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“Pyridine 3 Carboxyamide Derivative”

Abstract: Provided is a novel JAK3 inhibitor useful as a preventive and/or therapeutic agent for organ transplant rejection, graft versus host disease (GvHD), rheumatoid arthritis, multiple sclerosis, systemic lupus erythematosus, Sjogren’s syndrome, Behcet""s disease, type I diabetes mellitus, autoimmune thyroiditis, idiopathic thrombocytopenic purpura, ulcerative colitis, Crohn""s disease, asthma, allergic conjunctivitis, atopic dermatitis, contact dermatitis, urticaria, eczema, psoriasis, allergic conjunctivitis, uveitis, cancer, leukemia, etc. A pyridine-3-carboxyamide derivative represented by general formula (1) or a salt thereof or a solvate thereof or a salt or a solvate thereof.

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Notices, Deadlines & Correspondence

Patent Information

Application #
Filing Date
24 June 2011
Publication Number
33/2012
Publication Type
INA
Invention Field
CHEMICAL
Status
Email
ipo@knspartners.com
Parent Application

Applicants

KOWA COMPANY  LTD.
3-6-29  Nishiki  Naka-ku  Nagoya-shi  Aichi 460-8625  Japan

Inventors

1. KITAMURA  Takahiro
c/o Fuji Research Laboratories  KOWA COMPANY  LTD.  332-1  Oonoshinden  Fuji-Shi  Shizuoka 417-0845  Japan
2. YAMADA  Hajime
c/o Tokyo New Drug Research Laboratories  KOWA COMPANY  LTD.  2-17-43  Noguchi-cho  Higashimurayama-shi  Tokyo 189-0022  Japan
3. TAKEMURA  Shunji
c/o Tokyo New Drug Research Laboratories  KOWA COMPANY  LTD.  2-17-43  Noguchi-cho  Higashimurayama-shi  Tokyo 189-0022  Japan
4. ASHIKAWA  Masanori
c/o Tokyo New Drug Research Laboratories  KOWA COMPANY  LTD.  2-17-43  Noguchi-cho  Higashimurayama-shi  Tokyo 189-0022  Japan
5. ISHIKAWA  Tetsuya
c/o KOWA COMPANY  LTD.  3-4-14  Nihonbashi hon-cho  Chuo-ku  Tokyo 103-8433  Japan
6. MIYAKE  Yoshiharu
c/o Tokyo New Drug Research Laboratories  KOWA COMPANY  LTD.  2-17-43  Noguchi-cho  Higashimurayama-shi  Tokyo 189-0022  Japan
7. KOUKETSU  Akiyasu
c/o Tokyo New Drug Research Laboratories  KOWA COMPANY  LTD.  2-17-43  Noguchi-cho  Higashimurayama-shi  Tokyo 189-0022  Japan
8. SATO  Seiichi
c/o Tokyo New Drug Research Laboratories  KOWA COMPANY  LTD.  2-17-43  Noguchi-cho  Higashimurayama-shi  Tokyo 189-0022  Japan
9. ISHIWATA  Hiroyuki
c/o Tokyo New Drug Research Laboratories  KOWA COMPANY  LTD.  2-17-43  Noguchi-cho  Higashimurayama-shi  Tokyo 189-0022  Japan
10. TABUNOKI  Yuichiro
c/o Tokyo New Drug Research Laboratories  KOWA COMPANY  LTD.  2-17-43  Noguchi-cho  Higashimurayama-shi  Tokyo 189-0022  Japan
11. SHIBASAKI  Manabu
c/o Tokyo New Drug Research Laboratories  KOWA COMPANY  LTD.  2-17-43  Noguchi-cho  Higashimurayama-shi  Tokyo 189-0022  Japan
12. OZAWA  Takatoshi
c/o KOWA COMPANY  LTD.  3-4-14  Nihonbashi hon-cho  Chuo-ku  Tokyo 103-8433  Japan
13. SHIGEMI  Ryota
c/o Tokyo New Drug Research Laboratories  KOWA COMPANY  LTD.  2-17-43  Noguchi-cho  Higashimurayama-shi  Tokyo 189-0022  Japan
14. DOI  Takeshi
c/o Tokyo New Drug Research Laboratories  KOWA COMPANY  LTD.  2-17-43  Noguchi-cho  Higashimurayama-shi  Tokyo 189-0022  Japan
15. TAMURA  Masahiro
c/o Tokyo New Drug Research Laboratories  KOWA COMPANY  LTD.  2-17-43  Noguchi-cho  Higashimurayama-shi  Tokyo 189-0022  Japan

Specification

PLEASE SEE THE SPECIFICATION ATTACHED

Documents

Orders

Section Controller Decision Date

Application Documents

# Name Date
1 1323-MUMNP-2011-Claims-261214.pdf 2018-08-10
1 1323-MUMNP-2011-WO INTERNATIONAL PUBLICATION REPORT A9(13-10-2011).pdf 2011-10-13
2 1323-MUMNP-2011-CORRESPONDENCE(1-7-2011).pdf 2018-08-10
2 1323-MUMNP-2011-PCT-IB-311(13-10-2011).pdf 2011-10-13
3 1323-MUMNP-2011-CORRESPONDENCE(13-9-2011).pdf 2018-08-10
3 1323-MUMNP-2011-CORRESPONDENCE(13-10-2011).pdf 2011-10-13
4 1323-MUMNP-2011-FORM 3(30-12-2011).pdf 2011-12-30
4 1323-MUMNP-2011-CORRESPONDENCE(15-1-2014).pdf 2018-08-10
5 1323-MUMNP-2011-CORRESPONDENCE(30-12-2011).pdf 2011-12-30
5 1323-MUMNP-2011-CORRESPONDENCE(29-1-2014).pdf 2018-08-10
6 1323-MUMNP-2011-CORRESPONDENCE(IPO)-(FER)-(29-04-2014).pdf 2014-04-29
6 1323-MUMNP-2011-CORRESPONDENCE(31-7-2012).pdf 2018-08-10
7 1323-MUMNP-2011-FORM 3(01-07-2014).pdf 2014-07-01
7 1323-MUMNP-2011-CORRESPONDENCE(8-5-2015).pdf 2018-08-10
8 1323-MUMNP-2011-Correspondence-030615.pdf 2018-08-10
8 1323-MUMNP-2011-CORRESPONDENCE(01-07-2014).pdf 2014-07-01
9 1323-MUMNP-2011-Correspondence-091216.pdf 2018-08-10
9 1323-MUMNP-2011-REPLY TO EXAMINATION REPORT(29-10-2014).pdf 2014-10-29
10 1323-MUMNP-2011-Correspondence-220216.pdf 2018-08-10
10 1323-MUMNP-2011-OTHER DOCUMENT(29-10-2014).pdf 2014-10-29
11 1323-MUMNP-2011-ENGLISH TRANSLATION(1-7-2011).pdf 2018-08-10
11 1323-MUMNP-2011-FORM 3(29-10-2014).pdf 2014-10-29
12 1323-MUMNP-2011-Examination Report Reply Recieved-261214.pdf 2018-08-10
12 Form 3 [23-05-2016(online)].pdf 2016-05-23
13 1323-MUMNP-2011-CORRESPONDENCE(IPO)-(HEARING NOTICE)-(20-10-2016).pdf 2016-10-20
13 1323-MUMNP-2011-FORM 1(31-7-2012).pdf 2018-08-10
14 1323-MUMNP-2011-FORM 13(31-7-2012).pdf 2018-08-10
14 HEARING ADJOURNMENT [28-10-2016(online)].pdf 2016-10-28
15 1323-MUMNP-2011-FORM 18(13-9-2011).pdf 2018-08-10
15 HEARING ADJOURNMENT [28-11-2016(online)].pdf 2016-11-28
16 1323-MUMNP-2011-FORM 3(15-1-2014).pdf 2018-08-10
16 Form 26 [01-12-2016(online)].pdf 2016-12-01
17 Other Patent Document [18-01-2017(online)].pdf 2017-01-18
17 1323-MUMNP-2011-FORM 3(29-1-2014).pdf 2018-08-10
18 1323-MUMNP-2011-Form 3-030615.pdf 2018-08-10
18 1323-MUMNP-2011-Written submissions and relevant documents (MANDATORY) [07-03-2018(online)].pdf 2018-03-07
19 1323-MUMNP-2011-Form 3-220216.pdf 2018-08-10
19 Petition .pdf 2018-08-10
20 1323-MUMNP-2011-Form 3-261214.pdf 2018-08-10
20 Form-5.pdf 2018-08-10
21 1323-MUMNP-2011-HearingNoticeLetter.pdf 2018-08-10
21 Form-3.pdf 2018-08-10
22 1323-MUMNP-2011-OTHERS-261214.pdf 2018-08-10
22 Form-1.pdf 2018-08-10
23 1323-MUMNP-2011-Power of Attorney-091216.pdf 2018-08-10
23 ABSTRACT1.JPG 2018-08-10
24 1323-MUMNP-2011_EXAMREPORT.pdf 2018-08-10
25 ABSTRACT1.JPG 2018-08-10
25 1323-MUMNP-2011-Power of Attorney-091216.pdf 2018-08-10
26 1323-MUMNP-2011-OTHERS-261214.pdf 2018-08-10
26 Form-1.pdf 2018-08-10
27 1323-MUMNP-2011-HearingNoticeLetter.pdf 2018-08-10
27 Form-3.pdf 2018-08-10
28 1323-MUMNP-2011-Form 3-261214.pdf 2018-08-10
28 Form-5.pdf 2018-08-10
29 1323-MUMNP-2011-Form 3-220216.pdf 2018-08-10
29 Petition .pdf 2018-08-10
30 1323-MUMNP-2011-Form 3-030615.pdf 2018-08-10
30 1323-MUMNP-2011-Written submissions and relevant documents (MANDATORY) [07-03-2018(online)].pdf 2018-03-07
31 1323-MUMNP-2011-FORM 3(29-1-2014).pdf 2018-08-10
31 Other Patent Document [18-01-2017(online)].pdf 2017-01-18
32 1323-MUMNP-2011-FORM 3(15-1-2014).pdf 2018-08-10
32 Form 26 [01-12-2016(online)].pdf 2016-12-01
33 1323-MUMNP-2011-FORM 18(13-9-2011).pdf 2018-08-10
33 HEARING ADJOURNMENT [28-11-2016(online)].pdf 2016-11-28
34 1323-MUMNP-2011-FORM 13(31-7-2012).pdf 2018-08-10
34 HEARING ADJOURNMENT [28-10-2016(online)].pdf 2016-10-28
35 1323-MUMNP-2011-CORRESPONDENCE(IPO)-(HEARING NOTICE)-(20-10-2016).pdf 2016-10-20
35 1323-MUMNP-2011-FORM 1(31-7-2012).pdf 2018-08-10
36 Form 3 [23-05-2016(online)].pdf 2016-05-23
36 1323-MUMNP-2011-Examination Report Reply Recieved-261214.pdf 2018-08-10
37 1323-MUMNP-2011-ENGLISH TRANSLATION(1-7-2011).pdf 2018-08-10
37 1323-MUMNP-2011-FORM 3(29-10-2014).pdf 2014-10-29
38 1323-MUMNP-2011-Correspondence-220216.pdf 2018-08-10
38 1323-MUMNP-2011-OTHER DOCUMENT(29-10-2014).pdf 2014-10-29
39 1323-MUMNP-2011-Correspondence-091216.pdf 2018-08-10
39 1323-MUMNP-2011-REPLY TO EXAMINATION REPORT(29-10-2014).pdf 2014-10-29
40 1323-MUMNP-2011-CORRESPONDENCE(01-07-2014).pdf 2014-07-01
40 1323-MUMNP-2011-Correspondence-030615.pdf 2018-08-10
41 1323-MUMNP-2011-CORRESPONDENCE(8-5-2015).pdf 2018-08-10
41 1323-MUMNP-2011-FORM 3(01-07-2014).pdf 2014-07-01
42 1323-MUMNP-2011-CORRESPONDENCE(IPO)-(FER)-(29-04-2014).pdf 2014-04-29
42 1323-MUMNP-2011-CORRESPONDENCE(31-7-2012).pdf 2018-08-10
43 1323-MUMNP-2011-CORRESPONDENCE(30-12-2011).pdf 2011-12-30
43 1323-MUMNP-2011-CORRESPONDENCE(29-1-2014).pdf 2018-08-10
44 1323-MUMNP-2011-FORM 3(30-12-2011).pdf 2011-12-30
44 1323-MUMNP-2011-CORRESPONDENCE(15-1-2014).pdf 2018-08-10
45 1323-MUMNP-2011-CORRESPONDENCE(13-9-2011).pdf 2018-08-10
45 1323-MUMNP-2011-CORRESPONDENCE(13-10-2011).pdf 2011-10-13
46 1323-MUMNP-2011-PCT-IB-311(13-10-2011).pdf 2011-10-13
46 1323-MUMNP-2011-CORRESPONDENCE(1-7-2011).pdf 2018-08-10
47 1323-MUMNP-2011-Claims-261214.pdf 2018-08-10
47 1323-MUMNP-2011-WO INTERNATIONAL PUBLICATION REPORT A9(13-10-2011).pdf 2011-10-13