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Inhibitors Of 11 Beta Hydroxysteroid Dehydrogenase 1

Abstract: The present invention discloses novel compounds of Formula I: ( I ) possessing 11β-HSD type 1 antagonist activity, as well as methods for preparing such compounds. In another embodiment, the invention discloses pharmaceutical compositions comprising compounds of Formula I, as well as methods of using the compounds and compositions to treat diabetes, hyperglycemia, obesity, hypertension, hyperlipidemia, metabolic syndrome, cognitive disorders, and other conditions associated with 11β-HSD type 1 activity.

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Notices, Deadlines & Correspondence

Patent Information

Application #
Filing Date
23 October 2008
Publication Number
03/2009
Publication Type
INA
Invention Field
CHEMICAL
Status
Email
Parent Application
Patent Number
Legal Status
Grant Date
2013-02-20
Renewal Date

Applicants

ELI LILLY AND COMPANY
LILLY CORPORATE CENTER, INDIANAPOLIS, INDIANA 46285,

Inventors

1. LI, RENHUA
10493 Hollowood Court  Fishers  Indiana 46038   USA
2. WALLACE, OWEN, BRENDAN
13297 Mink Lane  Westfield  Indiana 46074  USA
3. XU, YANPING
6676 Pennan Court  Noblesville  Indiana 46062  USA

Specification

PLEASE SEE THE SPECIFICATION ATTACHED.

Documents

Application Documents

# Name Date
1 2277-MUMNP-2008-CLAIMS(AMENDED)-(15-5-2012).pdf 2018-08-09
1 2277-mumnp-2008-wo international publication report(23-10-2008).pdf 2008-10-23
2 2277-mumnp-2008-claims(amended)-(4-11-2008).pdf 2018-08-09
2 2277-mumnp-2008-form 5(23-10-2008).pdf 2008-10-23
3 2277-mumnp-2008-form 3(23-10-2008).pdf 2008-10-23
3 2277-MUMNP-2008-CLAIMS(GRANTED).pdf 2018-08-09
4 2277-mumnp-2008-form 2(title page)-(23-10-2008).pdf 2008-10-23
4 2277-MUMNP-2008-CLAIMS(MARKED COPY)-(15-5-2012).pdf 2018-08-09
5 2277-mumnp-2008-form 2(23-10-2008).pdf 2008-10-23
5 2277-MUMNP-2008-CORRESPONDENCE(13-4-2009).pdf 2018-08-09
6 2277-mumnp-2008-form 1(23-10-2008).pdf 2008-10-23
6 2277-MUMNP-2008-CORRESPONDENCE(14-9-2011).pdf 2018-08-09
7 2277-mumnp-2008-description(complete)-(23-10-2008).pdf 2008-10-23
7 2277-MUMNP-2008-CORRESPONDENCE(17-1-2013).pdf 2018-08-09
8 2277-MUMNP-2008-CORRESPONDENCE(26-7-2012).pdf 2018-08-09
8 2277-mumnp-2008-claims(23-10-2008).pdf 2008-10-23
9 2277-mumnp-2008-abstract(23-10-2008).pdf 2008-10-23
9 2277-MUMNP-2008-CORRESPONDENCE(30-8-2012).pdf 2018-08-09
10 2277-MUMNP-2008-CORRESPONDENCE(24-12-2008).pdf 2008-12-24
10 2277-MUMNP-2008-CORRESPONDENCE(IPO).pdf 2018-08-09
11 2277-MUMNP-2008-ASSIGNMENT(24-12-2008).pdf 2008-12-24
11 2277-MUMNP-2008-DESCRIPTION(GRANTED).pdf 2018-08-09
12 2277-MUMNP-2008-EP DOCUMENT(15-5-2012).pdf 2018-08-09
12 Form 27 [29-03-2016(online)].pdf 2016-03-29
13 2277-MUMNP-2008-FORM 1(30-8-2012).pdf 2018-08-09
13 Petition Under Rule 137 [11-04-2017(online)].pdf 2017-04-11
14 2277-MUMNP-2008-FORM 13(26-7-2012).pdf 2018-08-09
14 Form 27 [11-04-2017(online)].pdf 2017-04-11
15 2277-mumnp-2008-form 13(4-11-2008).pdf 2018-08-09
15 ipindiaonline.gov.in_epatentfiling_online_frmPreview.asp.pdf 2018-08-09
16 2277-mumnp-2008-form 18(4-11-2008).pdf 2018-08-09
16 Form-5.pdf 2018-08-09
17 Form-3.pdf 2018-08-09
17 2277-MUMNP-2008-FORM 2(TITLE PAGE)-(GRANTED).pdf 2018-08-09
18 2277-MUMNP-2008-FORM 26(14-9-2011).pdf 2018-08-09
18 Form-1.pdf 2018-08-09
19 2277-MUMNP-2008-FORM 26(15-5-2012).pdf 2018-08-09
19 abstract1.jpg 2018-08-09
20 2277-MUMNP-2008-FORM 3(13-4-2009).pdf 2018-08-09
20 2277-MUMNP-2008_EXAMREPORT.pdf 2018-08-09
21 2277-MUMNP-2008-FORM 3(15-5-2012).pdf 2018-08-09
21 2277-MUMNP-2008-US DOCUMENT(15-5-2012).pdf 2018-08-09
22 2277-MUMNP-2008-FORM2(GRANTED).pdf 2018-08-09
22 2277-MUMNP-2008-REPLY TO EXAMINATION REPORT(15-5-2012).pdf 2018-08-09
23 2277-mumnp-2008-marked copy(4-11-2008).pdf 2018-08-09
23 2277-MUMNP-2008-PETITION UNDER RULE-137(17-1-2013).pdf 2018-08-09
24 2277-MUMNP-2008-PETITION UNDER RULE 137(15-5-2012).pdf 2018-08-09
24 2277-MUMNP-2008-PCT CLAIMS(15-5-2012).pdf 2018-08-09
25 2277-MUMNP-2008-PCT CLAIMS(15-5-2012).pdf 2018-08-09
25 2277-MUMNP-2008-PETITION UNDER RULE 137(15-5-2012).pdf 2018-08-09
26 2277-mumnp-2008-marked copy(4-11-2008).pdf 2018-08-09
26 2277-MUMNP-2008-PETITION UNDER RULE-137(17-1-2013).pdf 2018-08-09
27 2277-MUMNP-2008-FORM2(GRANTED).pdf 2018-08-09
27 2277-MUMNP-2008-REPLY TO EXAMINATION REPORT(15-5-2012).pdf 2018-08-09
28 2277-MUMNP-2008-FORM 3(15-5-2012).pdf 2018-08-09
28 2277-MUMNP-2008-US DOCUMENT(15-5-2012).pdf 2018-08-09
29 2277-MUMNP-2008-FORM 3(13-4-2009).pdf 2018-08-09
29 2277-MUMNP-2008_EXAMREPORT.pdf 2018-08-09
30 2277-MUMNP-2008-FORM 26(15-5-2012).pdf 2018-08-09
30 abstract1.jpg 2018-08-09
31 2277-MUMNP-2008-FORM 26(14-9-2011).pdf 2018-08-09
31 Form-1.pdf 2018-08-09
32 2277-MUMNP-2008-FORM 2(TITLE PAGE)-(GRANTED).pdf 2018-08-09
32 Form-3.pdf 2018-08-09
33 2277-mumnp-2008-form 18(4-11-2008).pdf 2018-08-09
33 Form-5.pdf 2018-08-09
34 2277-mumnp-2008-form 13(4-11-2008).pdf 2018-08-09
34 ipindiaonline.gov.in_epatentfiling_online_frmPreview.asp.pdf 2018-08-09
35 2277-MUMNP-2008-FORM 13(26-7-2012).pdf 2018-08-09
35 Form 27 [11-04-2017(online)].pdf 2017-04-11
36 Petition Under Rule 137 [11-04-2017(online)].pdf 2017-04-11
36 2277-MUMNP-2008-FORM 1(30-8-2012).pdf 2018-08-09
37 2277-MUMNP-2008-EP DOCUMENT(15-5-2012).pdf 2018-08-09
37 Form 27 [29-03-2016(online)].pdf 2016-03-29
38 2277-MUMNP-2008-ASSIGNMENT(24-12-2008).pdf 2008-12-24
38 2277-MUMNP-2008-DESCRIPTION(GRANTED).pdf 2018-08-09
39 2277-MUMNP-2008-CORRESPONDENCE(24-12-2008).pdf 2008-12-24
39 2277-MUMNP-2008-CORRESPONDENCE(IPO).pdf 2018-08-09
40 2277-mumnp-2008-abstract(23-10-2008).pdf 2008-10-23
40 2277-MUMNP-2008-CORRESPONDENCE(30-8-2012).pdf 2018-08-09
41 2277-mumnp-2008-claims(23-10-2008).pdf 2008-10-23
41 2277-MUMNP-2008-CORRESPONDENCE(26-7-2012).pdf 2018-08-09
42 2277-mumnp-2008-description(complete)-(23-10-2008).pdf 2008-10-23
42 2277-MUMNP-2008-CORRESPONDENCE(17-1-2013).pdf 2018-08-09
43 2277-mumnp-2008-form 1(23-10-2008).pdf 2008-10-23
43 2277-MUMNP-2008-CORRESPONDENCE(14-9-2011).pdf 2018-08-09
44 2277-mumnp-2008-form 2(23-10-2008).pdf 2008-10-23
44 2277-MUMNP-2008-CORRESPONDENCE(13-4-2009).pdf 2018-08-09
45 2277-mumnp-2008-form 2(title page)-(23-10-2008).pdf 2008-10-23
45 2277-MUMNP-2008-CLAIMS(MARKED COPY)-(15-5-2012).pdf 2018-08-09
46 2277-mumnp-2008-form 3(23-10-2008).pdf 2008-10-23
46 2277-MUMNP-2008-CLAIMS(GRANTED).pdf 2018-08-09
47 2277-mumnp-2008-claims(amended)-(4-11-2008).pdf 2018-08-09
47 2277-mumnp-2008-form 5(23-10-2008).pdf 2008-10-23
48 2277-MUMNP-2008-CLAIMS(AMENDED)-(15-5-2012).pdf 2018-08-09
48 2277-mumnp-2008-wo international publication report(23-10-2008).pdf 2008-10-23

ERegister / Renewals

3rd: 17 May 2013

From 25/04/2009 - To 25/04/2010

4th: 17 May 2013

From 25/04/2010 - To 25/04/2011

5th: 17 May 2013

From 25/04/2011 - To 25/04/2012

6th: 17 May 2013

From 25/04/2012 - To 25/04/2013

7th: 17 May 2013

From 25/04/2013 - To 25/04/2014

8th: 19 Apr 2014

From 25/04/2014 - To 25/04/2015

9th: 08 Apr 2015

From 25/04/2015 - To 25/04/2016

10th: 05 Apr 2016

From 25/04/2016 - To 25/04/2017

11th: 05 Apr 2017

From 25/04/2017 - To 25/04/2018