Pyridine 3 Carboxyamide Derivative
Abstract:
20172800Provided is a novel JAK3 inhibitor useful as a preventive and/or therapeutic agent for organ transplant rejection, graft versus host disease (GvHD), rheumatoid arthritis, multiple sclerosis, systemic lupus erythematosus, Sjogren’s syndrome, Behcet"s disease, type I diabetes mellitus, autoimmune thyroiditis, idiopathic thrombocytopenic purpura, ulcerative colitis, Crohn"s disease, asthma, allergic conjunctivitis, atopic dermatitis, contact dermatitis, urticaria, eczema, psoriasis, allergic conjunctivitis, uveitis, cancer, leukemia, etc. A pyridine-3-carboxyamide derivative represented by general formula (1) or a salt thereof or a solvate thereof.2600
Patent Information
Filing Date
24 January 2017
Publication Number
15/2017
Invention Field
PHARMACEUTICALS
Email
ipo@knspartners.com
Applicants
Country: Japan
3-6-29, Nishiki
Naka-ku
Nagoya-shi
Aichi
JP
4608625
Inventors
Country: Japan
1. KITAMURA, Takahiro
c/o Fuji Research Laboratories, KOWA COMPANY, LTD., 332-1, Oonoshinden, Fuji-shi, Shizuoka 4170845, Japan.
Country: Japan
2. YAMADA, Hajime
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
Country: Japan
3. TAKEMURA, Shunji
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan
Country: Japan
4. ASHIKAWA, Masanori
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
Country: Japan
5. ISHIKAWA, Tetsuya
c/o KOWA COMPANY, LTD., 3-4-14, Nihonbashi hon-cho, Chuo-ku, Tokyo 1038433, Japan.
Country: Japan
6. MIYAKE, Yoshiharu
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
Country: Japan
7. KOUKETSU, Akiyasu
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan
Country: Japan
8. SATO, Seiichi
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
Country: Japan
9. ISHIWATA, Hiroyuki
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
Country: Japan
10. TABUNOKI, Yuichiro
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
Country: Japan
11. SHIBASAKI, Manabu
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
Country: Japan
12. OZAWA, Takatoshi
c/o KOWA COMPANY, LTD., 3-4-14, Nihonbashi hon-cho, Chuo-ku, Tokyo 1038433, Japan.
Country: Japan
13. SHIGEMI, Ryota
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
Country: Japan
14. DOI, Takeshi
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
Country: Japan
15. TAMURA, Masahiro
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
ERegister / Renewals
Ceased
3rd: 28 Oct 2021
CBR 24791
Renewal 28/10/2021
Renewal Amount ₹4,000
Certificate #29165
From 27/11/2011 - To 27/11/2012
4th: 28 Oct 2021
CBR 24791
Renewal 28/10/2021
Renewal Amount ₹4,000
Certificate #29166
From 27/11/2012 - To 27/11/2013
5th: 28 Oct 2021
CBR 24791
Renewal 28/10/2021
Renewal Amount ₹4,000
Certificate #29167
From 27/11/2013 - To 27/11/2014
6th: 28 Oct 2021
CBR 24791
Renewal 28/10/2021
Renewal Amount ₹4,000
Certificate #29168
From 27/11/2014 - To 27/11/2015
7th: 28 Oct 2021
CBR 24791
Renewal 28/10/2021
Renewal Amount ₹12,000
Certificate #29169
From 27/11/2015 - To 27/11/2016
8th: 28 Oct 2021
CBR 24791
Renewal 28/10/2021
Renewal Amount ₹12,000
Certificate #29170
From 27/11/2016 - To 27/11/2017
9th: 28 Oct 2021
CBR 24791
Renewal 28/10/2021
Renewal Amount ₹12,000
Certificate #29171
From 27/11/2017 - To 27/11/2018
10th: 28 Oct 2021
CBR 24791
Renewal 28/10/2021
Renewal Amount ₹12,000
Certificate #29172
From 27/11/2018 - To 27/11/2019
11th: 28 Oct 2021
CBR 24791
Renewal 28/10/2021
Renewal Amount ₹24,000
Certificate #29173
From 27/11/2019 - To 27/11/2020
12th: 28 Oct 2021
CBR 24791
Renewal 28/10/2021
Renewal Amount ₹24,000
Certificate #29174
From 27/11/2020 - To 27/11/2021
13th: 28 Oct 2021
CBR 24791
Renewal 28/10/2021
Renewal Amount ₹24,000
Certificate #29175
From 27/11/2021 - To 27/11/2022
14th: 18 Oct 2022
CBR 27502
Renewal 18/10/2022
Renewal Amount ₹24,000
Certificate #29416
From 27/11/2022 - To 27/11/2023
15th: 09 Oct 2023
CBR 41186
Renewal 09/10/2023
Renewal Amount ₹24,000
Certificate #40493
From 27/11/2023 - To 27/11/2024