Abstract: The present invention discloses novel compounds of Formula I: ( I ) possessing 11β-HSD type 1 antagonist activity, as well as methods for preparing such compounds. In another embodiment, the invention discloses pharmaceutical compositions comprising compounds of Formula I, as well as methods of using the compounds and compositions to treat diabetes, hyperglycemia, obesity, hypertension, hyperlipidemia, metabolic syndrome, cognitive disorders, and other conditions associated with 11β-HSD type 1 activity.
PLEASE SEE THE SPECIFICATION ATTACHED.
| # | Name | Date |
|---|---|---|
| 1 | 2277-MUMNP-2008-CLAIMS(AMENDED)-(15-5-2012).pdf | 2018-08-09 |
| 1 | 2277-mumnp-2008-wo international publication report(23-10-2008).pdf | 2008-10-23 |
| 2 | 2277-mumnp-2008-claims(amended)-(4-11-2008).pdf | 2018-08-09 |
| 2 | 2277-mumnp-2008-form 5(23-10-2008).pdf | 2008-10-23 |
| 3 | 2277-mumnp-2008-form 3(23-10-2008).pdf | 2008-10-23 |
| 3 | 2277-MUMNP-2008-CLAIMS(GRANTED).pdf | 2018-08-09 |
| 4 | 2277-mumnp-2008-form 2(title page)-(23-10-2008).pdf | 2008-10-23 |
| 4 | 2277-MUMNP-2008-CLAIMS(MARKED COPY)-(15-5-2012).pdf | 2018-08-09 |
| 5 | 2277-mumnp-2008-form 2(23-10-2008).pdf | 2008-10-23 |
| 5 | 2277-MUMNP-2008-CORRESPONDENCE(13-4-2009).pdf | 2018-08-09 |
| 6 | 2277-mumnp-2008-form 1(23-10-2008).pdf | 2008-10-23 |
| 6 | 2277-MUMNP-2008-CORRESPONDENCE(14-9-2011).pdf | 2018-08-09 |
| 7 | 2277-mumnp-2008-description(complete)-(23-10-2008).pdf | 2008-10-23 |
| 7 | 2277-MUMNP-2008-CORRESPONDENCE(17-1-2013).pdf | 2018-08-09 |
| 8 | 2277-MUMNP-2008-CORRESPONDENCE(26-7-2012).pdf | 2018-08-09 |
| 8 | 2277-mumnp-2008-claims(23-10-2008).pdf | 2008-10-23 |
| 9 | 2277-mumnp-2008-abstract(23-10-2008).pdf | 2008-10-23 |
| 9 | 2277-MUMNP-2008-CORRESPONDENCE(30-8-2012).pdf | 2018-08-09 |
| 10 | 2277-MUMNP-2008-CORRESPONDENCE(24-12-2008).pdf | 2008-12-24 |
| 10 | 2277-MUMNP-2008-CORRESPONDENCE(IPO).pdf | 2018-08-09 |
| 11 | 2277-MUMNP-2008-ASSIGNMENT(24-12-2008).pdf | 2008-12-24 |
| 11 | 2277-MUMNP-2008-DESCRIPTION(GRANTED).pdf | 2018-08-09 |
| 12 | 2277-MUMNP-2008-EP DOCUMENT(15-5-2012).pdf | 2018-08-09 |
| 12 | Form 27 [29-03-2016(online)].pdf | 2016-03-29 |
| 13 | 2277-MUMNP-2008-FORM 1(30-8-2012).pdf | 2018-08-09 |
| 13 | Petition Under Rule 137 [11-04-2017(online)].pdf | 2017-04-11 |
| 14 | 2277-MUMNP-2008-FORM 13(26-7-2012).pdf | 2018-08-09 |
| 14 | Form 27 [11-04-2017(online)].pdf | 2017-04-11 |
| 15 | 2277-mumnp-2008-form 13(4-11-2008).pdf | 2018-08-09 |
| 15 | ipindiaonline.gov.in_epatentfiling_online_frmPreview.asp.pdf | 2018-08-09 |
| 16 | 2277-mumnp-2008-form 18(4-11-2008).pdf | 2018-08-09 |
| 16 | Form-5.pdf | 2018-08-09 |
| 17 | Form-3.pdf | 2018-08-09 |
| 17 | 2277-MUMNP-2008-FORM 2(TITLE PAGE)-(GRANTED).pdf | 2018-08-09 |
| 18 | 2277-MUMNP-2008-FORM 26(14-9-2011).pdf | 2018-08-09 |
| 18 | Form-1.pdf | 2018-08-09 |
| 19 | 2277-MUMNP-2008-FORM 26(15-5-2012).pdf | 2018-08-09 |
| 19 | abstract1.jpg | 2018-08-09 |
| 20 | 2277-MUMNP-2008-FORM 3(13-4-2009).pdf | 2018-08-09 |
| 20 | 2277-MUMNP-2008_EXAMREPORT.pdf | 2018-08-09 |
| 21 | 2277-MUMNP-2008-FORM 3(15-5-2012).pdf | 2018-08-09 |
| 21 | 2277-MUMNP-2008-US DOCUMENT(15-5-2012).pdf | 2018-08-09 |
| 22 | 2277-MUMNP-2008-FORM2(GRANTED).pdf | 2018-08-09 |
| 22 | 2277-MUMNP-2008-REPLY TO EXAMINATION REPORT(15-5-2012).pdf | 2018-08-09 |
| 23 | 2277-mumnp-2008-marked copy(4-11-2008).pdf | 2018-08-09 |
| 23 | 2277-MUMNP-2008-PETITION UNDER RULE-137(17-1-2013).pdf | 2018-08-09 |
| 24 | 2277-MUMNP-2008-PETITION UNDER RULE 137(15-5-2012).pdf | 2018-08-09 |
| 24 | 2277-MUMNP-2008-PCT CLAIMS(15-5-2012).pdf | 2018-08-09 |
| 25 | 2277-MUMNP-2008-PCT CLAIMS(15-5-2012).pdf | 2018-08-09 |
| 25 | 2277-MUMNP-2008-PETITION UNDER RULE 137(15-5-2012).pdf | 2018-08-09 |
| 26 | 2277-mumnp-2008-marked copy(4-11-2008).pdf | 2018-08-09 |
| 26 | 2277-MUMNP-2008-PETITION UNDER RULE-137(17-1-2013).pdf | 2018-08-09 |
| 27 | 2277-MUMNP-2008-FORM2(GRANTED).pdf | 2018-08-09 |
| 27 | 2277-MUMNP-2008-REPLY TO EXAMINATION REPORT(15-5-2012).pdf | 2018-08-09 |
| 28 | 2277-MUMNP-2008-FORM 3(15-5-2012).pdf | 2018-08-09 |
| 28 | 2277-MUMNP-2008-US DOCUMENT(15-5-2012).pdf | 2018-08-09 |
| 29 | 2277-MUMNP-2008-FORM 3(13-4-2009).pdf | 2018-08-09 |
| 29 | 2277-MUMNP-2008_EXAMREPORT.pdf | 2018-08-09 |
| 30 | 2277-MUMNP-2008-FORM 26(15-5-2012).pdf | 2018-08-09 |
| 30 | abstract1.jpg | 2018-08-09 |
| 31 | 2277-MUMNP-2008-FORM 26(14-9-2011).pdf | 2018-08-09 |
| 31 | Form-1.pdf | 2018-08-09 |
| 32 | 2277-MUMNP-2008-FORM 2(TITLE PAGE)-(GRANTED).pdf | 2018-08-09 |
| 32 | Form-3.pdf | 2018-08-09 |
| 33 | 2277-mumnp-2008-form 18(4-11-2008).pdf | 2018-08-09 |
| 33 | Form-5.pdf | 2018-08-09 |
| 34 | 2277-mumnp-2008-form 13(4-11-2008).pdf | 2018-08-09 |
| 34 | ipindiaonline.gov.in_epatentfiling_online_frmPreview.asp.pdf | 2018-08-09 |
| 35 | 2277-MUMNP-2008-FORM 13(26-7-2012).pdf | 2018-08-09 |
| 35 | Form 27 [11-04-2017(online)].pdf | 2017-04-11 |
| 36 | Petition Under Rule 137 [11-04-2017(online)].pdf | 2017-04-11 |
| 36 | 2277-MUMNP-2008-FORM 1(30-8-2012).pdf | 2018-08-09 |
| 37 | 2277-MUMNP-2008-EP DOCUMENT(15-5-2012).pdf | 2018-08-09 |
| 37 | Form 27 [29-03-2016(online)].pdf | 2016-03-29 |
| 38 | 2277-MUMNP-2008-ASSIGNMENT(24-12-2008).pdf | 2008-12-24 |
| 38 | 2277-MUMNP-2008-DESCRIPTION(GRANTED).pdf | 2018-08-09 |
| 39 | 2277-MUMNP-2008-CORRESPONDENCE(24-12-2008).pdf | 2008-12-24 |
| 39 | 2277-MUMNP-2008-CORRESPONDENCE(IPO).pdf | 2018-08-09 |
| 40 | 2277-mumnp-2008-abstract(23-10-2008).pdf | 2008-10-23 |
| 40 | 2277-MUMNP-2008-CORRESPONDENCE(30-8-2012).pdf | 2018-08-09 |
| 41 | 2277-mumnp-2008-claims(23-10-2008).pdf | 2008-10-23 |
| 41 | 2277-MUMNP-2008-CORRESPONDENCE(26-7-2012).pdf | 2018-08-09 |
| 42 | 2277-mumnp-2008-description(complete)-(23-10-2008).pdf | 2008-10-23 |
| 42 | 2277-MUMNP-2008-CORRESPONDENCE(17-1-2013).pdf | 2018-08-09 |
| 43 | 2277-mumnp-2008-form 1(23-10-2008).pdf | 2008-10-23 |
| 43 | 2277-MUMNP-2008-CORRESPONDENCE(14-9-2011).pdf | 2018-08-09 |
| 44 | 2277-mumnp-2008-form 2(23-10-2008).pdf | 2008-10-23 |
| 44 | 2277-MUMNP-2008-CORRESPONDENCE(13-4-2009).pdf | 2018-08-09 |
| 45 | 2277-mumnp-2008-form 2(title page)-(23-10-2008).pdf | 2008-10-23 |
| 45 | 2277-MUMNP-2008-CLAIMS(MARKED COPY)-(15-5-2012).pdf | 2018-08-09 |
| 46 | 2277-mumnp-2008-form 3(23-10-2008).pdf | 2008-10-23 |
| 46 | 2277-MUMNP-2008-CLAIMS(GRANTED).pdf | 2018-08-09 |
| 47 | 2277-mumnp-2008-claims(amended)-(4-11-2008).pdf | 2018-08-09 |
| 47 | 2277-mumnp-2008-form 5(23-10-2008).pdf | 2008-10-23 |
| 48 | 2277-MUMNP-2008-CLAIMS(AMENDED)-(15-5-2012).pdf | 2018-08-09 |
| 48 | 2277-mumnp-2008-wo international publication report(23-10-2008).pdf | 2008-10-23 |