013-09-10 |
| 36 | 02868-kolnp-2006-priority document.pdf | 2011-10-07 |
| 37 | 2868-KOLNP-2006-(28-01-2016)-CORRESPONDENCE.pdf | 2016-01-28 |
| 37 | 2868-kolnp-2006-FORM 18.pdf | 2011-10-07 |
| 38 | 2868-KOLNP-2006-(20-12-2007)-FORM 13.pdf | 2007-12-20 |
| 38 | 2868-KOLNP-2006_EXAMREPORT.pdf | 2016-06-30 |