“Novel Process For The Preparation Of Bilastine And Intermediates

“Novel Process For The Preparation Of Bilastine And Intermediates Thereof”

Abstract: ABSTRACT "NOVEL PROCESS FOR THE PREPARATION OF BILASTINE AND INTERMEDIATES THEREOF" The present invention relates to a novel process for the preparation of 2-[4-[2-[4- [1-(2-ethoxyethyl) benzimidazol-2-yl] piperidin-1-yl] ethyl] phenyl]-2-methyl propionic acid (I). It further relates to a process for the purification of Bilastine (I), is having purity greater than 99.0% by High performance liquid chromatography (HPLC).

Patent Information

Application #

Filing Date

19 August 2021

Publication Number

12/2023

Publication Type

INA

Invention Field

CHEMICAL

Status

Email

radha@biophore.com

Parent Application

Applicants

Biophore India pharmaceuticals Pvt. Ltd

Plot#92; 1-98/2/92, Kavuri Hills – Phase II, Jubilee Hills, Hyderabad, Telangana India-500033.

Biophore India pharmaceuticals Pvt. Ltd

Plot#92; 1-98/2/92, Kavuri Hills – Phase II, Jubilee Hills, Hyderabad, Telangana India-500033.

Inventors

1. Manik Reddy Pullagurla

Plot#92; 1-98/2/92, Kavuri Hills – Phase II, Jubilee Hills, Hyderabad, Telangana India-500033

2. Manik Reddy Pullagurla

Plot#92; 1-98/2/92, Kavuri Hills – Phase II, Jubilee Hills, Hyderabad, Telangana India-500033

3. Bhaskar Reddy Pitta

Plot#92; 1-98/2/92, Kavuri Hills – Phase II, Jubilee Hills, Hyderabad, Telangana India-500033.

4. Bhaskar Reddy Pitta

Plot#92; 1-98/2/92, Kavuri Hills – Phase II, Jubilee Hills, Hyderabad, Telangana India-500033.

5. Jagadeesh Babu Rangisetty

Plot#92; 1-98/2/92, Kavuri Hills – Phase II, Jubilee Hills, Hyderabad, Telangana India-500033.

6. Jagadeesh Babu Rangisetty

Plot#92; 1-98/2/92, Kavuri Hills – Phase II, Jubilee Hills, Hyderabad, Telangana India-500033.

Specification

DESC:Enclosed ,CLAIMS:Enclosed

Documents

Application Documents

#	Name	Date
1	202141037570-PROVISIONAL SPECIFICATION [19-08-2021(online)].pdf	2021-08-19
2	202141037570-FORM 1 [19-08-2021(online)].pdf	2021-08-19
3	202141037570-FORM 3 [19-08-2022(online)].pdf	2022-08-19
4	202141037570-ENDORSEMENT BY INVENTORS [19-08-2022(online)].pdf	2022-08-19
5	202141037570-COMPLETE SPECIFICATION [19-08-2022(online)].pdf	2022-08-19
6	202141037570-FORM 3 [07-12-2022(online)].pdf	2022-12-07
7	202141037570-Request Letter-Correspondence [18-01-2023(online)].pdf	2023-01-18
8	202141037570-Form 1 (Submitted on date of filing) [18-01-2023(online)].pdf	2023-01-18
9	202141037570-Covering Letter [18-01-2023(online)].pdf	2023-01-18
10	202141037570-Covering Letter [23-01-2023(online)].pdf	2023-01-23
11	202141037570-FORM 3 [23-07-2024(online)].pdf	2024-07-23
12	202141037570-FORM 18 [19-08-2025(online)].pdf	2025-08-19