Abstract: The present invention relates to a novel and industrially advantageous process for the preparation of 5-substsituted indole derivative, particularly it relates to process for the preparation of 5-bromo-3-[(R)-l-methyl-pyrrolidin-2-ylmethyl]-lH-indol of formula I, a key intermediate for the synthesis of eletriptan or pharmaceutically acceptable salts thereof, through novel keto carbamate intermediate of formula, wherein R is selected from hydrogen, alkyl, alkoxy, aryloxy, nitrile, nitro, halo
| # | Name | Date |
|---|---|---|
| 1 | 1469-del-2011-Correspondence Others-(14-03-2013).pdf | 2013-03-14 |
| 1 | Abstract.jpg | 2012-01-27 |
| 2 | 1469-del-2011-Form-3-(14-03-2013).pdf | 2013-03-14 |
| 2 | 1469-del-2011-Form-5.pdf | 2012-01-27 |
| 3 | 1469-del-2011-Form-3.pdf | 2012-01-27 |
| 3 | 1469-del-2011-Abstract.pdf | 2012-01-27 |
| 4 | 1469-del-2011-Form-2.pdf | 2012-01-27 |
| 4 | 1469-del-2011-Claims.pdf | 2012-01-27 |
| 5 | 1469-del-2011-Correspondence-others.pdf | 2012-01-27 |
| 5 | 1469-del-2011-Form-1.pdf | 2012-01-27 |
| 6 | 1469-del-2011-Description (Complete).pdf | 2012-01-27 |
| 7 | 1469-del-2011-Correspondence-others.pdf | 2012-01-27 |
| 7 | 1469-del-2011-Form-1.pdf | 2012-01-27 |
| 8 | 1469-del-2011-Claims.pdf | 2012-01-27 |
| 8 | 1469-del-2011-Form-2.pdf | 2012-01-27 |
| 9 | 1469-del-2011-Abstract.pdf | 2012-01-27 |
| 9 | 1469-del-2011-Form-3.pdf | 2012-01-27 |
| 10 | 1469-del-2011-Form-5.pdf | 2012-01-27 |
| 10 | 1469-del-2011-Form-3-(14-03-2013).pdf | 2013-03-14 |
| 11 | Abstract.jpg | 2012-01-27 |
| 11 | 1469-del-2011-Correspondence Others-(14-03-2013).pdf | 2013-03-14 |