Process For Preparation Of Cabozantinib

Abstract: The present invention provides for novel amorphous solid dispersions of form of cabozantinib malate, and a pharmaceutically acceptable excipient and process for the preparation of cabozantinib malate. The invention also provides a novel crystalline polymorph of cabozantinib.

Patent Information

Application #

Filing Date

17 October 2023

Publication Number

47/2023

Publication Type

INA

Invention Field

CHEMICAL

Status

Email

Parent Application

Applicants

BIOCON LIMITED

20th Km Hosur Road, Electronic City Post, Karnataka Bangalore 560100

Inventors

1. BHAT, Ramakrishna Parameshwar

Kadekodi, Po: Dhareshwar, Ta: Kumta, Dist: Uttara Kannada Karnataka 581327

2. KUMAR, Narasimman

27 A, Aishwarya layout, Yadavanahalli, Attibele, Karnataka Bangalore 562107

3. DEVAIAH, Venu Thirunelimada

522, 6th Cross, AECS Layout, Kudlu, Karnataka Bangalore 560068

4. PATEL, Pratik Rameshchandra

C-701, Purva Panorama, Kaleena Agrahara, Karnataka Bangalore 560076

5. NAIR, Ranjeet

A-203, Ajmera Stone Park, 1st Cross Road, Neeladri Nagar, Electronic City Phase 1, Karnataka Bangalore 560100

6. MATTI, Lankeswararao

Nagayalanka Mandal, Remalavaripalem, Krishna District Andhra Pradesh 521120

7. CHETTY, Jithendrababu Raghunadha

No.4-70, Gopannagaripalli, Yellankivaaripalli, Pulicherla Mandal, Chittoor District Andhra Pradesh 517172

Specification

Documents

Application Documents

#	Name	Date
1	202347070534-STATEMENT OF UNDERTAKING (FORM 3) [17-10-2023(online)].pdf	2023-10-17
2	202347070534-PRIORITY DOCUMENTS [17-10-2023(online)].pdf	2023-10-17
3	202347070534-FORM 1 [17-10-2023(online)].pdf	2023-10-17
4	202347070534-DRAWINGS [17-10-2023(online)].pdf	2023-10-17
5	202347070534-DECLARATION OF INVENTORSHIP (FORM 5) [17-10-2023(online)].pdf	2023-10-17
6	202347070534-COMPLETE SPECIFICATION [17-10-2023(online)].pdf	2023-10-17
7	202347070534-Proof of Right [04-12-2023(online)].pdf	2023-12-04
8	202347070534-FORM-26 [18-12-2023(online)].pdf	2023-12-18
9	202347070534-FORM 18 [30-01-2025(online)].pdf	2025-01-30