Abstract: ABSTRACT The present invention relates to a novel process for the preparation of 5-[[[(2S)-2-amino-3-[4-(aminocarbonyl)-2,6-dimethylphenyl]-l-oxopropyl] [(lS)-l-(4-phenyl-lH-imidazol-2-yl) ethyl] amino] methyl]-2-methoxybenzoic acid (Eluxadoline (1) and its intermediates thereof.
soft copy attached in pdf
| # | Name | Date |
|---|---|---|
| 1 | 201941008476-PROVISIONAL SPECIFICATION [05-03-2019(online)].pdf | 2019-03-05 |
| 2 | 201941008476-FORM 1 [05-03-2019(online)].pdf | 2019-03-05 |
| 3 | Form-1_After Filing_14-03-2019.pdf | 2019-03-14 |
| 4 | Correspondence by Applicant_Form-1_14-03-2019.pdf | 2019-03-14 |
| 5 | 201941008476-FORM 3 [04-03-2020(online)].pdf | 2020-03-04 |
| 6 | 201941008476-ENDORSEMENT BY INVENTORS [04-03-2020(online)].pdf | 2020-03-04 |
| 7 | 201941008476-COMPLETE SPECIFICATION [04-03-2020(online)].pdf | 2020-03-04 |
| 8 | 201941008476-Abstract_04-03-2020.jpg | 2020-03-04 |
| 9 | 201941008476-Form5_After Filing_18-03-2020.pdf | 2020-03-18 |
| 10 | 201941008476-Form3_After Filing_18-03-2020.pdf | 2020-03-18 |
| 11 | 201941008476-Description Complete_After Filing_18-03-2020.pdf | 2020-03-18 |
| 12 | 201941008476-Correspondence_18-03-2020.pdf | 2020-03-18 |