Process For Preparing 6 O Alkenyl Substituted Erythromycin Deriv

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Process For Preparing 6 O Alkenyl Substituted Erythromycin Deriv Atives

Abstract: In one aspect, the invention relates to a process for preparing 6-O-substituted erythromycin derivatives comprising reacting 2'-substituted and optionally 4'-substituted 9-oxime erythromycin derivatives with an alkylating agent in the presence of a palladium catalyst and phosphine. In another aspect, the invention relates to processes for preparing 6-O-substituted erythromycin ketolides using the palladium-catalyzed alkylation reaction.

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Notices, Deadlines & Correspondence

Patent Information

Application #

Filing Date

19 December 2001

Publication Number

36/2007

Publication Type

INA

Invention Field

CHEMICAL

Status

Parent Application

Applicants

ABBOTT LABORATORIES

D377/AP6D, 100 Abbott Park Road, Abbott Park, IL 60064-6050,

Inventors

1. STONER, Eric, J.

3934 Taft Road, Kenosha, WI 53142,

2. PETERSON, Matthew, J.

3 Packard Lane, Gurnee, IL 60031,

3. KU, Yi-Yin

493 Satinwood Terrace, Buffalo Grove, IL 60089,

4. CINK, Russell, D.

1447 Fairport Drive, Grayslake, IL 60030,

5. COOPER, Arthur, J.;

65 Wesley Avenue, Lake Villa, IL 60046,

6. DESHPANDE, Mahendra, N.

216 Saratoga Court, Gurnee, IL 60031

7. GRIEME, Tim

4899 North Hermitage, #1, Chicago, IL 60640,

8. HAIGHT, Anthony, R.

40381 Reed Court, Wadsworth, IL 60083,

9. HILL, David, R.

Congress Court, Gurnee, IL 60031,

10. HSU, Margaret, Chi-Ping

321 Southfield Drive, Vernon Hills, IL 60061,

11. KING, Steven, A.

16713 Orchard Valley Drive, Gurnee, IL 60031,

12. LEANNA, Marvin, R.

1025 Popes Creek Circle, Grayslake, IL 60030,

13. LEE, Elaine, C.

1041 Franklin Street, Mundelein, IL 60060,

14. MCLAUGHLIN, Maureen, A.

637 Hinman Avenue, Evanston, IL 60202,

15. MORTON, Howard, E.

6088 Indian Trail Road, Gurnee, IL 60031,

16. NAPIER, James, J.

1058 White Pine Drive, Antioch, IL 60002,

17. PLATA, Daniel, J.

14265 West Shelley Lane, Wadsworth, IL 60085,

18. RAJE, Prasad, S.

215 Thrush Circle, Lindenhurst, IL 60046,

19. RASMUSSEN, Michael

1256 Sheridan Road, Kenosha, WI 53140,

20. RILEY, David

5904 80th Place, Kenosha, WI 53142,

21. TIEN, Jien-Heh, J.

1287 North Maidstone Drive, Vernon Hills, IL 60061,

22. WITTENBERGER, Steven, J.

45 South Pershing Avenue, Mundelein, IL 60060,

Specification

Documents

Application Documents

#	Name	Date
1	in-pct-2001-01610-mum-wo international publication report(19-12-2001).pdf	2001-12-19
2	in-pct-2001-01610-mum-form 19(17-5-2004).pdf	2018-08-08
3	IN-PCT-2001-01610-MUM-CORRESPONDENCE(IPO).pdf	2018-08-08
4	in-pct-2001-01610-mum-correspondence(ipo)-(27-1-2010).pdf	2018-08-08
5	in-pct-2001-01610-mum-correspondence(10-5-2004).pdf	2018-08-08