Abstract: ABSTRACT "PURIFICATION METHOD FOR 1-[[N-METHYL-N-3- [(METHYLAMINO)ACETOXYMETHYL] PYRIDIN-2-YL] CARBAMOYLOXY] ETHYL- 1-[(2R,3R)-2-(2,5-DIFLUOROPHENYL)-2- HYDROXY-3-[4-(4-CYANOPHENYL) THIAZOL-2-YL] BUTYL]-1H- [1,2,4]-TRIAZO-4-IUMSULFATE" The present invention relates to a method for the purification of 1-[[N-methyl-N-3- [(methylamino)acetoxymethyl] pyridin-2-yl] carbamoyloxy] ethyl- 1-[(2R,3R)-2- (2,5-difluorophenyl)-2-hydroxy-3-[4-(4-cyanophenyl) thiazol-2-yl] butyl]-1H- [1,2,4]-triazo-4-iumsulfate (1) having purity greater than 99.5% by Highperformance liquid chromatography (HPLC).
DESC:Enclosed ,CLAIMS:Enclosed
| # | Name | Date |
|---|---|---|
| 1 | 202241059148-PROVISIONAL SPECIFICATION [17-10-2022(online)].pdf | 2022-10-17 |
| 2 | 202241059148-FORM 1 [17-10-2022(online)].pdf | 2022-10-17 |
| 3 | 202241059148-DRAWINGS [17-10-2022(online)].pdf | 2022-10-17 |
| 4 | 202241059148-FORM 3 [16-10-2023(online)].pdf | 2023-10-16 |
| 5 | 202241059148-ENDORSEMENT BY INVENTORS [16-10-2023(online)].pdf | 2023-10-16 |
| 6 | 202241059148-DRAWING [16-10-2023(online)].pdf | 2023-10-16 |
| 7 | 202241059148-COMPLETE SPECIFICATION [16-10-2023(online)].pdf | 2023-10-16 |