Abstract: ABSTRACT A PROCESS OF PREPARATION OF AN ANTIBACTERIAL COMPOUND AND ITS INTERMEDIATES THEREOF The present disclosure provides a process of preparation of an antibacterial compound of Formula I, (S)-6-(5-(((2-(7-fluoro-1-methyl-2-oxo-1,2-5 dihydroquinolin-8-yl) ethyl) amino) methyl)-2-oxooxazolidin-3-yl)-2H-pyrazino[2,3-b] [1,4] oxazin-3(4H)-one formate salt. The present disclosure also provides intermediates of the compound of Formula I and its preparation thereof. The present disclosure further provides a process of preparation of compound of Formula I with improved yield and high purity.
DESC:A PROCESS OF PREPARATION OF AN ANTIBACTERIAL COMPOUND AND ITS INTERMEDIATES THEREOF ,CLAIMS:AS ATTACHED
| # | Name | Date |
|---|---|---|
| 1 | 202341039331-STATEMENT OF UNDERTAKING (FORM 3) [08-06-2023(online)].pdf | 2023-06-08 |
| 2 | 202341039331-PROVISIONAL SPECIFICATION [08-06-2023(online)].pdf | 2023-06-08 |
| 3 | 202341039331-FORM FOR STARTUP [08-06-2023(online)].pdf | 2023-06-08 |
| 4 | 202341039331-FORM FOR SMALL ENTITY(FORM-28) [08-06-2023(online)].pdf | 2023-06-08 |
| 5 | 202341039331-FORM 1 [08-06-2023(online)].pdf | 2023-06-08 |
| 6 | 202341039331-EVIDENCE FOR REGISTRATION UNDER SSI(FORM-28) [08-06-2023(online)].pdf | 2023-06-08 |
| 7 | 202341039331-FORM-26 [10-08-2023(online)].pdf | 2023-08-10 |
| 8 | 202341039331-Proof of Right [15-11-2023(online)].pdf | 2023-11-15 |
| 9 | 202341039331-CORRESPONDENCE-OTHERS [07-06-2024(online)].pdf | 2024-06-07 |
| 10 | 202341039331-COMPLETE SPECIFICATION [07-06-2024(online)].pdf | 2024-06-07 |
| 11 | 202341039331-Request Letter-Correspondence [20-06-2024(online)].pdf | 2024-06-20 |
| 12 | 202341039331-Power of Attorney [20-06-2024(online)].pdf | 2024-06-20 |
| 13 | 202341039331-FORM28 [20-06-2024(online)].pdf | 2024-06-20 |
| 14 | 202341039331-Form 1 (Submitted on date of filing) [20-06-2024(online)].pdf | 2024-06-20 |
| 15 | 202341039331-Covering Letter [20-06-2024(online)].pdf | 2024-06-20 |
| 16 | 202341039331-CERTIFIED COPIES TRANSMISSION TO IB [20-06-2024(online)].pdf | 2024-06-20 |