Preparation Of N1 (2' Pyridyl) 1,2 Propanediamine Sulfamic Acid And

Preparation Of N1 (2' Pyridyl) 1,2 Propanediamine Sulfamic Acid And Its Use In The Synthesis Of Biologically Active Piperazines

A process for making an N1-(2’-pyridyl)-1,2-alkanediamine sulfamic acid of formula (II) by reacting a compound of formula (I) with NH2R’, wherein R and R’ are as defined in the specification. The invention also includes the compound of formula (II), and optical isomers thereof. The compound of formula (II) is an intermediate useful for making chiral piperazine derivatives which are active at the 5-HT1A receptor. (FIG. NIL).

Patent Information

Application #

Filing Date

10 September 2004

Publication Number

21/2006

Publication Type

Invention Field

CHEMICAL

Status

Email

Parent Application

Patent Number

Legal Status

Grant Date

2008-05-21

Renewal Date

Applicants

WYETH

FIVE GIRALDA FARMS, MADISON, USA.

Inventors

1. CHAN ANITA WAI-YIN

1600, CENTER AVENUE, AP0ARTMENT 6D FORT LEE USA.

2. FEIGELSON GREG BRIAN

ONE INDEPENDENCE LANE USA.

3. ZELDIS JOPSEPH

195 LONG CLOVE ROAD NEW CITY USA.

4. JIRKOVSKY IVO

P.O.BOX 1209 WAITSFIELD USA.

Specification

Documents

Application Documents

#	Name	Date
1	1336-kolnp-2004-granted-specification.pdf	2011-10-07
2	1336-kolnp-2004-granted-reply to examination report.pdf	2011-10-07
3	1336-kolnp-2004-granted-letter patent.pdf	2011-10-07
4	1336-kolnp-2004-granted-gpa.pdf	2011-10-07
5	1336-kolnp-2004-granted-form 5.pdf	2011-10-07
6	1336-kolnp-2004-granted-form 3.pdf	2011-10-07
7	1336-kolnp-2004-granted-form 18.pdf	2011-10-07
8	1336-kolnp-2004-granted-form 13.pdf	2011-10-07
9	1336-kolnp-2004-granted-form 1.pdf	2011-10-07
10	1336-kolnp-2004-granted-examination report.pdf	2011-10-07
11	1336-kolnp-2004-granted-description (complete).pdf	2011-10-07
12	1336-kolnp-2004-granted-correspondence.pdf	2011-10-07
13	1336-kolnp-2004-granted-claims.pdf	2011-10-07
14	1336-kolnp-2004-granted-assignment.pdf	2011-10-07
15	1336-kolnp-2004-granted-abstract.pdf	2011-10-07