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Tetrahydrocyclopenta[B] Indole Compounds As Androgen Receptor Modulators

Abstract: The present invention provides a compound of the formula: Formula (I) or a pharmaceutically acceptable salt thereof; pharmaceutical compositions comprising aa compound of Formula (I) in combination with a suitable carrier, diluent, or excipient; and methods for treating physiological disorders, particularly reduced bones mass, osteoporosis, osteopenia, or reduced muscle mass or strength, comprising administering a compound of Formula (I), or a pharmaceutically acceptable salt thereof. X-17142.

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Notices, Deadlines & Correspondence

Patent Information

Application #
Filing Date
13 April 2009
Publication Number
21/2009
Publication Type
INA
Invention Field
PHARMACEUTICALS
Status
Email
Parent Application
Patent Number
Legal Status
Grant Date
2012-04-27
Renewal Date

Applicants

ELI LILLY AND COMPANY
Lilly Corporate Center  City of Indianapolis  State of Indiana 46285  United States of America

Inventors

1. GAVARDINAS  Konstantinos
3642 Marie Court West  Monrovia  Indiana 46157  United States of America;
2. GREEN  Jonathan  Edward
7464 Glendale Drive  Avon  Indiana 46123  United States of America
3. JADHAV  Prabhakar  Kondaji
7422 Fox hollow Ridge  Zionsville  Indiana 46077  United States of America
4. MATTHEWS  Donald  Paul
7736 Wawasee Drive  Indianapolis  Indiana 46250  United States of America

Specification

PLEASE SEE THE SPECIFICATION ATTACHED.

Documents

Application Documents

# Name Date
1 702-MUMNP-2009-RELEVANT DOCUMENTS [14-09-2021(online)].pdf 2021-09-14
1 Form 27 [29-03-2016(online)].pdf 2016-03-29
2 702-MUMNP-2009-RELEVANT DOCUMENTS [16-01-2020(online)].pdf 2020-01-16
2 Form 27 [15-03-2017(online)].pdf 2017-03-15
3 702-MUMNP-2009-RELEVANT DOCUMENTS [17-01-2019(online)].pdf 2019-01-17
3 702-MUMNP-2009-RELEVANT DOCUMENTS [07-02-2018(online)].pdf 2018-02-07
4 ipindiaonline.gov.in_epatentfiling_online_frmPreview.asp.pdf 2018-08-10
4 702-MUMNP-2009-ABSTRACT(12-3-2012).pdf 2018-08-10
5 Form-5.pdf 2018-08-10
5 702-MUMNP-2009-ABSTRACT(16-4-2009).pdf 2018-08-10
6 Form-3.pdf 2018-08-10
6 702-MUMNP-2009-ABSTRACT(GRANTED)-(27-4-2012).pdf 2018-08-10
7 Form-1.pdf 2018-08-10
7 702-mumnp-2009-affidavit(14-5-2009).pdf 2018-08-10
8 702-MUMNP-2009_EXAMREPORT.pdf 2018-08-10
8 702-mumnp-2009-assignment(14-5-2009).pdf 2018-08-10
9 702-MUMNP-2009-CLAIMS(16-4-2009).pdf 2018-08-10
9 702-MUMNP-2009-WO INTERNATIONAL PUBLICATION REPORT A3(16-4-2009).pdf 2018-08-10
10 702-MUMNP-2009-CLAIMS(AMENDED)-(12-3-2012).pdf 2018-08-10
10 702-MUMNP-2009-US DOCUMENT(12-3-2012).pdf 2018-08-10
11 702-MUMNP-2009-CLAIMS(GRANTED)-(27-4-2012).pdf 2018-08-10
11 702-MUMNP-2009-SPECIFICATION(AMENDED)-(12-3-2012).pdf 2018-08-10
12 702-MUMNP-2009-CORRESPONDENCE(14-5-2009).pdf 2018-08-10
12 702-MUMNP-2009-REPLY TO EXAMINATION REPORT(12-3-2012).pdf 2018-08-10
13 702-MUMNP-2009-CORRESPONDENCE(16-4-2009).pdf 2018-08-10
13 702-MUMNP-2009-RECEIPT(IPO)-(16-4-2009).pdf 2018-08-10
14 702-MUMNP-2009-CORRESPONDENCE(20-8-2009).pdf 2018-08-10
14 702-MUMNP-2009-PETITION UNDER RULE-137(12-3-2012).pdf 2018-08-10
15 702-MUMNP-2009-CORRESPONDENCE(IPO)-(27-4-2012).pdf 2018-08-10
15 702-MUMNP-2009-PCT-REQUEST(16-4-2009).pdf 2018-08-10
16 702-MUMNP-2009-DESCRIPTION(COMPLETE)-(16-4-2009).pdf 2018-08-10
16 702-MUMNP-2009-PCT-ISA-220(16-4-2009).pdf 2018-08-10
17 702-MUMNP-2009-PCT-IPEA-401(16-4-2009).pdf 2018-08-10
17 702-MUMNP-2009-DESCRIPTION(GRANTED)-(27-4-2012).pdf 2018-08-10
18 702-MUMNP-2009-EP DOCUMENT(12-3-2012).pdf 2018-08-10
18 702-MUMNP-2009-PCT-IB-304(16-4-2009).pdf 2018-08-10
19 702-MUMNP-2009-FORM 1(12-3-2012).pdf 2018-08-10
19 702-MUMNP-2009-OTHER DOCUMENT(16-4-2009).pdf 2018-08-10
20 702-MUMNP-2009-FORM 1(16-4-2009).pdf 2018-08-10
20 702-MUMNP-2009-FORM 5(16-4-2009).pdf 2018-08-10
21 702-MUMNP-2009-FORM 18(16-4-2009).pdf 2018-08-10
21 702-MUMNP-2009-FORM 3(20-8-2009).pdf 2018-08-10
22 702-mumnp-2009-form 2(16-4-2009).pdf 2018-08-10
22 702-MUMNP-2009-FORM 3(16-4-2009).pdf 2018-08-10
23 702-MUMNP-2009-FORM 2(GRANTED)-(27-4-2012).pdf 2018-08-10
23 702-MUMNP-2009-FORM 3(12-3-2012).pdf 2018-08-10
24 702-MUMNP-2009-FORM 26(12-3-2012).pdf 2018-08-10
24 702-MUMNP-2009-FORM 2(TITLE PAGE)-(12-3-2012).pdf 2018-08-10
25 702-MUMNP-2009-FORM 2(TITLE PAGE)-(16-4-2009).pdf 2018-08-10
25 702-MUMNP-2009-FORM 2(TITLE PAGE)-(GRANTED)-(27-4-2012).pdf 2018-08-10
26 702-MUMNP-2009-FORM 2(TITLE PAGE)-(16-4-2009).pdf 2018-08-10
26 702-MUMNP-2009-FORM 2(TITLE PAGE)-(GRANTED)-(27-4-2012).pdf 2018-08-10
27 702-MUMNP-2009-FORM 2(TITLE PAGE)-(12-3-2012).pdf 2018-08-10
27 702-MUMNP-2009-FORM 26(12-3-2012).pdf 2018-08-10
28 702-MUMNP-2009-FORM 2(GRANTED)-(27-4-2012).pdf 2018-08-10
28 702-MUMNP-2009-FORM 3(12-3-2012).pdf 2018-08-10
29 702-mumnp-2009-form 2(16-4-2009).pdf 2018-08-10
29 702-MUMNP-2009-FORM 3(16-4-2009).pdf 2018-08-10
30 702-MUMNP-2009-FORM 18(16-4-2009).pdf 2018-08-10
30 702-MUMNP-2009-FORM 3(20-8-2009).pdf 2018-08-10
31 702-MUMNP-2009-FORM 1(16-4-2009).pdf 2018-08-10
31 702-MUMNP-2009-FORM 5(16-4-2009).pdf 2018-08-10
32 702-MUMNP-2009-FORM 1(12-3-2012).pdf 2018-08-10
32 702-MUMNP-2009-OTHER DOCUMENT(16-4-2009).pdf 2018-08-10
33 702-MUMNP-2009-EP DOCUMENT(12-3-2012).pdf 2018-08-10
33 702-MUMNP-2009-PCT-IB-304(16-4-2009).pdf 2018-08-10
34 702-MUMNP-2009-DESCRIPTION(GRANTED)-(27-4-2012).pdf 2018-08-10
34 702-MUMNP-2009-PCT-IPEA-401(16-4-2009).pdf 2018-08-10
35 702-MUMNP-2009-PCT-ISA-220(16-4-2009).pdf 2018-08-10
35 702-MUMNP-2009-DESCRIPTION(COMPLETE)-(16-4-2009).pdf 2018-08-10
36 702-MUMNP-2009-CORRESPONDENCE(IPO)-(27-4-2012).pdf 2018-08-10
36 702-MUMNP-2009-PCT-REQUEST(16-4-2009).pdf 2018-08-10
37 702-MUMNP-2009-CORRESPONDENCE(20-8-2009).pdf 2018-08-10
37 702-MUMNP-2009-PETITION UNDER RULE-137(12-3-2012).pdf 2018-08-10
38 702-MUMNP-2009-CORRESPONDENCE(16-4-2009).pdf 2018-08-10
38 702-MUMNP-2009-RECEIPT(IPO)-(16-4-2009).pdf 2018-08-10
39 702-MUMNP-2009-CORRESPONDENCE(14-5-2009).pdf 2018-08-10
39 702-MUMNP-2009-REPLY TO EXAMINATION REPORT(12-3-2012).pdf 2018-08-10
40 702-MUMNP-2009-CLAIMS(GRANTED)-(27-4-2012).pdf 2018-08-10
40 702-MUMNP-2009-SPECIFICATION(AMENDED)-(12-3-2012).pdf 2018-08-10
41 702-MUMNP-2009-CLAIMS(AMENDED)-(12-3-2012).pdf 2018-08-10
41 702-MUMNP-2009-US DOCUMENT(12-3-2012).pdf 2018-08-10
42 702-MUMNP-2009-CLAIMS(16-4-2009).pdf 2018-08-10
42 702-MUMNP-2009-WO INTERNATIONAL PUBLICATION REPORT A3(16-4-2009).pdf 2018-08-10
43 702-mumnp-2009-assignment(14-5-2009).pdf 2018-08-10
43 702-MUMNP-2009_EXAMREPORT.pdf 2018-08-10
44 702-mumnp-2009-affidavit(14-5-2009).pdf 2018-08-10
44 Form-1.pdf 2018-08-10
45 702-MUMNP-2009-ABSTRACT(GRANTED)-(27-4-2012).pdf 2018-08-10
45 Form-3.pdf 2018-08-10
46 Form-5.pdf 2018-08-10
46 702-MUMNP-2009-ABSTRACT(16-4-2009).pdf 2018-08-10
47 ipindiaonline.gov.in_epatentfiling_online_frmPreview.asp.pdf 2018-08-10
47 702-MUMNP-2009-ABSTRACT(12-3-2012).pdf 2018-08-10
48 702-MUMNP-2009-RELEVANT DOCUMENTS [17-01-2019(online)].pdf 2019-01-17
48 702-MUMNP-2009-RELEVANT DOCUMENTS [07-02-2018(online)].pdf 2018-02-07
49 Form 27 [15-03-2017(online)].pdf 2017-03-15
49 702-MUMNP-2009-RELEVANT DOCUMENTS [16-01-2020(online)].pdf 2020-01-16
50 702-MUMNP-2009-RELEVANT DOCUMENTS [14-09-2021(online)].pdf 2021-09-14

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3rd: 19 Jun 2012

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