"Heterocyclically Substituted Aryl Compounds As Hif Inhibitors"


Updated about 1 year ago

Abstract

The present application relates to novel aryl compounds with heterocyclic substituents, processes for their preparation, their use for treatment and/or prevention of diseases and their use for the preparation of medicaments for treatment and/or prevention of diseases, in particular for treatment and/or prevention of hyperproliferative and angiogenic diseases and those diseases which arise from metabolic adaptation to hypoxic states. Such treatments can be carried out as monotherapy or also in combination with other medicaments or further therapeutic measures.

Information

Application ID 3901/DELNP/2011
Invention Field CHEMICAL
Date of Application 2011-05-25
Publication Number 14/2012

Applicants

Name Address Country Nationality
BAYER SCHERING PHARMA AKTIENGESELLSCHAFT MULLERSTRASSE 178, 13353 BERLIN, GERMANY Germany Germany

Inventors

Name Address Country Nationality
MICHAEL HARTER ERNST-LUDWIG-KIRCHNER-STR. 56, 51375 LEVERKUSEN, GERMANY Germany Germany
HARTMUT BECK LOKOMOTIVSTR. 64, 50733 KOLN, GERMANY Germany Germany
PETER ELLINGHAUS AUF DER OBSTWIESE 3, 49324 MELLE, GERMANY Germany Germany
KERSTIN BERHOERSTER AM VOGELHERD 15, 45239 ESSEN, GERMANY Germany Germany
SUSANNE GRESCHAT IM COLLMOOR 6, 49419 WAGENFELD, GERMANY Germany Germany
KARL-HEINZ THIERAUCH HOCHWILDFAD 45, 14169 BERLIN, GERMANY Germany Germany
FRANK SUSSMEIER BAUBERGERSTR. 5, 80992 MUNCHEN, GERMANY Germany Germany

Specification

Documents

Name Date
3901-DELNP-2011-From-3-(08-11-2011).pdf 2011-11-08
3901-DELNP-2011-Correspondence-Others-(08-11-2011).pdf 2011-11-08
3901-delnp-2011-GPA.pdf 2012-02-02
3901-delnp-2011-Form-5.pdf 2012-02-02
3901-delnp-2011-Form-3.pdf 2012-02-02
3901-delnp-2011-Form-2.pdf 2012-02-02
3901-delnp-2011-Correspondence-others.pdf 2012-02-02
3901-delnp-2011-Form-1.pdf 2012-02-02
3901-delnp-2011-Abstract.pdf 2012-02-02
3901-delnp-2011-Form-3 (15-03-2012).pdf 2012-03-15
3901-delnp-2011-Claims.pdf 2012-02-02
3901-delnp-2011-Correspondence others-(15-03-2012).pdf 2012-03-15
3901-delnp-2011-Correspondence-Others-(20-07-2012).pdf 2012-07-20
3901-delnp-2011-Form-3-(20-07-2012).pdf 2012-07-20
3901-delnp-2011-Form 18-(05-11-2012).pdf 2012-11-05
3901-delnp-2011-Correspondence-Others-(05-11-2012).pdf 2012-11-05
3901-DELNP-2011-Form-3-(30-01-2013).pdf 2013-01-30
3901-DELNP-2011-Correspondence-Others-(30-01-2013).pdf 2013-01-30
3901-delnp-2011-GPA-(13-02-2013).pdf 2013-02-13
3901-delnp-2011-Form-2-(13-02-2013).pdf 2013-02-13
3901-delnp-2011-Description (Complete).pdf 2012-02-02
3901-delnp-2011-Correspondence Others-(13-02-2013).pdf 2013-02-13
3901-delnp-2011-Correspondence-Others-(18-02-2014).pdf 2014-02-18
3901-delnp-2011-Correspondence-Others-(12-08-2014).pdf 2014-08-12
3901-delnp-2011-Assignment-(13-02-2013).pdf 2013-02-13
3901-delnp-2011-Form-3-(18-02-2014).pdf 2014-02-18
3901-delnp-2011-Form-3-(12-08-2014).pdf 2014-08-12
3901-delnp-2011-Correspondance Others-(16-02-2015).pdf 2015-02-16
3901-delnp-2011-Form-3-(16-02-2015).pdf 2015-02-16
3901-DELNP-2011-FER.pdf 2017-06-14
3901-DELNP-2011-AbandonedLetter.pdf 2018-01-30
3901-DELNP-2011-From-3-(08-11-2011).pdf 2011-11-08
3901-delnp-2011-Form-1.pdf 2012-02-02
3901-delnp-2011-Abstract.pdf 2012-02-02
3901-delnp-2011-Form-5.pdf 2012-02-02
3901-DELNP-2011-Correspondence-Others-(08-11-2011).pdf 2011-11-08
3901-delnp-2011-Form-2.pdf 2012-02-02
3901-delnp-2011-Correspondence-Others-(20-07-2012).pdf 2012-07-20
3901-delnp-2011-Form-3.pdf 2012-02-02
3901-delnp-2011-Correspondence-others.pdf 2012-02-02
3901-delnp-2011-Form-2-(13-02-2013).pdf 2013-02-13
3901-delnp-2011-Form 18-(05-11-2012).pdf 2012-11-05
3901-delnp-2011-Correspondence others-(15-03-2012).pdf 2012-03-15
3901-delnp-2011-Form-3 (15-03-2012).pdf 2012-03-15
3901-delnp-2011-Correspondence-Others-(12-08-2014).pdf 2014-08-12
3901-delnp-2011-Correspondence-Others-(05-11-2012).pdf 2012-11-05
3901-delnp-2011-Assignment-(13-02-2013).pdf 2013-02-13
3901-delnp-2011-Claims.pdf 2012-02-02
3901-delnp-2011-Correspondence Others-(13-02-2013).pdf 2013-02-13
3901-DELNP-2011-Correspondence-Others-(30-01-2013).pdf 2013-01-30
3901-delnp-2011-Form-3-(12-08-2014).pdf 2014-08-12
3901-delnp-2011-GPA-(13-02-2013).pdf 2013-02-13
3901-DELNP-2011-Form-3-(30-01-2013).pdf 2013-01-30
3901-delnp-2011-Form-3-(18-02-2014).pdf 2014-02-18
3901-DELNP-2011-FER.pdf 2017-06-14
3901-delnp-2011-Form-3-(20-07-2012).pdf 2012-07-20
3901-DELNP-2011-AbandonedLetter.pdf 2018-01-30
3901-delnp-2011-Correspondence-Others-(18-02-2014).pdf 2014-02-18
3901-delnp-2011-Form-3-(16-02-2015).pdf 2015-02-16
3901-delnp-2011-GPA.pdf 2012-02-02
3901-delnp-2011-Correspondance Others-(16-02-2015).pdf 2015-02-16
3901-delnp-2011-Description (Complete).pdf 2012-02-02

Orders

Applicant Section Controller Decision Date URL