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Methods For Protecting And Deprotecting Diol Group, And Diol Group Protective Agent
Abstract: An object of the present invention is to provide methods for protecting and deprotecting a diol group, and a protective agent for a diol group.
Notices, Deadlines & Correspondence
Patent Information
Applicants
FUJIFILM Corporation
Inventors
1. NAKAMURA, Koki
2. NAGASE, Hisato
3. FUJINO, Yuuta
4. WATANABE, Katsuyuki
5. KATSUMATA, Taiji
Claims
1. A method for protecting a 1,2-diol group or a 1,3-diol group, comprising reacting a 1,2-diol group or a 1,3-diol group with a group represented by Formula (19) in the presence of a base, (in the formula, Rla and Rlb are the same as or different from each other and each represent a hydrogen atom or a carboxy protective group; and * is a binding position).
2. A method for protecting a 1,2-diol group or a 1,3-diol group, comprising manufacturing a compound represented by Formula (21) by reacting a 1,2-diol group or a 1,3-diol group of a compound represented by Formula (20) with a compound represented by Formula (9) in the presence of a base, HO-Y1-OH (20) (in the formula, Y is a C2-3 alkylene group which may be substituted), (in the formula, each of Rla and Rlb are the same as or different from each other and each represent a hydrogen atom or a carboxy protective group; and R6 is a C1-6 alkyl group which may be substituted), and (in the formula, each of Rla, Rlb, and Y1 has the same definition as described above).
3. A method for deprotecting a protected 1,2-diol group or 1,3-diol group, comprising reacting a 1,2-diol group or a 1,3-diol group protected with a group represented by Formula (19) with a base, (in the formula, Rla and Rlb are the same as or different from each other and each represent a hydrogen atom or a carboxy protective group; and * is a binding position).
4. A method for deprotecting a protected 1,2-diol group or 1,3-diol group, comprising manufacturing a compound represented by Formula (20) by reacting a compound which is represented by Formula (21) and has a protected 1,2-diol group or a protected 1,3-diol group with a base, (in the formula, Rla and Rlb are the same as or different from each other and each represent a hydrogen atom or a carboxy protective group; and Y is a C2-3 alkylene group which may be substituted), and IH0-Y1«0H (20) (in the formula, Y1 has the same definition as described above).
Specification
WE CLAIM:
1. A method for protecting a 1,2-diol group or a 1,3-diol group, comprising reacting a 1,2-diol group or a 1,3-diol group with a group represented by Formula (19) in the presence of a base,
(in the formula, Rla and Rlb are the same as or different from each other and each represent a hydrogen atom or a carboxy protective group; and * is a binding position).
2. A method for protecting a 1,2-diol group or a 1,3-diol group, comprising manufacturing a compound represented by Formula (21) by reacting a 1,2-diol group or a 1,3-diol group of a compound represented by Formula (20) with a compound represented by Formula (9) in the presence of a base,
HO-Y1-OH (20) (in the formula, Y is a C2-3 alkylene group which may be substituted),
(in the formula, each of Rla and Rlb are the same as or different from each other and each represent a hydrogen atom or a carboxy protective group; and R6 is a C1-6 alkyl group which may be substituted), and
(in the formula, each of Rla, Rlb, and Y1 has the same definition as described above).
3. A method for deprotecting a protected 1,2-diol group or 1,3-diol group, comprising reacting a 1,2-diol group or a 1,3-diol group protected with a group represented by Formula (19) with a base,
(in the formula, Rla and Rlb are the same as or different from each other and each represent a hydrogen atom or a carboxy protective group; and * is a binding position).
4. A method for deprotecting a protected 1,2-diol group or 1,3-diol group, comprising manufacturing a compound represented by Formula (20) by reacting a compound which is represented by Formula (21) and has a protected 1,2-diol group or a protected 1,3-diol group with a base,
(in the formula, Rla and Rlb are the same as or different from each other and each represent a hydrogen atom or a carboxy protective group; and Y is a C2-3 alkylene group which may be substituted), and
IH0-Y1«0H (20)
(in the formula, Y1 has the same definition as described above).
Documents
Application Documents
| # | Name | Date |
|---|---|---|
| 1 | 201948005433-TRANSLATIOIN OF PRIOIRTY DOCUMENTS ETC. [12-02-2019(online)].pdf | 2019-02-12 |
| 2 | 201948005433-STATEMENT OF UNDERTAKING (FORM 3) [12-02-2019(online)].pdf | 2019-02-12 |
| 3 | 201948005433-REQUEST FOR EXAMINATION (FORM-18) [12-02-2019(online)].pdf | 2019-02-12 |
| 4 | 201948005433-POWER OF AUTHORITY [12-02-2019(online)].pdf | 2019-02-12 |
| 5 | 201948005433-FORM 18 [12-02-2019(online)].pdf | 2019-02-12 |
| 6 | 201948005433-FORM 1 [12-02-2019(online)].pdf | 2019-02-12 |
| 7 | 201948005433-FIGURE OF ABSTRACT [12-02-2019(online)].pdf | 2019-02-12 |
| 8 | 201948005433-DECLARATION OF INVENTORSHIP (FORM 5) [12-02-2019(online)].pdf | 2019-02-12 |
| 9 | 201948005433-COMPLETE SPECIFICATION [12-02-2019(online)].pdf | 2019-02-12 |
| 10 | 201948005433-CLAIMS UNDER RULE 1 (PROVISIO) OF RULE 20 [12-02-2019(online)].pdf | 2019-02-12 |
| 11 | Correspondence by Agent_Form1_05-08-2019.pdf | 2019-08-05 |
| 12 | 201948005433-Proof of Right (MANDATORY) [05-08-2019(online)].pdf | 2019-08-05 |
| 13 | 201948005433-FORM 3 [05-08-2019(online)].pdf | 2019-08-05 |
| 14 | 201948005433-FER.pdf | 2019-11-28 |
| 15 | 201948005433-FORM 3 [19-02-2020(online)].pdf | 2020-02-19 |
| 16 | 201948005433-FER_SER_REPLY [19-02-2020(online)].pdf | 2020-02-19 |
| 17 | 201948005433-US(14)-HearingNotice-(HearingDate-20-05-2020).pdf | 2020-04-24 |
| 18 | 201948005433-Correspondence to notify the Controller [15-05-2020(online)].pdf | 2020-05-15 |
| 19 | 201948005433-Written submissions and relevant documents [02-06-2020(online)].pdf | 2020-06-02 |
| 20 | 201948005433-Retyped Pages under Rule 14(1) [02-06-2020(online)].pdf | 2020-06-02 |
| 21 | 201948005433-2. Marked Copy under Rule 14(2) [02-06-2020(online)].pdf | 2020-06-02 |
| 22 | 201948005433-PatentCertificate26-06-2020.pdf | 2020-06-26 |
| 23 | 201948005433-Marked up Claims_Granted 339503_26-06-2020.pdf | 2020-06-26 |
| 24 | 201948005433-IntimationOfGrant26-06-2020.pdf | 2020-06-26 |
| 25 | 201948005433-Description_Granted 339503_26-06-2020.pdf | 2020-06-26 |
| 26 | 201948005433-Claims_Granted 339503_26-06-2020.pdf | 2020-06-26 |
| 27 | 201948005433-Abstract_Granted 339503_26-06-2020.pdf | 2020-06-26 |
| 28 | 201948005433-RELEVANT DOCUMENTS [14-09-2022(online)].pdf | 2022-09-14 |
| 29 | 201948005433-RELEVANT DOCUMENTS [16-09-2023(online)].pdf | 2023-09-16 |
Search Strategy
| 1 | ss_15-11-2019.pdf |