"Antibacterial 1 H Indazole And 1 H Indole Derivatives"

Abstract: 123AB221A2A3Atrans1BtranscisThe invention relates to antibacterial compounds of formula (I) wherein X is N or CH; R is H or halogen; R is alkynyloxy or the group M; R is H or halogen; M is one of the groups M and M represented below wherein A is a bond CHCH CH=CH or C=C; R is H or halogen; R is H alkoxy or halogen; R is H alkoxy hydroxyalkoxy alkoxyalkoxy thioalkoxy trifluoromethoxy amino hydroxyalkyl 2 hydroxyacetamido 1 aminocyclopropyl 1 hydroxymethyl cycloprop l yl l ((phosphonooxy)methyl)cyclopropyl l (((dimethylglycyl)oxy)methyl)cyclopropyl 2 hydroxymethyl cycloprop 1 yl 1 2 dihydroxy ethyl 3 hydroxyoxetan 3 yl 3 (hydroxyalkyl)oxetan 3 yl 3 aminooxetan 3 yl 3 hydroxythietan 3 yl morpholin 4 ylalkoxy morpholin 4 yl alkyl oxazol 2 yl or [l 2 3]triazol 2 yl; and R is hydroxyalkyl dihydroxyalkyl aminoalkyl 1 hydroxymethyl cycloprop 1 yl 1 aminomethyl cycloprop 1 yl iraws 2 hydroxymethyl cycloprop l yl 3 hydroxyoxetan 3 yl 3 hydroxythietan 3 yl 1 (2 hydroxyacetyl)azetidin 3 yl l (2 aminoacetyl)azetidin 3 yl l glycylazetidin 3 yl l (2 amino 2 methylpropanoyl)azetidin 3 yl 3 (2 aminoacetamido)cyclopentyl ( 3 4 dihydroxy) cyclopent 1 yl or 3 hydroxymethylbicyclo [1 1 1]pentan 1 yl; and salts thereof.

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