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Substituted Carbinol Compound Having Cyclic Linker

Abstract: It is to provide a novel LXRß agonist that is useful as a preventative and/or therapeutic agent for atherosclerosis; arteriosclerosis such as those resulting from diabetes; dyslipidemia; hypercholesterolemia; lipid-related diseases; inflammatory diseases that are caused by inflammatory cytokines; skin diseases such as allergic skin diseases; diabetes; or Alzheimer's disease. It is a carbinol compound represented by the following general formula (I) or salt thereof, or their solvate.

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Notices, Deadlines & Correspondence

Patent Information

Application #
Filing Date
24 November 2010
Publication Number
09/2012
Publication Type
INA
Invention Field
CHEMICAL
Status
Email
Parent Application

Applicants

KOWA COMPANY, LTD.
6-29, NISHIKI 3-CHOME, NAKA-KU, NAGOYA-SHI, AICHI 4608625 JAPAN

Inventors

1. YAMAGUCHI, YUKI
C/O KOWA COMPANY, LTD., TOKYO NEW DRUG RESEARCH LABORATORIES, 2-17-43, NOGUCHI-CHO, HIGASHIMURAYAMA-SHI, TOKYO 189-0022, JAPAN
2. KOURA, MINORU
C/O KOWA COMPANY, LTD., TOKYO NEW DRUG RESEARCH LABORATORIES, 2-17-43, NOGUCHI-CHO, HIGASHIMURAYAMA-SHI, TOKYO 189-0022, JAPAN
3. KUROBUCHI, SAYAKA
C/O KOWA COMPANY, LTD., TOKYO NEW DRUG RESEARCH LABORATORIES, 2-17-43, NOGUCHI-CHO, HIGASHIMURAYAMA-SHI, TOKYO 189-0022, JAPAN
4. MATSUDA, TAKAYUKI
C/O KOWA COMPANY, LTD., TOKYO NEW DRUG RESEARCH LABORATORIES, 2-17-43, NOGUCHI-CHO, HIGASHIMURAYAMA-SHI, TOKYO 189-0022, JAPAN
5. OKUDA, AYUMU
C/O KOWA COMPANY, LTD., TOKYO NEW DRUG RESEARCH LABORATORIES, 2-17-43, NOGUCHI-CHO, HIGASHIMURAYAMA-SHI, TOKYO 189-0022, JAPAN
6. SUMIDA, HISASHI
C/O KOWA COMPANY, LTD., TOKYO NEW DRUG RESEARCH LABORATORIES, 2-17-43, NOGUCHI-CHO, HIGASHIMURAYAMA-SHI, TOKYO 189-0022, JAPAN
7. WATANABE, YUICHIRO
C/O KOWA COMPANY, LTD., TOKYO NEW DRUG RESEARCH LABORATORIES, 2-17-43, NOGUCHI-CHO, HIGASHIMURAYAMA-SHI, TOKYO 189-0022, JAPAN
8. ENOMOTO, TAKASHI
C/O KOWA COMPANY, LTD., TOKYO NEW DRUG RESEARCH LABORATORIES, 2-17-43, NOGUCHI-CHO, HIGASHIMURAYAMA-SHI, TOKYO 189-0022, JAPAN
9. SHIBUYA, KIMIYUKI
C/O KOWA COMPANY, LTD., TOKYO NEW DRUG RESEARCH LABORATORIES, 2-17-43, NOGUCHI-CHO, HIGASHIMURAYAMA-SHI, TOKYO 189-0022, JAPAN

Specification

Documents

Application Documents

# Name Date
1 8314-DELNP-2010-AbandonedLetter.pdf 2017-11-13
1 8314-DELNP-2010-GPA-(18-01-2011).pdf 2011-01-18
2 8314-DELNP-2010-FER.pdf 2017-02-03
2 8314-DELNP-2010-Form-1-(18-01-2011).pdf 2011-01-18
3 8314-delnp-2010-PCT-210.pdf 2015-10-07
3 8314-DELNP-2010-Correspondence-Others-(18-01-2011).pdf 2011-01-18
4 8314-delnp-2010-PCT-237.pdf 2015-10-07
4 8314-DELNP-2010-Correspondence-Others-(23-02-2011).pdf 2011-02-23
5 8314-delnp-2010-PCT-338.pdf 2015-10-07
5 8314-DELNP-2010-Form-3-(20-05-2011).pdf 2011-05-20
6 8314-delnp-2010-PCT-373.pdf 2015-10-07
6 8314-DELNP-2010-Correspondence-Others-(20-05-2011).pdf 2011-05-20
7 abstract.jpg 2011-08-20
7 8314-dekbo-2010-Correspondence Others-(17-05-2012).pdf 2012-05-17
8 8314-delnp-2010-form-5.pdf 2011-08-20
8 8314-dekbo-2010-Form-13-(17-05-2012).pdf 2012-05-17
9 8314-delnp-2010-Correspondence-Others-(27-04-2012).pdf 2012-04-27
9 8314-delnp-2010-form-3.pdf 2011-08-20
10 8314-delnp-2010-Form-18-(27-04-2012).pdf 2012-04-27
10 8314-delnp-2010-form-2.pdf 2011-08-20
11 8314-delnp-2010-abstract.pdf 2011-08-20
11 8314-delnp-2010-form-1.pdf 2011-08-20
12 8314-delnp-2010-claims.pdf 2011-08-20
12 8314-delnp-2010-description (complete).pdf 2011-08-20
13 8314-delnp-2010-correspondence-others.pdf 2011-08-20
14 8314-delnp-2010-claims.pdf 2011-08-20
14 8314-delnp-2010-description (complete).pdf 2011-08-20
15 8314-delnp-2010-abstract.pdf 2011-08-20
15 8314-delnp-2010-form-1.pdf 2011-08-20
16 8314-delnp-2010-Form-18-(27-04-2012).pdf 2012-04-27
16 8314-delnp-2010-form-2.pdf 2011-08-20
17 8314-delnp-2010-form-3.pdf 2011-08-20
17 8314-delnp-2010-Correspondence-Others-(27-04-2012).pdf 2012-04-27
18 8314-dekbo-2010-Form-13-(17-05-2012).pdf 2012-05-17
18 8314-delnp-2010-form-5.pdf 2011-08-20
19 abstract.jpg 2011-08-20
19 8314-dekbo-2010-Correspondence Others-(17-05-2012).pdf 2012-05-17
20 8314-delnp-2010-PCT-373.pdf 2015-10-07
20 8314-DELNP-2010-Correspondence-Others-(20-05-2011).pdf 2011-05-20
21 8314-delnp-2010-PCT-338.pdf 2015-10-07
21 8314-DELNP-2010-Form-3-(20-05-2011).pdf 2011-05-20
22 8314-delnp-2010-PCT-237.pdf 2015-10-07
22 8314-DELNP-2010-Correspondence-Others-(23-02-2011).pdf 2011-02-23
23 8314-delnp-2010-PCT-210.pdf 2015-10-07
23 8314-DELNP-2010-Correspondence-Others-(18-01-2011).pdf 2011-01-18
24 8314-DELNP-2010-Form-1-(18-01-2011).pdf 2011-01-18
24 8314-DELNP-2010-FER.pdf 2017-02-03
25 8314-DELNP-2010-AbandonedLetter.pdf 2017-11-13
25 8314-DELNP-2010-GPA-(18-01-2011).pdf 2011-01-18

Search Strategy

1 8314search_03-02-2017.pdf