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Pyridine 3 Carboxyamide Derivative

Abstract: 20172800Provided is a novel JAK3 inhibitor useful as a preventive and/or therapeutic agent for organ transplant rejection, graft versus host disease (GvHD), rheumatoid arthritis, multiple sclerosis, systemic lupus erythematosus, Sjogren’s syndrome, Behcet"s disease, type I diabetes mellitus, autoimmune thyroiditis, idiopathic thrombocytopenic purpura, ulcerative colitis, Crohn"s disease, asthma, allergic conjunctivitis, atopic dermatitis, contact dermatitis, urticaria, eczema, psoriasis, allergic conjunctivitis, uveitis, cancer, leukemia, etc. A pyridine-3-carboxyamide derivative represented by general formula (1) or a salt thereof or a solvate thereof.2600

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Notices, Deadlines & Correspondence

Patent Information

Application #
Filing Date
24 January 2017
Publication Number
15/2017
Publication Type
INA
Invention Field
PHARMACEUTICALS
Status
Email
ipo@knspartners.com
Parent Application
Patent Number
Legal Status
Grant Date
2021-08-10
Renewal Date

Applicants

KOWA COMPANY, LTD.
3-6-29, Nishiki Naka-ku Nagoya-shi Aichi JP 4608625

Inventors

1. KITAMURA, Takahiro
c/o Fuji Research Laboratories, KOWA COMPANY, LTD., 332-1, Oonoshinden, Fuji-shi, Shizuoka 4170845, Japan.
2. YAMADA, Hajime
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
3. TAKEMURA, Shunji
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan
4. ASHIKAWA, Masanori
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
5. ISHIKAWA, Tetsuya
c/o KOWA COMPANY, LTD., 3-4-14, Nihonbashi hon-cho, Chuo-ku, Tokyo 1038433, Japan.
6. MIYAKE, Yoshiharu
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
7. KOUKETSU, Akiyasu
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan
8. SATO, Seiichi
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
9. ISHIWATA, Hiroyuki
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
10. TABUNOKI, Yuichiro
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
11. SHIBASAKI, Manabu
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
12. OZAWA, Takatoshi
c/o KOWA COMPANY, LTD., 3-4-14, Nihonbashi hon-cho, Chuo-ku, Tokyo 1038433, Japan.
13. SHIGEMI, Ryota
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
14. DOI, Takeshi
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.
15. TAMURA, Masahiro
c/o Tokyo New Drug Research Laboratories, KOWA COMPANY, LTD., 2-17-43, Noguchi-cho, Higashimurayama-shi, Tokyo 1890022, Japan.

Specification

Claims:PLEASE SEE ATTACHED , Description:PLEASE SEE ATTACHED

Documents

Application Documents

# Name Date
1 201728002600-RELEVANT DOCUMENTS [12-09-2023(online)].pdf 2023-09-12
1 Form 5 [24-01-2017(online)].pdf 2017-01-24
2 Form 3 [24-01-2017(online)].pdf 2017-01-24
2 201728002600-FER.pdf 2021-10-18
3 Description(Complete) [24-01-2017(online)].pdf_303.pdf 2017-01-24
3 201728002600-IntimationOfGrant10-08-2021.pdf 2021-08-10
4 Description(Complete) [24-01-2017(online)].pdf 2017-01-24
4 201728002600-PatentCertificate10-08-2021.pdf 2021-08-10
5 Other Patent Document [15-02-2017(online)].pdf 2017-02-15
5 201728002600-CLAIMS [30-07-2021(online)].pdf 2021-07-30
6 201728002600-ORIGINAL UNDER RULE 6(1A) -20-02-20170001.pdf 2017-02-20
6 201728002600-FER_SER_REPLY [30-07-2021(online)].pdf 2021-07-30
7 Form 26 [16-03-2017(online)].pdf 2017-03-16
7 201728002600-OTHERS [30-07-2021(online)].pdf 2021-07-30
8 201728002600-PETITION UNDER RULE 137 [30-07-2021(online)].pdf 2021-07-30
8 201728002600-ORIGINAL UNDER RULE 6 (1A)-23-03-2017.pdf 2017-03-23
9 Form 3 [24-04-2017(online)].pdf 2017-04-24
9 201728002600-FORM 4(ii) [01-05-2021(online)].pdf 2021-05-01
10 ABSTRACT1.jpg 2018-08-11
10 Other Patent Document [05-05-2017(online)].pdf 2017-05-05
11 201728002600-ORIGINAL UNDER RULE 6(1A)-11-05-2017.pdf 2017-05-11
11 Form 18 [05-07-2017(online)].pdf 2017-07-05
12 201728002600-ORIGINAL UNDER RULE 6(1A)-11-05-2017.pdf 2017-05-11
12 Form 18 [05-07-2017(online)].pdf 2017-07-05
13 ABSTRACT1.jpg 2018-08-11
13 Other Patent Document [05-05-2017(online)].pdf 2017-05-05
14 201728002600-FORM 4(ii) [01-05-2021(online)].pdf 2021-05-01
14 Form 3 [24-04-2017(online)].pdf 2017-04-24
15 201728002600-ORIGINAL UNDER RULE 6 (1A)-23-03-2017.pdf 2017-03-23
15 201728002600-PETITION UNDER RULE 137 [30-07-2021(online)].pdf 2021-07-30
16 201728002600-OTHERS [30-07-2021(online)].pdf 2021-07-30
16 Form 26 [16-03-2017(online)].pdf 2017-03-16
17 201728002600-FER_SER_REPLY [30-07-2021(online)].pdf 2021-07-30
17 201728002600-ORIGINAL UNDER RULE 6(1A) -20-02-20170001.pdf 2017-02-20
18 201728002600-CLAIMS [30-07-2021(online)].pdf 2021-07-30
18 Other Patent Document [15-02-2017(online)].pdf 2017-02-15
19 Description(Complete) [24-01-2017(online)].pdf 2017-01-24
19 201728002600-PatentCertificate10-08-2021.pdf 2021-08-10
20 Description(Complete) [24-01-2017(online)].pdf_303.pdf 2017-01-24
20 201728002600-IntimationOfGrant10-08-2021.pdf 2021-08-10
21 Form 3 [24-01-2017(online)].pdf 2017-01-24
21 201728002600-FER.pdf 2021-10-18
22 Form 5 [24-01-2017(online)].pdf 2017-01-24
22 201728002600-RELEVANT DOCUMENTS [12-09-2023(online)].pdf 2023-09-12

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