“Novel Intermediate And Process Useful In The Preparation Of {2 [1

“Novel Intermediate And Process Useful In The Preparation Of {2 [1 (3,5 Bis Trifluoromethyl Benzyl) 5 Pyridin 4 Yl 1 H [1,2,3]Triazol 4 Yl] Pyridin 3 Yl} (2 Chlorophenyl) Methanone”

Abstract: The present invention relates to novel compounds, (2-chlorophenyl)-[2-(2-hydroxy-2-pyridin-4-yl-vinyl)pyridin-3-yl]methanone benzoate, and (2-chlorophenyl)-[2-(2-hydroxy-2-pyridin-4-yl-vinyl)pyridin-3-yl]methanone toluate, which are useful intermediates for the preparation of the compound of Formula I: (I) The present invention further relates to novel processes for preparing a crystalline compound, which is {2-[1-(3,5-bis-trifluoromethyl-benzyl)-5-pyridin-4-yl-1H-[1,2,3]triazol-4-yl]-pyridin-3-yl}-(2-chlorophenyl)-methanone, Form IV.

Patent Information

Application #

Filing Date

26 May 2009

Publication Number

24/2009

Publication Type

INA

Invention Field

CHEMICAL

Status

Email

Parent Application

Applicants

ELI LILLY AND COMPANY

Lilly Corporate Center City of Indianapolis State of Indiana United States of America.

Inventors

1. KOBIERSKI Michael Edward

3969 Shadow Hill Court Greenwood Indiana 46142 United States of America.

2. KOPACH Michael E.

843 Breaside Lane Greenwood Indiana 46143 United States of America.

3. CHEN Pingyun

105 Westchester Place Chapel Hill North Carolina 27514 United States of America.

Specification

PLEASE SEE THE SPECIFICATION ATTACHED.

Documents

Application Documents

#	Name	Date
1	1030-MUMNP-2009- PCT DOCUMENTS.pdf	2022-08-23
1	1030-MUMNP-2009-FORM 3(18-11-2009).pdf	2009-11-18
2	1030-MUMNP-2009-CORRESPONDENCE(18-11-2009).pdf	2009-11-18
2	1030-mumnp-2009-abstract(26-5-2009).pdf	2018-08-10
3	1030-mumnp-2009-assignment(15-6-2009).pdf	2018-08-10
4	1030-mumnp-2009-claims(complete)-(26-5-2009).pdf	2018-08-10
5	Form-1.pdf	2018-08-10
5	1030-mumnp-2009-correspondence(15-6-2009).pdf	2018-08-10
6	1030-MUMNP-2009_EXAMREPORT.pdf	2018-08-10
6	1030-MUMNP-2009-CORRESPONDENCE(28-5-2009).pdf	2018-08-10
7	1030-mumnp-2009-wo international publication report(26-5-2009).pdf	2018-08-10
7	1030-MUMNP-2009-CORRESPONDENCE(IPO)-(14-1-2013).pdf	2018-08-10
8	1030-mumnp-2009-form 5(26-5-2009).pdf	2018-08-10
8	1030-mumnp-2009-correspondence(ipo)-(26-5-2009).pdf	2018-08-10
9	1030-mumnp-2009-form 3(26-5-2009).pdf	2018-08-10
9	1030-mumnp-2009-description(complete)-(26-5-2009).pdf	2018-08-10
10	1030-mumnp-2009-form 1(26-5-2009).pdf	2018-08-10
10	1030-mumnp-2009-form 2(title page)-(complete)-(26-5-2009).pdf	2018-08-10
11	1030-MUMNP-2009-FORM 18(29-5-2009).pdf	2018-08-10
11	1030-mumnp-2009-form 2(complete)-(26-5-2009).pdf	2018-08-10
12	1030-MUMNP-2009-FORM 18(29-5-2009).pdf	2018-08-10
12	1030-mumnp-2009-form 2(complete)-(26-5-2009).pdf	2018-08-10
13	1030-mumnp-2009-form 1(26-5-2009).pdf	2018-08-10
13	1030-mumnp-2009-form 2(title page)-(complete)-(26-5-2009).pdf	2018-08-10
14	1030-mumnp-2009-description(complete)-(26-5-2009).pdf	2018-08-10
14	1030-mumnp-2009-form 3(26-5-2009).pdf	2018-08-10
15	1030-mumnp-2009-correspondence(ipo)-(26-5-2009).pdf	2018-08-10
15	1030-mumnp-2009-form 5(26-5-2009).pdf	2018-08-10
16	1030-MUMNP-2009-CORRESPONDENCE(IPO)-(14-1-2013).pdf	2018-08-10
16	1030-mumnp-2009-wo international publication report(26-5-2009).pdf	2018-08-10
17	1030-MUMNP-2009_EXAMREPORT.pdf	2018-08-10
17	1030-MUMNP-2009-CORRESPONDENCE(28-5-2009).pdf	2018-08-10
18	Form-1.pdf	2018-08-10
18	1030-mumnp-2009-correspondence(15-6-2009).pdf	2018-08-10
19	1030-mumnp-2009-claims(complete)-(26-5-2009).pdf	2018-08-10
20	1030-mumnp-2009-assignment(15-6-2009).pdf	2018-08-10
21	1030-MUMNP-2009-CORRESPONDENCE(18-11-2009).pdf	2009-11-18
21	1030-mumnp-2009-abstract(26-5-2009).pdf	2018-08-10
22	1030-MUMNP-2009-FORM 3(18-11-2009).pdf	2009-11-18
22	1030-MUMNP-2009- PCT DOCUMENTS.pdf	2022-08-23