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Novel Form Of Irbesartan, Methods For Obtaining Said Form And Pharmaceutical Compositions Containing Same

Abstract: The invention concerns irbesartan form A having a modified crystalline habit such that length/width ratio ranges between 1:1 and 10:1, preferably between 1:1 and 5:1 and a method for preparing said crystalline habit. The method is characterised in that it consists in either subjecting a crystalline suspension of irbesartan form A having acicular habit to at least a temperature oscillating step, or in subjecting a crystalline suspension of irbesartan form A having acicular habit to a mechanical shearing. The invention also concerns a pharmaceutical composition containing said irbesartan crystalline habit.

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Notices, Deadlines & Correspondence

Patent Information

Application #
Filing Date
13 December 2000
Publication Number
26/2005
Publication Type
INA
Invention Field
PHARMACEUTICALS
Status
Email
Parent Application

Applicants

SANOFI-SYNTHELABO
174, avenue de France F-75013 Paris

Inventors

1. BRUNO FRANC
6, rue de l'Oratoire F-30650 Saze
2. CHRISTIAN HOFF
Mazet de l'Escoraille F-30126 Saint Laurent des Arbres
3. SAN KIANG
16 Highland Avenue Madison, New Jersey 07940
4. MARK D. LINDRUD
25 Ridgedale Avenue Madison, New Jersey 07940
5. OLIVIR MONNIER
20, route de Poussan F-34560 Villeveyrac
6. CHENKOU WEI
44 Windsor Drive Princeton Junction, New Jersey 08688

Specification

Documents

Application Documents

# Name Date
1 in-pct-2000-00727-mum-wo international publication report(13-12-2000).pdf 2000-12-13
2 in-pct-2000-00727-mum-form 3(13-12-2000).pdf 2000-12-13
3 in-pct-2000-00727-mum-form 1(13-12-2000).pdf 2000-12-13
4 in-pct-2000-00727-mum-drawing(13-12-2000).pdf 2000-12-13
5 in-pct-2000-00727-mum-description(complete)-(13-12-2000).pdf 2000-12-13
6 in-pct-2000-00727-mum-claims(13-12-2000).pdf 2000-12-13
7 in-pct-2000-00727-mum-power of authority(21-6-2001).pdf 2018-08-08
8 in-pct-2000-00727-mum-form 19(17-5-2004).pdf 2018-08-08
9 in-pct-2000-00727-mum-correspondence(ipo)-(6-8-2009).pdf 2018-08-08
10 in-pct-2000-00727-mum-correspondence 2(15-7-2009).pdf 2018-08-08
11 in-pct-2000-00727-mum-correspondence 1(17-5-2004).pdf 2018-08-08