N (Heterrocyclyl) Benzene Or Pyridine Sulphonamides As Antithrombotic

N (Heterrocyclyl) Benzene Or Pyridine Sulphonamides As Antithrombotic And Anticoagulant Agents

Abstract: The invention concerns compounds of formula (I) wherein W can represent a -(CH¿2?)¿2?-, -(CH¿2?)-C$m(Z)C- or -CH¿2?-CH=CH- group; R¿2? can in particular represent a piperidinyl group, a 1,2,3,6-tetrahydropyridinyl group optionally substituted, a hexahydro-1(H)-azepinyl group, a piperazinyl group optionally substituted or a morphinopolinyl group; R¿3? can represent a -COR¿1? group; A can in particular represent a phenyl group optionally substituted, a heterocycle or a cyclopentyl group and B can in particular represent a pyridyl group, an aminopyrazinyl group, an aminopyridazinyl group, a pyrimidinyl group optionally substituted by an amino group, a piperidinyl group or an aminopyridinyl group optionally substituted on the pyridine by a (C¿1?-C¿4?) alkyl or (C¿1?-C¿4?) alkoxy group, the amino group capable of being optionally substituted by a (C¿1?-C¿4?) alkyl group. The invention also concerns the preparation of said compounds and their therapeutic use.

Patent Information

Application #

Filing Date

05 September 2002

Publication Number

26/2004

Publication Type

INA

Invention Field

GENERAL ENGINEERING

Status

Email

Parent Application

Applicants

SANOFI-SYNTHELABO

174 Avenue de F-75013 paris

Inventors

1. JEAN-MICHEL ALTENBURGER

7 AVENUE LES MOLIERES, F-78470 SAINT REMY-LES-CHEVEREUSE

2. GERARD CREMER

35 RUE DE SABLES, F-91420 MORANGIS

3. GILBERT LASSALLE

15 RUE DE LA CROIX VALENTIN, F-91470 LES MOLIERES

4. MOSTAFA MATROUGUI

24-26 IMPASSE DE LA CERISAIE, F-91120 PALAISEAU

Specification

NIL

Documents

Application Documents

#	Name	Date
1	in-pct-2002-01213-mum-wo international publication report(5-9-2002).pdf	2018-08-08
2	in-pct-2002-01213-mum-power of authority(8-11-2002).pdf	2018-08-08
3	in-pct-2002-01213-mum-form 3(5-9-2002).pdf	2018-08-08
4	in-pct-2002-01213-mum-form 19(2-4-2004).pdf	2018-08-08
5	in-pct-2002-01213-mum-form 1(5-9-2002).pdf	2018-08-08
6	in-pct-2002-01213-mum-description(complete)-(5-9-2002).pdf	2018-08-08
7	in-pct-2002-01213-mum-declaration(5-9-2002).pdf	2018-08-08
8	in-pct-2002-01213-mum-correspondence(ipo)-(11-2-2009).pdf	2018-08-08
9	in-pct-2002-01213-mum-correspondence(29-3-2004).pdf	2018-08-08
10	in-pct-2002-01213-mum-claims(complete)-(5-9-2002).pdf	2018-08-08