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2 (1 2 3 Triazol 2 Yl)benzamide And 3 (1 2 3 Triazol 2 Yl)picolinamide Derivatives As Orexin Receptor Antagonists

Abstract: 115The present invention relates to 2 (1 2 3 triazol 2 yl)benzamide and 3 (1 2 3 triazol 2 yl)picolinamide derivatives of formula (I) Formula (I) wherein Ar Q and R to R are as described in the description to their preparation to pharmaceutically acceptable salts thereof and to their use as pharmaceuticals to pharmaceutical compositions containing one or more compounds of formula (I) and especially to their use as orexin receptor antagonists.

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Notices, Deadlines & Correspondence

Patent Information

Application #
Filing Date
03 June 2014
Publication Number
28/2015
Publication Type
INA
Invention Field
CHEMICAL
Status
Email
patent@depenning.com
Parent Application
Patent Number
Legal Status
Grant Date
2020-11-16
Renewal Date

Applicants

ACTELION PHARMACEUTICALS LTD
Gewerbestrasse 16 CH 4123 Allschwil

Inventors

1. BOLLI Martin
c/o Actelion Pharmaceuticals Ltd Gewerbestrasse 16 CH 4123 Allschwil
2. BOSS Christoph
c/o Actelion Pharmaceuticals Ltd Gewerbestrasse 16 CH 4123 Allschwil
3. BROTSCHI Christine
c/o Actelion Pharmaceuticals Ltd Gewerbestrasse 16 CH 4123 Allschwil
4. HEIDMANN Bibia
c/o Actelion Pharmaceuticals Ltd Gewerbestrasse 16 4123 Allschwil
5. SIFFERLEN Thierry
c/o Actelion Pharmaceuticals Ltd Gewerbestrasse 16 4123 Allschwil
6. WILLIAMS Jodi T.
c/o Actelion Pharmaceuticals Ltd Gewerbestrasse 16 CH 4123 Allschwil

Specification

Documents

Application Documents

# Name Date
1 4127-CHENP-2014-RELEVANT DOCUMENTS [17-05-2023(online)].pdf 2023-05-17
1 OTHERS.pdf 2014-06-09
2 4127-CHENP-2014-RELEVANT DOCUMENTS [25-09-2022(online)].pdf 2022-09-25
2 Form 5.pdf 2014-06-09
3 Form 3.pdf 2014-06-09
3 4127-CHENP-2014-IntimationOfGrant16-11-2020.pdf 2020-11-16
4 CLAIMS.pdf 2014-06-09
4 4127-CHENP-2014-PatentCertificate16-11-2020.pdf 2020-11-16
5 actelion pharmaceuticals ltd.pdf 2014-06-09
5 4127-CHENP-2014-FORM 3 [26-08-2020(online)].pdf 2020-08-26
6 4127-CHENP-2014.pdf 2014-07-10
6 4127-CHENP-2014-FORM 3 [20-02-2020(online)].pdf 2020-02-20
7 4127-CHENP-2014-FORM 3 [22-08-2019(online)].pdf 2019-08-22
7 4127-CHENP-2014 FORM-3 24-11-2014.pdf 2014-11-24
8 4127-CHENP-2014-FORM 3 [19-02-2019(online)].pdf 2019-02-19
8 4127-CHENP-2014 CORRESPONDENCE OTHERS 24-11-2014.pdf 2014-11-24
9 4127-CHENP-2014 FORM-3 07-05-2015.pdf 2015-05-07
9 4127-CHENP-2014-ABSTRACT [17-01-2019(online)].pdf 2019-01-17
10 4127-CHENP-2014 CORRESPONDENCE OTHERS 07-05-2015.pdf 2015-05-07
10 4127-CHENP-2014-CLAIMS [17-01-2019(online)].pdf 2019-01-17
11 4127-CHENP-2014 CORRESPONDENCE OTHERS 24-07-2015.pdf 2015-07-24
11 4127-CHENP-2014-FER_SER_REPLY [17-01-2019(online)].pdf 2019-01-17
12 4127-CHENP-2014 CORRESPONDENCE OTHERS 31-07-2015.pdf 2015-07-31
12 4127-CHENP-2014-FORM 3 [17-01-2019(online)].pdf 2019-01-17
13 4127-CHENP-2014-Form 3-220915.pdf 2015-11-30
13 4127-CHENP-2014-FORM-26 [17-01-2019(online)].pdf 2019-01-17
14 4127-CHENP-2014-Correspondence-220915.pdf 2015-11-30
14 4127-CHENP-2014-OTHERS [17-01-2019(online)].pdf 2019-01-17
15 4127-CHENP-2014-Form 3-080316.pdf 2016-07-12
15 4127-CHENP-2014-PETITION UNDER RULE 137 [17-01-2019(online)].pdf 2019-01-17
16 4127-CHENP-2014-Correspondence-F3-080316.pdf 2016-07-12
16 4127-CHENP-2014-FER.pdf 2018-07-19
17 Form 3 [06-09-2016(online)].pdf 2016-09-06
17 4127-CHENP-2014-FORM 3 [17-03-2018(online)].pdf 2018-03-17
18 4127-CHENP-2014-8(i)-Substitution-Change Of Applicant - Form 6 [15-11-2017(online)].pdf 2017-11-15
18 Form 3 [08-03-2017(online)].pdf 2017-03-08
19 4127-CHENP-2014-ASSIGNMENT DOCUMENTS [15-11-2017(online)].pdf 2017-11-15
19 4127-CHENP-2014-FORM 3 [11-09-2017(online)].pdf 2017-09-11
20 4127-CHENP-2014-PA [15-11-2017(online)].pdf 2017-11-15
21 4127-CHENP-2014-ASSIGNMENT DOCUMENTS [15-11-2017(online)].pdf 2017-11-15
21 4127-CHENP-2014-FORM 3 [11-09-2017(online)].pdf 2017-09-11
22 4127-CHENP-2014-8(i)-Substitution-Change Of Applicant - Form 6 [15-11-2017(online)].pdf 2017-11-15
22 Form 3 [08-03-2017(online)].pdf 2017-03-08
23 4127-CHENP-2014-FORM 3 [17-03-2018(online)].pdf 2018-03-17
23 Form 3 [06-09-2016(online)].pdf 2016-09-06
24 4127-CHENP-2014-FER.pdf 2018-07-19
24 4127-CHENP-2014-Correspondence-F3-080316.pdf 2016-07-12
25 4127-CHENP-2014-PETITION UNDER RULE 137 [17-01-2019(online)].pdf 2019-01-17
25 4127-CHENP-2014-Form 3-080316.pdf 2016-07-12
26 4127-CHENP-2014-Correspondence-220915.pdf 2015-11-30
26 4127-CHENP-2014-OTHERS [17-01-2019(online)].pdf 2019-01-17
27 4127-CHENP-2014-Form 3-220915.pdf 2015-11-30
27 4127-CHENP-2014-FORM-26 [17-01-2019(online)].pdf 2019-01-17
28 4127-CHENP-2014 CORRESPONDENCE OTHERS 31-07-2015.pdf 2015-07-31
28 4127-CHENP-2014-FORM 3 [17-01-2019(online)].pdf 2019-01-17
29 4127-CHENP-2014 CORRESPONDENCE OTHERS 24-07-2015.pdf 2015-07-24
29 4127-CHENP-2014-FER_SER_REPLY [17-01-2019(online)].pdf 2019-01-17
30 4127-CHENP-2014 CORRESPONDENCE OTHERS 07-05-2015.pdf 2015-05-07
30 4127-CHENP-2014-CLAIMS [17-01-2019(online)].pdf 2019-01-17
31 4127-CHENP-2014 FORM-3 07-05-2015.pdf 2015-05-07
31 4127-CHENP-2014-ABSTRACT [17-01-2019(online)].pdf 2019-01-17
32 4127-CHENP-2014 CORRESPONDENCE OTHERS 24-11-2014.pdf 2014-11-24
32 4127-CHENP-2014-FORM 3 [19-02-2019(online)].pdf 2019-02-19
33 4127-CHENP-2014 FORM-3 24-11-2014.pdf 2014-11-24
33 4127-CHENP-2014-FORM 3 [22-08-2019(online)].pdf 2019-08-22
34 4127-CHENP-2014-FORM 3 [20-02-2020(online)].pdf 2020-02-20
34 4127-CHENP-2014.pdf 2014-07-10
35 4127-CHENP-2014-FORM 3 [26-08-2020(online)].pdf 2020-08-26
35 actelion pharmaceuticals ltd.pdf 2014-06-09
36 4127-CHENP-2014-PatentCertificate16-11-2020.pdf 2020-11-16
36 CLAIMS.pdf 2014-06-09
37 Form 3.pdf 2014-06-09
37 4127-CHENP-2014-IntimationOfGrant16-11-2020.pdf 2020-11-16
38 Form 5.pdf 2014-06-09
38 4127-CHENP-2014-RELEVANT DOCUMENTS [25-09-2022(online)].pdf 2022-09-25
39 OTHERS.pdf 2014-06-09
39 4127-CHENP-2014-RELEVANT DOCUMENTS [17-05-2023(online)].pdf 2023-05-17

Search Strategy

1 ss_18-07-2018.pdf

ERegister / Renewals

3rd: 14 Dec 2020

From 07/11/2014 - To 07/11/2015

4th: 14 Dec 2020

From 07/11/2015 - To 07/11/2016

5th: 14 Dec 2020

From 07/11/2016 - To 07/11/2017

6th: 14 Dec 2020

From 07/11/2017 - To 07/11/2018

7th: 14 Dec 2020

From 07/11/2018 - To 07/11/2019

8th: 14 Dec 2020

From 07/11/2019 - To 07/11/2020

9th: 14 Dec 2020

From 07/11/2020 - To 07/11/2021

10th: 28 Oct 2021

From 07/11/2021 - To 07/11/2022

11th: 29 Oct 2022

From 07/11/2022 - To 07/11/2023