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Imidazopyridine Compound

Abstract: [Problem] To provide an excellent therapeutic or prophylactic agent for cardiovascular diseases on the basis of cGMP production increasing activity attributed to soluble guanylate cyclase activating activity. [Solution] It was discovered that an imidazopyridine compound having a carbamoyl group at the 3 position of an imidazo[1 2 a]pyridine skeleton and having a substituent attached to the 8 position of the skeleton through an oxygen atom exhibits cGMP production increasing activity attributed to potent soluble guanylate cyclase activating activity and can be used in an excellent therapeutic or prophylactic agent for various cardiovascular diseases associated with soluble guanylate cyclase and the invention was completed.

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Notices, Deadlines & Correspondence

Patent Information

Application #
Filing Date
26 November 2013
Publication Number
11/2015
Publication Type
INA
Invention Field
CHEMICAL
Status
Email
patent@depenning.com
Parent Application

Applicants

Astellas Pharma Inc.
3 11 Nihonbashi Honcho 2 chome Chuo ku Tokyo 1038411

Inventors

1. KOGA Yuji
c/o Astellas Pharma Inc. 3 11 Nihonbashi Honcho 2 chome Chuo ku Tokyo 1038411
2. MAENO Kyoichi
c/o Astellas Pharma Inc. 3 11 Nihonbashi Honcho 2 chome Chuo ku Tokyo 1038411
3. SATO Ippei
c/o Astellas Pharma Inc. 3 11 Nihonbashi Honcho 2 chome Chuo ku Tokyo 1038411
4. IMAMURA Yoshimasa
c/o Astellas Pharma Inc. 3 11 Nihonbashi Honcho 2 chome Chuo ku Tokyo 1038411
5. HANAZAWA Takeshi
c/o Astellas Pharma Inc. 3 11 Nihonbashi Honcho 2 chome Chuo ku Tokyo 1038411
6. IIDA Maiko
c/o Astellas Pharma Inc. 3 11 Nihonbashi Honcho 2 chome Chuo ku Tokyo 1038411
7. OHNE Kazuhiko
c/o Astellas Pharma Inc. 3 11 Nihonbashi Honcho 2 chome Chuo ku Tokyo 1038411
8. IMAMURA Kenichiro
c/o Astellas Pharma Inc. 3 11 Nihonbashi Honcho 2 chome Chuo ku Tokyo 1038411
9. WATANABE Tsubasa
c/o Astellas Pharma Inc. 3 11 Nihonbashi Honcho 2 chome Chuo ku Tokyo 1038411
10. NOZAWA Eisuke
c/o Astellas Pharma Inc. 3 11 Nihonbashi Honcho 2 chome Chuo ku Tokyo 1038411
11. SHIBATA Hiroshi
c/o Astellas Pharma Inc. 3 11 Nihonbashi Honcho 2 chome Chuo ku Tokyo 1038411

Specification

PLS SEE ATTACHEMENTS.

Documents

Application Documents

# Name Date
1 9465-CHENP-2013 FORM-3 14-07-2014.pdf 2014-07-14
1 9465-CHENP-2013 POWER OF ATTORNEY 26-11-2013.pdf 2013-11-26
2 9465-CHENP-2013.pdf 2014-01-10
2 9465-CHENP-2013 PCT 26-11-2013.pdf 2013-11-26
3 9465-CHENP-2013 FORM-5 26-11-2013.pdf 2013-11-26
3 9465-CHENP-2013 ABSTRACT 26-11-2013.pdf 2013-11-26
4 9465-CHENP-2013 CLAIMS 26-11-2013.pdf 2013-11-26
4 9465-CHENP-2013 FORM-3 26-11-2013.pdf 2013-11-26
5 9465-CHENP-2013 FORM-2 26-11-2013.pdf 2013-11-26
5 9465-CHENP-2013 CORRESPONDENCE OTHERS 26-11-2013.pdf 2013-11-26
6 9465-CHENP-2013 FORM-1 26-11-2013.pdf 2013-11-26
6 9465-CHENP-2013 DESCRIPTION (COMPLETE) 26-11-2013.pdf 2013-11-26
7 9465-CHENP-2013 ENGLISH TRANSLATION 26-11-2013.pdf 2013-11-26
7 9465-CHENP-2013 DESCRIPTION (COMPLETE)1 26-11-2013.pdf 2013-11-26
8 9465-CHENP-2013 ENGLISH TRANSLATION 26-11-2013.pdf 2013-11-26
8 9465-CHENP-2013 DESCRIPTION (COMPLETE)1 26-11-2013.pdf 2013-11-26
9 9465-CHENP-2013 FORM-1 26-11-2013.pdf 2013-11-26
9 9465-CHENP-2013 DESCRIPTION (COMPLETE) 26-11-2013.pdf 2013-11-26
10 9465-CHENP-2013 CORRESPONDENCE OTHERS 26-11-2013.pdf 2013-11-26
10 9465-CHENP-2013 FORM-2 26-11-2013.pdf 2013-11-26
11 9465-CHENP-2013 CLAIMS 26-11-2013.pdf 2013-11-26
11 9465-CHENP-2013 FORM-3 26-11-2013.pdf 2013-11-26
12 9465-CHENP-2013 FORM-5 26-11-2013.pdf 2013-11-26
12 9465-CHENP-2013 ABSTRACT 26-11-2013.pdf 2013-11-26
13 9465-CHENP-2013.pdf 2014-01-10
13 9465-CHENP-2013 PCT 26-11-2013.pdf 2013-11-26
14 9465-CHENP-2013 POWER OF ATTORNEY 26-11-2013.pdf 2013-11-26
14 9465-CHENP-2013 FORM-3 14-07-2014.pdf 2014-07-14